calcileap injection - Uses, Price, Side Effects & Substitutes
What is calcileap injection used for?
Calcirol 600000IU Injection (Calcitriol) is used to treat VITAMINS MINERALS NUTRIENTS. It contains Calcitriol (1mcg), which Calcitriol binds to vitamin D receptors (VDR) in target tissues, regulating calc. Always consult your doctor before use. Take as prescribed.
- Generic Name: Calcitriol
- Manufacturer: Genix Lifescience Pvt Ltd
- Form: Allopathy
- Pregnancy Category: C
- Prescription Required: Yes
๐ calcileap injection Uses & Benefits
Hypocalcemia due to chronic renal failure, hypoparathyroidism, osteoporosis, rickets, osteomalacia.
Off-label uses: Psoriasis, autoimmune diseases, secondary hyperparathyroidism.
๐ Drug Information
| Generic Name(s) | Calcitriol |
| Brand Name | Calcirol 600000IU Injection |
| Manufacturer | Genix Lifescience Pvt Ltd |
| Packaging / Form | Varies by brand (Allopathy) |
| Therapeutic Class | VITAMINS MINERALS NUTRIENTS |
| Action Class | Vitamins |
| Route of Administration | Intramuscular injection |
| Storage | Store at 20-25ยฐC; protect from light. |
| Shelf Life | As per manufacturer |
๐ฌ Pharmacology (PK/PD)
Pharmacokinetics
How It Works
Calcitriol binds to vitamin D receptors (VDR) in target tissues, regulating calcium and phosphate homeostasis by increasing intestinal absorption, renal reabsorption, and bone resorption.
Mechanism Steps
๐ก How to Take calcileap injection
Follow your doctor's prescription exactly.
โ ๏ธ Side Effects of calcileap injection
โ Common Side Effects
- Hypercalcemia
- Hypercalciuria
- Nausea
- Vomiting
- Constipation
- Headache
๐จ Serious Side Effects
- Arrhythmias
- Renal impairment
- Pancreatitis
- Psychiatric disturbances
โ ๏ธ Rare Side Effects
- Allergic reactions
- Metastatic calcification
Consult your doctor if you experience any unusual symptoms.
๐ฌ Drug Interactions
| โ ๏ธ Drug | Severity | Effect |
|---|---|---|
| Digitalis glycosides | Major | Increased risk of arrhythmias due to hypercalcemia. |
| Thiazide diuretics | Major | Increased risk of hypercalcemia. |
| Corticosteroids | Moderate | Reduced calcitriol efficacy. |
| Cholestyramine | Moderate | Reduced absorption of calcitriol. |
| Phenytoin | Moderate | Increased metabolism of calcitriol. |
| Barbiturates | Moderate | Increased metabolism of calcitriol. |
| Magnesium-containing antacids | Minor | Possible hypermagnesemia. |
| Calcium supplements | Minor | Increased risk of hypercalcemia. |
๐จ Major Interactions
- Digitalis glycosides
- Thiazide diuretics
โก Moderate Interactions
- Corticosteroids
- Cholestyramine
- Phenytoin
- Barbiturates
โน๏ธ Minor Interactions
- Magnesium-containing antacids
- Calcium supplements
๐ฝ๏ธ Food Interactions
High calcium intake may increase risk of hypercalcemia.
๐ท Alcohol Interaction
No significant interaction reported.
๐ก๏ธ Safety & Warnings
๐ซ Contraindications
Hypercalcemia, vitamin D toxicity, hypersensitivity to calcitriol.
๐ Monitoring Parameters
Serum calcium, phosphate, alkaline phosphatase, and parathyroid hormone levels; renal function.
๐คฑ Lactation Safety
Excreted in breast milk; caution advised.
๐ Overdose Management
Discontinue calcitriol; treat hypercalcemia with hydration, loop diuretics, corticosteroids, and calcitonin if severe.
โฐ Missed Dose
Administer as soon as remembered; do not double dose.
๐จโโ๏ธ Reviewed by Expert
๐ Substitutes for calcileap injection
View AllAlternative brands with exact same active ingredient (Calcitriol (1mcg)):
-
calcijet injectionLG Lifesciences โน120.58 6.5% CHEAPER
-
laretol 1mcg injectionLa Renon Healthcare Pvt Ltd โน138.00 7% COSTLIER
Medical Note: Always consult your doctor before switching medications.