graphyllin tablet - Etofylline (77mg) + Theophylline (23mg) medicine

Dericip 77mg/23mg Tablet: Complete Medicine Guide

No reviews yet
🏭 Gracure Pharmaceuticals Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 25, 2026
📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Evidence: Moderate
Reviewed by
SaathiMed Expert Panel | Sep 25, 2026

When to Call Your Doctor IMMEDIATELY

  • Severe nausea or vomiting
  • Irregular or rapid heartbeat
  • Seizures
  • Difficulty breathing or chest tightness
  • Severe headache with visual changes
  • Swelling of face, lips, or throat
  • Blood in vomit or stool

If experiencing severe symptoms, call emergency services immediately.

What is graphyllin tablet used for?

This medicine is a bronchodilator combination used to treat asthma and COPD. It works by relaxing airway muscles to make breathing easier. Take it exactly as prescribed, usually 2-3 times daily with food.

  • Generic Name: Etofylline (77mg) + Theophylline (23mg)
  • Manufacturer: Gracure Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 graphyllin tablet के बारे में (Hindi Summary)

उपयोग: यह दवा एटोफिलिन और थियोफिलिन का संयोजन है, जिसका उपयोग अस्थमा, क्रोनिक ब्रोंकाइटिस और सीओपीडी जैसी सांस की बीमारियों में किया जाता है। यह वायुमार्ग की मांसपेशियों को आराम देकर सांस लेने में मदद करती है। इसे डॉक्टर के निर्देशानुसार नियमित रूप से लें।

साइड इफेक्ट्स: आम दुष्प्रभावों में मतली, उल्टी, सिरदर्द, बेचैनी और दिल की धड़कन बढ़ना शामिल हैं। गंभीर दुष्प्रभाव दुर्लभ हैं लेकिन यदि दिल की धड़कन अनियमित हो, दौरा पड़े या सांस लेने में कठिनाई हो तो तुरंत डॉक्टर से मिलें।

सुरक्षा सलाह: इस दवा को डॉक्टर के बताए अनुसार ही लें। इसे चबाएं या तोड़ें नहीं। खाने के साथ लें। शराब और कैफीन से बचें। यदि आपको हृदय, यकृत या गुर्दे की समस्या है तो डॉक्टर को बताएं।

💡 Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

💊 graphyllin tablet Uses & Benefits

[{"condition":"Asthma","description":"Helps prevent and control asthma symptoms by relaxing airway muscles.","evidence":"Well-established"},{"condition":"Chronic bronchitis","description":"Used to relieve bronchospasm and improve breathing in chronic bronchitis.","evidence":"Well-established"},{"condition":"COPD","description":"May be used as a bronchodilator in chronic obstructive pulmonary disease.","evidence":"Moderate"}]

Off-label uses: [{"condition":"Apnea of prematurity","description":"Sometimes used off-label in premature infants, but not for this formulation.","evidence":"Limited"}]

Primary treatment for: Asthma

Also treats: Chronic bronchitis, COPD

📋 Drug Information

Generic Name(s)Etofylline (77mg) + Theophylline (23mg)
Brand Namegraphyllin tablet
ManufacturerGracure Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassRESPIRATORY
Action Class
Route of AdministrationOral
StorageStore at room temperature (15-30°C) in a dry place, away from direct sunlight. Keep in the original container.
Shelf Life24 months from the date of manufacture.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Take this medicine with food to reduce stomach upset.
2
Avoid caffeine and alcohol while taking this medicine.
3
Do not crush or chew the tablet; swallow it whole.
4
Take at the same times each day for best effect.
5
Inform your doctor if you have heart, liver, or kidney problems.
6
Do not use this medicine for sudden breathing attacks; use your rescue inhaler.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

✅
Wheezing
This medicine is commonly prescribed for this.
Likely Use
✅
Shortness of breath
This medicine helps relieve bronchospasm.
Likely Use
❌
Fever
This medicine is not a primary fever reducer.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionEtofylline and theophylline are well absorbed from the gastrointestinal tract after oral administration. The presence of food may affect the rate but not the extent of absorption.
DistributionBoth components are distributed widely throughout body fluids and tissues. They cross the placenta and are excreted in breast milk.
Protein BindingTheophylline is approximately 40% bound to plasma proteins; etofylline binding is not well established.
MetabolismTheophylline is metabolized in the liver by cytochrome P450 enzymes, primarily CYP1A2 and CYP3A4. Etofylline is also metabolized in the liver.
Half-LifeThe elimination half-life of theophylline varies widely (3-12 hours) depending on age, liver function, and other factors. Etofylline half-life is not well established.
ExcretionBoth drugs and their metabolites are excreted primarily in the urine.
BioavailabilityTheophylline oral bioavailability is approximately 96%. Etofylline bioavailability is not well established.
Onset of ActionBronchodilation occurs within 30 minutes to 2 hours after oral administration.
Peak Plasma TimePeak plasma concentrations are reached in about 1-2 hours for immediate-release formulations.
Duration of ActionBronchodilation lasts for approximately 6-8 hours.

How It Works

This medicine works by inhibiting phosphodiesterase enzymes, which leads to increased levels of cyclic AMP in bronchial smooth muscle cells. This causes relaxation of the muscles around the airways, resulting in bronchodilation. Additionally, it blocks adenosine receptors, which contributes to its bronchodilator and mild anti-inflammatory effects.

Mechanism Steps

1
Phosphodiesterase inhibition: This medicine inhibits phosphodiesterase enzymes, increasing cyclic AMP levels in smooth muscle cells.
2
Smooth muscle relaxation: Elevated cyclic AMP leads to relaxation of bronchial smooth muscle, widening the airways.
3
Adenosine receptor blockade: This medicine blocks adenosine receptors, preventing adenosine-induced bronchoconstriction.
4
Improved breathing: The combined effects result in easier breathing and reduced symptoms of asthma and COPD.

💡 How to Take graphyllin tablet

Strength: Each tablet contains etofylline 77 mg and theophylline 23 mg.

1Swallow the tablet whole with a glass of water.
2Do not crush, chew, or break the tablet.
3Take with food to reduce stomach upset.
4Take at the same times each day for best effect.
5If you miss a dose, follow the missed dose instructions.

Dosage Information

Adult DosageThe usual adult dose is one tablet taken orally two to three times daily, or as directed by your physician. Dosage may be adjusted based on clinical response and serum theophylline levels. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician.
Elderly DosageElderly patients may require lower doses due to reduced clearance. Dose must be individualized by a qualified clinician based on renal and hepatic function.
Renal ImpairmentUse with caution in renal impairment. Dose adjustment may be necessary. Consult your doctor.
Hepatic ImpairmentUse with caution in hepatic impairment. Dose reduction may be required. Consult your doctor.
Maximum Daily DoseThe maximum daily dose should not exceed 3 tablets (231 mg etofylline and 69 mg theophylline) unless otherwise directed by a physician. Individual dosing must be determined by a qualified clinician.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With food
Take with meals
Reduces stomach upset.
Caffeine
Avoid
May increase stimulant effects and side effects.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of graphyllin tablet

✅ Common Side Effects

Nausea (Common (5-10%))
Take with food to reduce nausea. If it persists, consult your doctor.
Headache (Common (5-10%))
Rest and stay hydrated. Consult doctor if severe.
Insomnia (Common (5-10%))
Avoid taking close to bedtime. Consult doctor if persistent.
Restlessness (Common (5-10%))
Usually temporary. Consult doctor if bothersome.
Increased heart rate (Common (5-10%))
Monitor pulse. If persistent or symptomatic, seek medical advice.

🚨 Serious Side Effects

Cardiac arrhythmias (Rare (<0.1%))
Seek immediate medical attention if you experience palpitations, dizziness, or fainting.
Seizures (Rare (<0.1%))
Call emergency services immediately if seizures occur.
Severe allergic reactions (Rare (<0.1%))
Seek emergency care if you develop rash, swelling, or difficulty breathing.

⚠️ Rare Side Effects

Hyperglycemia
Monitor blood sugar if diabetic. Consult doctor if levels rise.
Hypokalemia
Report muscle weakness or cramps to your doctor.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Ciprofloxacin Major
Propranolol Major
Phenytoin Moderate
Cimetidine Moderate
Erythromycin Moderate
Rifampicin Moderate
Oral contraceptives Moderate
Allopurinol Minor
Aminoglutethimide Minor
Ketoconazole Minor

🚨 Major Interactions

  • Ciprofloxacin
  • Propranolol

⚡ Moderate Interactions

  • Phenytoin
  • Cimetidine

🍷 Alcohol Interaction

Alcohol may increase the risk of side effects such as nausea, headache, and rapid heart rate. It is best to avoid alcohol while taking this medicine.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Hypersensitivity to etofylline, theophylline, or any component of the formulation","Active peptic ulcer disease","Uncontrolled seizure disorders","Severe cardiac arrhythmias","Acute porphyria"]

⚠️ Warnings & Precautions

["Use with caution in patients with heart disease, hypertension, or hyperthyroidism.","May impair ability to drive or operate machinery due to dizziness or restlessness.","Avoid excessive caffeine intake.","Do not exceed prescribed dose; toxicity can occur.","Use with caution in elderly patients and those with liver or kidney impairment.","Inform your doctor if you are pregnant, planning to become pregnant, or breastfeeding."]

🤱 Lactation Safety

This medicine passes into breast milk and may cause irritability or insomnia in the infant. Consult your doctor before breastfeeding.

💊 Overdose Management

Overdose can cause severe nausea, vomiting, seizures, and cardiac arrhythmias. Seek emergency medical attention immediately. Treatment is supportive and symptomatic; there is no specific antidote. Gastric lavage may be considered if recent ingestion. Monitor vital signs and electrolytes.

⏰ Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule. Do not double the dose to catch up.

Additional Safety Advice

General Safety

Take this medicine exactly as prescribed. Do not crush or chew the tablet; swallow it whole with water. Avoid alcohol and caffeine while taking this medicine as they can increase side effects. Inform your doctor if you have heart, liver, or kidney problems. Do not start or stop this medicine without consulting your doctor. Keep out of reach of children.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients may be more sensitive to the effects of this medicine and may require lower doses. Regular monitoring of heart rate and theophylline levels is advised.

🤰 Pregnancy Planning (TTC)

Consult your doctor if you are planning pregnancy. This medicine should be used during pregnancy only if clearly needed and prescribed by a doctor.

🏥 Post-Surgery Considerations

Inform your surgeon and anesthesiologist that you are taking this medicine. It may interact with anesthetic agents and affect heart rate.

🦷 Dental Procedures

Inform your dentist that you are taking this medicine. It may cause dry mouth or increase heart rate during dental procedures.

💚 Lifestyle Tips for Better Results

🏃
Avoid smoking and exposure to secondhand smoke.
🥗
Maintain a healthy weight to reduce breathing effort.
😴
Practice breathing exercises as advised by your doctor.
💧
Stay hydrated to keep airways moist.
🧘
Get adequate rest and manage stress.

🏋️ Exercise Considerations

Moderate exercise is generally safe, but avoid strenuous activity in cold or polluted air. Consult your doctor before starting any new exercise program.

🥗 Diet Recommendations

Eat a balanced diet rich in fruits and vegetables.
Limit caffeine intake.
Avoid heavy, high-fat meals close to dosing times.
Stay well hydrated.

💼 Impact on Daily Work & Life

This medicine may cause dizziness or restlessness in some people. Avoid driving or operating heavy machinery until you know how it affects you.

🛑 When to Stop This Medicine

Do not stop this medicine without consulting your doctor. If you experience severe side effects, seek medical advice immediately.

📅 Long-Term Use Effects

Long-term use may require periodic monitoring of theophylline levels, heart rate, and liver function. Tolerance to the bronchodilator effect is rare. Do not stop suddenly without consulting your doctor.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Inhaled corticosteroids

Can complement or be an alternative for asthma control.

Evidence: Well-established
Leukotriene receptor antagonists

Oral medications for asthma prophylaxis.

Evidence: Well-established

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

No specific vaccine interactions are established. However, consult your doctor about flu and pneumonia vaccines, which are recommended for people with chronic respiratory diseases.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate unless specified

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✈️ Traveling with This Medicine

Carry this medicine in its original packaging with a copy of your prescription. Store at room temperature and protect from direct sunlight. If traveling across time zones, adjust dosing times gradually as advised by your doctor. Check customs regulations for carrying prescription medicines.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 55-year-old man with chronic asthma
He was prescribed this medicine twice daily. After two weeks, his wheezing episodes decreased significantly. He learned to take it with breakfast and dinner to avoid stomach upset.
💡 Lesson: Consistent timing with meals improves tolerability and effectiveness.
👤 A 62-year-old woman with COPD
She started this medicine and noticed improved breathing during daily walks. She was advised to avoid caffeine, which helped reduce her palpitations.
💡 Lesson: Avoiding caffeine can minimize side effects like rapid heartbeat.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: This medicine usually starts working within 30 minutes to 2 hours after taking a dose.

Q: Can I take it with food?

A: Yes, taking it with food helps reduce stomach upset.

Q: What should I do if I miss a dose?

A: Take it as soon as you remember, but if it's almost time for your next dose, skip the missed dose and continue with your regular schedule.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?

🔄 Substitutes for graphyllin tablet

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: This medicine can be used as a rescue inhaler for sudden attacks.
    Fact: This medicine is for maintenance therapy, not for acute attacks. Use a rescue inhaler for sudden symptoms.
  • Myth: It is safe to take extra doses if breathing is difficult.
    Fact: Taking extra doses can cause serious side effects. Follow your doctor's instructions exactly.

🔄 Alternative Options

Generic Alternatives

  • Etofylline + Theophylline tablet

Brand Alternatives

  • Dericip 77mg/23mg tablet

📊 Comparison with Similar Medicines

[{"medicine":"Dericip 77mg/23mg tablet","composition":"Etofylline 77mg + Theophylline 23mg","onset":"30-60 minutes","duration":"6-8 hours"},{"medicine":"Theophylline 100mg tablet","composition":"Theophylline 100mg","onset":"30-60 minutes","duration":"6-8 hours"}]

😊 Was this information helpful?

Browse Medicines A-Z

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory