azunate l 480 mg/80 mg tablet - Artesunate (480mg) + Lumefantrine (80mg) medicine

azunate l 480 mg/80 mg tablet

4.8 (13 reviews)
๐Ÿญ Macleods Pharmaceuticals Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Aug 21, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Aug 21, 2026

What is azunate l 480 mg/80 mg tablet used for?

Azunate L 480 mg/80 mg Tablet (Artesunate + Lumefantrine) is used to treat ANTI MALARIALS. It contains Artesunate (480mg) + Lumefantrine (80mg), which Artesunate produces free radicals that damage parasite proteins; Lumefantrine in. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Artesunate + Lumefantrine
  • Manufacturer: Macleods Pharmaceuticals Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š azunate l 480 mg/80 mg tablet Uses & Benefits

Uncomplicated Plasmodium falciparum malaria, chloroquine-resistant malaria.

Off-label uses: Severe malaria (IV artesunate preferred), mixed infections.

๐Ÿ“‹ Drug Information

Generic Name(s)Artesunate + Lumefantrine
Brand NameAzunate L 480 mg/80 mg Tablet
ManufacturerMacleods Pharmaceuticals Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI MALARIALS
Action ClassAntimalarial
Route of AdministrationOral
StorageStore at 25ยฐC (77ยฐF); excursions permitted to 15-30ยฐC (59-86ยฐF). Protect from moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionArtesunate is rapidly absorbed; lumefantrine absorption is enhanced with food.
DistributionArtesunate widely distributed; lumefantrine highly protein-bound and distributed to tissues.
Protein BindingArtesunate: 93%; Lumefantrine: 99.7%
MetabolismArtesunate: hydrolyzed to dihydroartemisinin (active); Lumefantrine: metabolized by CYP3A4.
Half-LifeArtesunate: ~1 hour; Dihydroartemisinin: ~45 min; Lumefantrine: 4-6 days.
ExcretionArtesunate: urine and feces; Lumefantrine: primarily feces.
BioavailabilityArtesunate: high; Lumefantrine: variable, increased with fat.
Onset of ActionRapid (within hours)
Peak Plasma TimeArtesunate: 1-2 hours; Lumefantrine: 6-8 hours.
Duration of ActionLong (lumefantrine provides sustained effect)

How It Works

Artesunate produces free radicals that damage parasite proteins; Lumefantrine inhibits heme polymerization.

Mechanism Steps

1Artesunate is hydrolyzed to dihydroartemisinin (DHA).
2DHA reacts with heme iron, producing free radicals that damage parasite proteins and membranes.
3Lumefantrine inhibits ฮฒ-hematin formation, preventing heme detoxification.

๐Ÿ’ก How to Take azunate l 480 mg/80 mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of azunate l 480 mg/80 mg tablet

โœ… Common Side Effects

  • Headache
  • Nausea
  • Vomiting
  • Diarrhea
  • Abdominal pain
  • Cough

๐Ÿšจ Serious Side Effects

  • QT prolongation
  • Severe allergic reaction
  • Hemolytic anemia (artesunate)
  • Hepatotoxicity

โš ๏ธ Rare Side Effects

  • Seizures
  • Acute renal failure
  • Stevens-Johnson syndrome

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Rifampin Major Reduced lumefantrine levels
Ketoconazole Major Increased lumefantrine levels
Halofantrine Major Increased QT prolongation risk
Warfarin Moderate Increased INR
Oral contraceptives Moderate Reduced efficacy
Antacids Minor Reduced absorption

๐Ÿšจ Major Interactions

  • CYP3A4 inducers (rifampin, carbamazepine)
  • CYP3A4 inhibitors (ketoconazole, ritonavir)
  • Antimalarials with QT prolongation (halofantrine)

โšก Moderate Interactions

  • Anticoagulants (warfarin)
  • Oral contraceptives
  • Antiepileptics

โ„น๏ธ Minor Interactions

  • Antacids
  • Cimetidine

๐Ÿฝ๏ธ Food Interactions

Take with fatty food to enhance lumefantrine absorption.

๐Ÿท Alcohol Interaction

Avoid alcohol due to potential hepatotoxicity.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity, severe hepatic impairment, first trimester of pregnancy (unless no alternative).

๐Ÿ“Š Monitoring Parameters

Parasite count, ECG (QT interval), liver function, renal function.

๐Ÿคฑ Lactation Safety

Excreted in milk; use with caution.

๐Ÿ’Š Overdose Management

Symptomatic and supportive; monitor ECG and electrolytes.

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose. Do not double.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Last reviewed on: Aug 21, 2026

๐Ÿ”— View Profile

โญ User Reviews

Trusted Reviewer Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

Regular Customer Jul 10, 2026

Helpful and effective medicine as per my experience. Always consult a doctor.

Verified User Jul 10, 2026

Found this to be a helpful product. Good results.

Certified Buyer Jul 10, 2026

Effective and reliable. Worked as expected.

Regular Customer Jul 10, 2026

Found this to be a helpful product. Good results.

๐Ÿ˜Š Was this information helpful?

Browse Medicines A-Z

Search our extensive medical database alphabetically.

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory