azoprine 50mg tablet - Azathioprine (50mg) medicine

Azoprine 50mg Tablet - Uses, Price, Side Effects

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๐Ÿญ Vhb Life Sciences Inc ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is azoprine 50mg tablet used for?

Azoprine 50mg Tablet contains Azathioprine, an immunosuppressant that works by inhibiting DNA synthesis in rapidly dividing cells, thereby suppressing the immune system. It is primarily used to prevent organ transplant rejection and to treat autoimmune diseases such as rheumatoid arthritis and lupus.

  • Generic Name: Azathioprine
  • Manufacturer: Vhb Life Sciences Inc
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š azoprine 50mg tablet Uses & Benefits

Prevention of organ transplant rejection, rheumatoid arthritis, systemic lupus erythematosus, inflammatory bowel disease (Crohn's disease, ulcerative colitis), autoimmune hepatitis.

Off-label uses: Behรงet's disease, myasthenia gravis, pemphigus vulgaris, atopic dermatitis, multiple sclerosis.

๐Ÿ“‹ Drug Information

Generic Name(s)Azathioprine
Brand NameAzoran Tablet
ManufacturerVhb Life Sciences Inc
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI NEOPLASTICS
Action ClassImmunosuppressant- Purine analogs
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionWell absorbed orally, approximately 50% bioavailability.
DistributionDistributes widely into body tissues, including liver and kidneys.
Protein BindingApproximately 30% bound to plasma proteins.
MetabolismMetabolized in the liver to 6-mercaptopurine (active) and other metabolites via xanthine oxidase and TPMT.
Half-LifeApproximately 5 hours for azathioprine; 3-5 hours for 6-mercaptopurine.
ExcretionPrimarily renal excretion of metabolites; small amount unchanged in urine.
BioavailabilityApproximately 50% (oral).
Onset of ActionDelayed; clinical effects may take weeks to months.
Peak Plasma Time1-2 hours after oral administration.
Duration of ActionProlonged; effects persist for weeks after discontinuation.

How It Works

Azathioprine is a purine analog that inhibits DNA and RNA synthesis, suppressing immune cell proliferation.

Mechanism Steps

1Azathioprine is converted to 6-mercaptopurine (6-MP) in the liver.
26-MP is metabolized to 6-thioguanine nucleotides (6-TGNs) via hypoxanthine-guanine phosphoribosyltransferase (HGPRT).
36-TGNs incorporate into DNA and RNA, inhibiting purine synthesis.

๐Ÿ’ก How to Take azoprine 50mg tablet

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โœ… ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of azoprine 50mg tablet

โœ… Common Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Leukopenia
  • Anemia
  • Thrombocytopenia
  • Increased liver enzymes

๐Ÿšจ Serious Side Effects

  • Severe bone marrow suppression
  • Hepatotoxicity
  • Pancreatitis
  • Serious infections
  • Lymphoma
  • Skin cancer

โš ๏ธ Rare Side Effects

  • Pulmonary fibrosis
  • Venocclusive disease of liver
  • Alopecia
  • Rash
  • Arthralgia
  • Hypersensitivity reactions

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Major Increased bleeding risk
Allopurinol Major Increased azathioprine toxicity
Ribavirin Major Increased myelosuppression

๐Ÿšจ Major Interactions

  • Allopurinol
  • Warfarin
  • Ribavirin
  • Febuxostat
  • Co-trimoxazole

โšก Moderate Interactions

  • ACE inhibitors
  • Methotrexate
  • Cyclosporine
  • Infliximab
  • Mycophenolate

โ„น๏ธ Minor Interactions

  • Antacids
  • Oral contraceptives
  • Cimetidine
  • Furosemide
  • Indomethacin

๐Ÿฝ๏ธ Food Interactions

Grapefruit may increase levels; avoid.

๐Ÿท Alcohol Interaction

Alcohol may increase hepatotoxicity risk; avoid or limit.

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Moderate
Kidney
Low
Heart
Low
Pregnancy
Category A

๐Ÿšซ Contraindications

Hypersensitivity to azathioprine, severe infections, pregnancy (unless essential), lactation, severe bone marrow suppression.

๐Ÿ“Š Monitoring Parameters

Complete blood count (CBC), liver function tests (LFTs), renal function, TPMT genotype before therapy.

๐Ÿคฑ Lactation Safety

Not recommended; excreted in breast milk; may cause immunosuppression in infant.

๐Ÿ’Š Overdose Management

Induce vomiting or gastric lavage; monitor for myelosuppression; supportive care; consider hemodialysis.

โฐ Missed Dose

Take as soon as remembered unless near next dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for azoprine 50mg tablet

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Alternative brands with exact same active ingredient (Azathioprine (50mg)):

Medical Note: Always consult your doctor before switching medications.

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