ativak 500mg injection - Amikacin (500mg) medicine

Ativak 500mg Injection - Uses, Price, Side Effects

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๐Ÿญ H & Care Incorp ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is ativak 500mg injection used for?

Ativak 500mg Injection contains Amikacin, an aminoglycoside antibiotic used to treat serious bacterial infections such as septicemia, respiratory tract infections, urinary tract infections, and intra-abdominal infections. It works by binding to bacterial ribosomes, inhibiting protein synthesis, and causing bacterial cell death. It is typically administered intravenously or intramuscularly under medical supervision.

  • Generic Name: Amikacin
  • Manufacturer: H & Care Incorp
  • Form: Allopathy
  • Pregnancy Category: D
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India has the highest number of USFDA-compliant plants outside the USA.

๐Ÿ’Š ativak 500mg injection Uses & Benefits

Serious Gram-negative infections (sepsis, pneumonia, complicated UTI, intra-abdominal infections); adjunct in tuberculosis; neonatal sepsis.

Off-label uses: Brucellosis, Plague, Tularemia

๐Ÿ“‹ Drug Information

Generic Name(s)Amikacin
Brand NameAmikacin Sulphate 500mg Injection
ManufacturerH & Care Incorp
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassOPHTHAL
Action ClassAminoglycosides
Route of AdministrationIntramuscular, Intravenous
StorageStore at 20-25ยฐC; protect from light; do not freeze.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed after intramuscular injection; peak plasma concentrations achieved within 1 hour.
DistributionDistributes widely into extracellular fluids; high concentrations in urine, bile, and synovial fluid; crosses placenta; minimal penetration into cerebrospinal fluid unless meninges inflamed.
Protein Binding0-11%
MetabolismMinimal hepatic metabolism; primarily excreted unchanged.
Half-Life2-3 hours (normal renal function); up to 30-60 hours in renal impairment.
ExcretionRenal excretion (90-98% unchanged) via glomerular filtration.
Bioavailability100% (IM); not absorbed orally.
Onset of ActionRapid (within 1 hour for IM).
Peak Plasma Time1 hour (IM); end of infusion (IV).
Duration of Action8-12 hours (dose-dependent).

How It Works

Binds to 30S ribosomal subunit, causing misreading of mRNA and inhibition of protein synthesis.

Mechanism Steps

1Binds to 30S ribosomal subunit
2Interferes with initiation complex
3Causes misreading of mRNA codons

๐Ÿ’ก How to Take ativak 500mg injection

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โœ… ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of ativak 500mg injection

โœ… Common Side Effects

  • Nephrotoxicity
  • Ototoxicity (vestibular and cochlear)
  • Nausea
  • Vomiting
  • Rash

๐Ÿšจ Serious Side Effects

  • Acute renal failure
  • Irreversible hearing loss
  • Neuromuscular blockade
  • Anaphylaxis

โš ๏ธ Rare Side Effects

  • Superinfection
  • Clostridium difficile colitis
  • Hypomagnesemia

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Gentamicin Major Increased risk of nephrotoxicity and ototoxicity
Furosemide Major Increased risk of ototoxicity
Cisplatin Major Increased risk of nephrotoxicity and ototoxicity
Vancomycin Moderate Increased risk of nephrotoxicity
Neuromuscular blocking agents Moderate Enhanced neuromuscular blockade

๐Ÿšจ Major Interactions

  • Neuromuscular blocking agents
  • Other aminoglycosides
  • Cisplatin
  • Loop diuretics
  • Vancomycin

โšก Moderate Interactions

  • Penicillins (synergy)
  • Cephalosporins
  • NSAIDs
  • Methoxyflurane

โ„น๏ธ Minor Interactions

  • Dimercaprol
  • Indomethacin

๐Ÿฝ๏ธ Food Interactions

No significant food interactions.

๐Ÿท Alcohol Interaction

No known interaction.

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Moderate
Heart
Low
Pregnancy
Category D

๐Ÿšซ Contraindications

Hypersensitivity to amikacin or other aminoglycosides; myasthenia gravis; pre-existing severe renal impairment.

๐Ÿ“Š Monitoring Parameters

Renal function (serum creatinine, BUN), urine output, audiometry, serum drug levels (peak and trough).

๐Ÿคฑ Lactation Safety

Caution; small amounts excreted in breast milk; monitor infant for diarrhea, candidiasis.

๐Ÿ’Š Overdose Management

Supportive care; hemodialysis may enhance elimination; monitor renal function and hearing.

โฐ Missed Dose

Administer as soon as remembered; if near next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for ativak 500mg injection

View All

Alternative brands with exact same active ingredient (Amikacin (500mg)):

Medical Note: Always consult your doctor before switching medications.

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