apriglim-m 0.5 tablet sr - Glimepiride (0.5mg) + Metformin (500mg) medicine

Azulix 0.5 MF Tablet: Comprehensive Guide to Uses, Side Effects, and Safety

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🏭 Aprica Pharmaceuticals Pvt Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 20, 2026
📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Evidence: Well-established for the combination in type 2 diabetes.
Reviewed by
SaathiMed Expert Panel | Sep 20, 2026

When to Call Your Doctor IMMEDIATELY

  • Blood in stool or vomit
  • Severe abdominal pain
  • Chest pain or difficulty breathing
  • Severe headache with visual changes
  • Sudden swelling of face, lips, or throat
  • Yellowing of skin or eyes
  • Decreased urine output
  • Confusion or seizures

If experiencing severe symptoms, call emergency services immediately.

What is apriglim-m 0.5 tablet sr used for?

This medicine is a combination of Glimepiride and Metformin used to treat type 2 diabetes. It lowers blood sugar by increasing insulin release and improving insulin sensitivity. Take it with meals as prescribed.

  • Generic Name: Glimepiride + Metformin
  • Manufacturer: Aprica Pharmaceuticals Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 apriglim-m 0.5 tablet sr के बारे में (Hindi Summary)

उपयोग: यह दवा ग्लिमेपिराइड और मेटफॉर्मिन का संयोजन है, जिसका उपयोग टाइप 2 डायबिटीज में रक्त शर्करा को नियंत्रित करने के लिए किया जाता है। यह अग्न्याशय से इंसुलिन के स्राव को बढ़ाती है और शरीर की इंसुलिन के प्रति संवेदनशीलता को सुधारती है। यह दवा आहार और व्यायाम के साथ ली जानी चाहिए।

साइड इफेक्ट्स: इस दवा के सामान्य दुष्प्रभावों में हाइपोग्लाइसीमिया (कम रक्त शर्करा), मतली, दस्त, पेट में असुविधा और मुँह में धातु जैसा स्वाद शामिल हैं। गंभीर दुष्प्रभावों में लैक्टिक एसिडोसिस और गंभीर हाइपोग्लाइसीमिया शामिल हैं, जिनके लिए तत्काल चिकित्सा की आवश्यकता होती है।

सुरक्षा सलाह: इस दवा को अपने डॉक्टर के निर्देशानुसार भोजन के साथ लें। नियमित रूप से रक्त शर्करा की जांच करें। शराब का सेवन न करें क्योंकि इससे लैक्टिक एसिडोसिस और हाइपोग्लाइसीमिया का खतरा बढ़ सकता है। गुर्दे या यकृत की समस्या होने पर डॉक्टर को बताएं। हाइपोग्लाइसीमिया के लक्षणों के लिए तुरंत इलाज करें।

💡 Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

💊 apriglim-m 0.5 tablet sr Uses & Benefits

[{"condition":"Type 2 Diabetes Mellitus","description":"Used as an adjunct to diet and exercise to improve glycemic control in adults with type 2 diabetes who are not achieving adequate control on monotherapy.","evidence":"Well-established"}]

Off-label uses: []

Primary treatment for: Type 2 Diabetes Mellitus

Also treats: Obesity, Dyslipidemia, Hypertension

📋 Drug Information

Generic Name(s)Glimepiride + Metformin
Brand NameAmaryl M 1mg Tablet PR
ManufacturerAprica Pharmaceuticals Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI DIABETIC
Action ClassSulfonylurea + Biguanide
Route of AdministrationOral
StorageStore at room temperature (15-30°C) in a dry place, away from direct sunlight. Keep in the original container.
Shelf Life24 months from the date of manufacture.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Take this medicine with meals to reduce stomach upset and lower the risk of hypoglycemia.
2
Monitor your blood sugar regularly and keep a record to share with your doctor.
3
Carry a source of fast-acting sugar (like glucose tablets) at all times in case of hypoglycemia.
4
Avoid alcohol completely while on this medicine to prevent lactic acidosis.
5
Inform your doctor if you are scheduled for surgery or imaging tests with contrast dyes.
6
Report any unusual muscle pain, difficulty breathing, or extreme fatigue immediately.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

High blood sugar
This medicine is commonly prescribed for this.
Likely Use
Fever
This medicine is not a primary fever reducer.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionGlimepiride is rapidly and completely absorbed after oral administration. Metformin is slowly and incompletely absorbed from the gastrointestinal tract, with bioavailability of about 50-60%.
DistributionGlimepiride is widely distributed in the body, with a volume of distribution of about 8.8 L. Metformin is rapidly distributed to various tissues, including the gastrointestinal tract, liver, and kidneys, with a volume of distribution of 63-276 L.
Protein BindingGlimepiride is more than 99% bound to plasma proteins. Metformin is negligibly bound to plasma proteins.
MetabolismGlimepiride is extensively metabolized in the liver by cytochrome P450 2C9 to a cyclohexyl hydroxyl methyl derivative (M1) and a carboxyl derivative (M2). Metformin is not metabolized in the body.
Half-LifeThe elimination half-life of Glimepiride is approximately 5-8 hours. Metformin has a plasma elimination half-life of approximately 6.5 hours.
ExcretionGlimepiride is excreted primarily in urine (about 60%) and feces (about 40%) as metabolites. Metformin is excreted unchanged in the urine by active tubular secretion.
BioavailabilityGlimepiride has a bioavailability of approximately 100%. Metformin has an absolute bioavailability of about 50-60%.
Onset of ActionThe blood glucose-lowering effect of Glimepiride begins within 1-2 hours after oral administration. Metformin's effect on glucose control develops over several days to weeks.
Peak Plasma TimeGlimepiride reaches peak plasma concentrations 2-3 hours after oral administration. Metformin reaches peak plasma concentrations in 2-3 hours.
Duration of ActionThe glucose-lowering effect of Glimepiride lasts up to 24 hours. Metformin's effect is sustained with continued dosing.

How It Works

This medicine combines two antidiabetic agents with complementary mechanisms. Glimepiride, a sulfonylurea, binds to ATP-sensitive potassium channels on pancreatic beta cells, causing depolarization and increased insulin secretion. Metformin, a biguanide, decreases hepatic glucose production, reduces intestinal absorption of glucose, and improves insulin sensitivity by increasing peripheral glucose uptake and utilization.

Mechanism Steps

1
Glimepiride binding: Glimepiride binds to the sulfonylurea receptor on pancreatic beta cells, closing ATP-sensitive potassium channels.
2
Beta cell depolarization: Closure of potassium channels leads to depolarization of the beta cell membrane.
3
Calcium influx and insulin release: Depolarization opens voltage-gated calcium channels, increasing intracellular calcium and triggering insulin secretion.
4
Metformin action on liver: Metformin reduces hepatic glucose production by inhibiting gluconeogenesis and glycogenolysis.
5
Metformin action on peripheral tissues: Metformin improves insulin sensitivity, increasing glucose uptake and utilization in skeletal muscle and adipose tissue.

💡 How to Take apriglim-m 0.5 tablet sr

Strength: Glimepiride 0.5 mg and Metformin 500 mg immediate-release tablet.

1Take this medicine orally with a meal to reduce stomach upset.
2Swallow the tablet whole with a glass of water.
3Do not crush, chew, or break the tablet.
4Take at the same time each day to maintain consistent blood levels.
5Follow your doctor's instructions regarding dose and frequency.

Dosage Information

Adult DosageThe usual starting dose is one tablet of Glimepiride 0.5 mg and Metformin 500 mg once daily with a meal. The dose may be increased gradually based on blood glucose levels, up to a maximum of Glimepiride 8 mg and Metformin 2000 mg per day. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician.
Elderly DosageElderly patients are at increased risk of hypoglycemia. Start with the lowest effective dose and monitor renal function closely. Dose must be individualized by a qualified clinician.
Renal ImpairmentUse is contraindicated in severe renal impairment (eGFR <30 mL/min/1.73 m²). In mild to moderate renal impairment, dose adjustment may be needed based on eGFR. Consult a clinician for individualized dosing.
Hepatic ImpairmentUse with caution in patients with hepatic impairment. Dose adjustment may be necessary. Consult a clinician for individualized dosing.
Maximum Daily DoseGlimepiride 8 mg and Metformin 2000 mg per day.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With meals
Take with meals
Reduces stomach upset and lowers hypoglycemia risk.
Alcohol
Avoid
Increases risk of lactic acidosis and hypoglycemia.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of apriglim-m 0.5 tablet sr

✅ Common Side Effects

Hypoglycemia (Common (5-10%))
Consume fast-acting sugar if symptoms occur. Adjust dose if recurrent.
Nausea (Common (5-10%))
Take with food. Usually resolves with continued use.
Diarrhea (Common (5-10%))
Stay hydrated. Consult doctor if persistent.
Abdominal discomfort (Common (5-10%))
Take with meals. Report if severe.
Metallic taste (Common (5-10%))
Usually temporary. Chewing sugar-free gum may help.

🚨 Serious Side Effects

Lactic acidosis (Rare (<0.1%))
Seek immediate medical attention if you experience muscle pain, difficulty breathing, stomach discomfort, or extreme fatigue.
Severe hypoglycemia (Uncommon (0.1-1%))
Seek emergency care if you have confusion, seizures, or loss of consciousness.
Hemolytic anemia (Rare (<0.1%))
Report unusual tiredness, pale skin, or jaundice to your doctor immediately.
Severe allergic reaction (Rare (<0.1%))
Seek emergency help if you develop rash, swelling, or difficulty breathing.

⚠️ Rare Side Effects

Cholestatic jaundice
Report yellowing of skin or eyes to your doctor.
Agranulocytosis
Report signs of infection such as fever, sore throat, or mouth ulcers.
Thrombocytopenia
Report unusual bruising or bleeding.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Contrast media Major
Alcohol Major
Beta-blockers Major
Diuretics Moderate
Corticosteroids Moderate
ACE inhibitors Moderate
Cimetidine Minor
Rifampicin Minor

🚨 Major Interactions

  • Contrast media (iodinated)
  • Alcohol
  • Beta-blockers

⚡ Moderate Interactions

  • Diuretics (thiazides, loop)
  • Corticosteroids
  • ACE inhibitors

🍷 Alcohol Interaction

Alcohol should be avoided while taking this medicine due to an increased risk of lactic acidosis and severe hypoglycemia. Alcohol can also worsen diabetes control and lead to other health complications.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Type 1 diabetes mellitus","Diabetic ketoacidosis","Severe renal impairment (eGFR

⚠️ Warnings & Precautions

["Risk of lactic acidosis with Metformin, especially in renal impairment, sepsis, dehydration, or alcohol use.","Hypoglycemia risk with Glimepiride, particularly in elderly, malnourished, or those with adrenal/pituitary insufficiency.","Discontinue before surgery or contrast imaging and restart only after renal function is normal.","Avoid in patients with conditions that predispose to tissue hypoxia (e.g., heart failure, respiratory failure).","May cause vitamin B12 deficiency with long-term use; monitor levels.","Use with caution in elderly patients due to increased risk of hypoglycemia."]

🤱 Lactation Safety

Not established from the available information. Consult your doctor before breastfeeding while taking this medicine.

💊 Overdose Management

Overdose can cause severe hypoglycemia and lactic acidosis. Immediate medical attention is required. Treatment includes supportive care, monitoring of blood glucose, and administration of intravenous glucose for hypoglycemia. Lactic acidosis may require hemodialysis. Contact a poison control center or emergency department immediately.

⏰ Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule. Do not take a double dose to make up for a missed one.

Additional Safety Advice

General Safety

Take this medicine exactly as prescribed by your doctor, with meals to reduce stomach upset and lower the risk of hypoglycemia. Do not skip meals while on this medicine. Monitor your blood sugar regularly as advised. Avoid alcohol, as it can increase the risk of lactic acidosis and low blood sugar. Inform your doctor if you have kidney or liver problems, or if you are scheduled for surgery or imaging tests with contrast dyes. Do not take this medicine if you are pregnant or planning pregnancy without consulting your doctor. Keep a source of fast-acting sugar (like glucose tablets) with you at all times in case of hypoglycemia. Do not share this medicine with others.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients are at higher risk of hypoglycemia and renal impairment. Start with the lowest dose and monitor closely. Regular renal function tests are recommended.

🤰 Pregnancy Planning (TTC)

This medicine is not recommended during pregnancy. If you are planning pregnancy, consult your doctor to switch to a safer alternative, such as insulin.

🏥 Post-Surgery Considerations

Discontinue this medicine before surgery and restart only after your doctor confirms normal renal function and stable blood sugar.

🦷 Dental Procedures

Inform your dentist about this medicine. Hypoglycemia risk may require adjusting meal timing around dental procedures.

💚 Lifestyle Tips for Better Results

🏃
Maintain a healthy weight to improve insulin sensitivity.
🥗
Engage in regular physical activity like walking or swimming.
😴
Follow a balanced diet rich in fiber and low in refined sugars.
💧
Monitor your blood sugar regularly as advised.
🧘
Get adequate sleep and manage stress.

🏋️ Exercise Considerations

Exercise can lower blood sugar. Monitor your levels before and after exercise, and carry a source of fast-acting sugar. Adjust medication timing with your doctor's advice.

🥗 Diet Recommendations

Include whole grains, fruits, and vegetables.
Limit intake of sugary drinks and processed foods.
Eat small, frequent meals to avoid blood sugar spikes.
Stay hydrated with water.

💼 Impact on Daily Work & Life

This medicine may cause hypoglycemia, which can affect your ability to drive or operate machinery. Avoid these activities if you feel shaky or confused. Inform your employer about your condition if necessary.

🛑 When to Stop This Medicine

Do not stop this medicine without consulting your doctor. Stopping suddenly can cause blood sugar levels to rise. Your doctor may adjust or change the medicine based on your condition.

📅 Long-Term Use Effects

Long-term use may lead to vitamin B12 deficiency, requiring periodic monitoring. Renal function should be checked regularly. The risk of hypoglycemia persists, especially in elderly patients. Cardiovascular benefits may be seen with good glycemic control.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Lifestyle modifications

Diet and exercise are essential for managing type 2 diabetes and can reduce medication needs.

Evidence: Well-established
Other oral antidiabetics

DPP-4 inhibitors, SGLT2 inhibitors, or GLP-1 receptor agonists may be alternatives.

Evidence: Well-established

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

No specific vaccine interactions are established. However, maintain routine vaccinations, including influenza and pneumococcal vaccines, as diabetes increases infection risk.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate unless specified

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✈️ Traveling with This Medicine

Carry this medicine in its original packaging with a copy of your prescription. Store at room temperature and protect from moisture. If traveling across time zones, adjust dosing times gradually in consultation with your doctor. Keep a supply of fast-acting sugar and a glucometer handy. Check customs regulations for carrying prescription medicines.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 52-year-old man with type 2 diabetes not controlled on Metformin alone.
He was prescribed this medicine as an add-on. After 4 weeks, his fasting blood sugar improved significantly. He experienced mild nausea initially, which resolved after taking it with breakfast. He now maintains a healthy diet and walks daily.
💡 Lesson: Taking this medicine with food improves tolerability and consistency leads to better sugar control.
👤 A 65-year-old woman with type 2 diabetes and mild renal impairment.
She was started on this medicine with careful monitoring of renal function. Her blood sugar improved, but she had one episode of mild hypoglycemia. The dose was adjusted, and she was advised to eat regular meals.
💡 Lesson: Elderly patients need lower doses and regular monitoring to prevent hypoglycemia.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: This medicine starts lowering blood sugar within a few hours, but full effects may take 1-2 weeks. Regular monitoring is important.

Q: Can I take this medicine if I have kidney disease?

A: It depends on the severity of kidney disease. Your doctor will adjust the dose or choose an alternative if needed.

Q: What should I do if I experience low blood sugar?

A: Immediately consume fast-acting sugar like glucose tablets or fruit juice, and inform your doctor.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?

🔄 Substitutes for apriglim-m 0.5 tablet sr

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: This medicine can cure diabetes.
    Fact: This medicine helps control blood sugar but does not cure diabetes. Lifestyle modifications and ongoing treatment are essential.
  • Myth: You can stop taking this medicine once your sugar levels are normal.
    Fact: Normal sugar levels are due to the medicine. Stopping without medical advice can cause sugar levels to rise again.
  • Myth: This medicine causes kidney damage.
    Fact: Metformin is excreted by the kidneys but does not cause kidney damage. However, it should be used with caution in kidney disease.

🔄 Alternative Options

Generic Alternatives

  • Glimepiride + Metformin combination generics

Brand Alternatives

  • Azulix 0.5 MF Tablet PR

📊 Comparison with Similar Medicines

[{"medicine":"This medicine","composition":"Glimepiride 0.5 mg + Metformin 500 mg","release_type":"Immediate release","frequency":"Once or twice daily"},{"medicine":"Glimepiride 1 mg + Metformin 500 mg","composition":"Glimepiride 1 mg + Metformin 500 mg","release_type":"Immediate release","frequency":"Once or twice daily"}]

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