agopride injection - Leuprolide (1mg/ml) medicine

Agopride Injection (Leuprolide 1mg/ml) - Uses, Price, Side Effects

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๐Ÿญ Alkem Laboratories Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is agopride injection used for?

Agopride Injection contains Leuprolide, a GnRH agonist that reduces estrogen levels. It is used to treat endometriosis, uterine fibroids, and advanced prostate cancer. By suppressing ovarian or testicular hormone production, it helps relieve symptoms and shrink abnormal tissue. Administered as a subcutaneous injection, it is typically given once a month.

  • Generic Name: Leuprolide
  • Manufacturer: Alkem Laboratories Ltd
  • Form: Allopathy
  • Pregnancy Category: X
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

๐Ÿ’Š agopride injection Uses & Benefits

Endometriosis, uterine fibroids, central precocious puberty, prostate cancer (male), assisted reproduction

Off-label uses: Breast cancer, transgender hormone therapy, hirsutism

๐Ÿ“‹ Drug Information

Generic Name(s)Leuprolide
Brand NameAgopride Injection
ManufacturerAlkem Laboratories Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassGYNAECOLOGICAL
Action ClassGNRH agonists/analogue
Route of AdministrationSubcutaneous or intramuscular injection
StorageStore at 20-25ยฐC; protect from light
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed after subcutaneous or intramuscular injection
DistributionDistributes widely; volume of distribution ~27 L
Protein Binding~43-49% bound to plasma proteins
MetabolismMetabolized primarily by peptidases; not significantly hepatic
Half-Life~3 hours (single dose); prolonged with depot formulations
ExcretionRenal (primarily as metabolites)
Bioavailability~90% after subcutaneous injection
Onset of ActionInitial flare (1-2 weeks) then suppression (2-4 weeks)
Peak Plasma Time1-2 hours after injection
Duration of Action1 month (depot formulation)

How It Works

GnRH agonist; continuous stimulation downregulates pituitary GnRH receptors, reducing LH and FSH secretion, thereby suppressing gonadal steroid production

Mechanism Steps

1Binds to GnRH receptors on pituitary gonadotropes
2Initial stimulation causes LH and FSH release (flare effect)
3Continuous exposure desensitizes receptors

๐Ÿ’ก How to Take agopride injection

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โŒ ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of agopride injection

โœ… Common Side Effects

  • Hot flashes
  • Sweating
  • Headache
  • Nausea
  • Injection site reactions
  • Vaginal dryness
  • Decreased libido

๐Ÿšจ Serious Side Effects

  • Anaphylaxis
  • Seizures
  • Pituitary apoplexy
  • Spinal cord compression
  • QT prolongation

โš ๏ธ Rare Side Effects

  • Osteoporosis
  • Hyperglycemia
  • Depression
  • Thromboembolism

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
NSAIDs Moderate Increased risk of fluid retention
Anticoagulants Moderate Increased bleeding risk
Corticosteroids Moderate Increased risk of hyperglycemia

๐Ÿšจ Major Interactions

  • Estrogen-containing medications
  • Progestins
  • Gonadotropins

โšก Moderate Interactions

  • Antidiabetic agents
  • Corticosteroids
  • Anticoagulants

โ„น๏ธ Minor Interactions

  • None significant

๐Ÿฝ๏ธ Food Interactions

None known

๐Ÿท Alcohol Interaction

No known interaction

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Low
Heart
Low
Pregnancy
Category X

๐Ÿšซ Contraindications

Pregnancy, lactation, undiagnosed vaginal bleeding, hypersensitivity to GnRH agonists

๐Ÿ“Š Monitoring Parameters

Hormone levels (LH, FSH, estradiol/testosterone), bone density, lipid profile, blood glucose

๐Ÿคฑ Lactation Safety

Not recommended; may suppress lactation

๐Ÿ’Š Overdose Management

Supportive care; no specific antidote

โฐ Missed Dose

Administer as soon as remembered; do not double dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for agopride injection

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Alternative brands with exact same active ingredient (Leuprolide (1mg/ml)):

Medical Note: Always consult your doctor before switching medications.

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