daslemia 100 tablet - Dasatinib (100mg) medicine

daslemia 100 tablet - Uses, Price, Side Effects & Substitutes

No reviews yet
๐Ÿญ Intas Pharmaceuticals Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jul 1, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jul 01, 2026

What is daslemia 100 tablet used for?

Alsatinib (Dasatinib) is used to treat ANTI NEOPLASTICS. It contains Dasatinib (100mg), which Inhibits BCR-ABL tyrosine kinase, SRC family kinases, and other oncogenic kinase. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Dasatinib
  • Manufacturer: Intas Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š daslemia 100 tablet Uses & Benefits

Chronic myeloid leukemia (CML) in chronic, accelerated, or blast phase; Philadelphia chromosome-positive acute lymphoblastic leukemia (Ph+ ALL).

Off-label uses: GIST (gastrointestinal stromal tumor) with specific mutations; other solid tumors with SRC activation.

๐Ÿ“‹ Drug Information

Generic Name(s)Dasatinib
Brand NameAlsatinib
ManufacturerIntas Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI NEOPLASTICS
Action ClassTyrosine kinase inhibitors
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF); protect from moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed after oral administration; peak plasma concentrations achieved within 0.5-6 hours.
DistributionWidely distributed; highly bound to plasma proteins (approximately 96%).
Protein Binding96%
MetabolismExtensively metabolized by CYP3A4, with minor contributions from flavin-containing monooxygenase 3 (FMO3) and UGT.
Half-Life3-5 hours
ExcretionPrimarily in feces (85%) and to a lesser extent in urine (4%).
Bioavailability14-34% (oral)
Onset of ActionWithin 2 hours
Peak Plasma Time0.5-6 hours
Duration of Action12-24 hours

How It Works

Inhibits BCR-ABL tyrosine kinase, SRC family kinases, and other oncogenic kinases.

Mechanism Steps

1Dasatinib binds to the ATP-binding site of BCR-ABL tyrosine kinase.
2Inhibits phosphorylation of downstream signaling proteins (e.g., STAT5, CRKL).
3Blocks cell proliferation and induces apoptosis in BCR-ABL-positive cells.

๐Ÿ’ก How to Take daslemia 100 tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of daslemia 100 tablet

โœ… Common Side Effects

  • Myelosuppression (neutropenia, thrombocytopenia, anemia)
  • Fluid retention (pleural effusion, peripheral edema)
  • Diarrhea
  • Headache
  • Fatigue
  • Nausea

๐Ÿšจ Serious Side Effects

  • Pleural effusion
  • Pulmonary arterial hypertension
  • QT prolongation
  • Severe hemorrhage
  • Hepatotoxicity

โš ๏ธ Rare Side Effects

  • Pancreatitis
  • Colitis
  • Severe skin reactions (Stevens-Johnson syndrome)
  • Tumor lysis syndrome

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Ketoconazole Major Increased dasatinib exposure (AUC increased 5-fold)
Rifampin Major Decreased dasatinib exposure (AUC decreased 82%)
Antacids Major Reduced absorption; separate by at least 2 hours
Grapefruit juice Moderate Increased dasatinib levels
Warfarin Minor Potential increased INR; monitor

๐Ÿšจ Major Interactions

  • CYP3A4 inhibitors (e.g., ketoconazole, clarithromycin)
  • CYP3A4 inducers (e.g., rifampin, phenytoin)
  • Antacids
  • H2 antagonists
  • Proton pump inhibitors

โšก Moderate Interactions

  • Grapefruit juice
  • St. John's wort
  • Calcium channel blockers
  • Statins

โ„น๏ธ Minor Interactions

  • Acetaminophen
  • Warfarin (monitor INR)

๐Ÿฝ๏ธ Food Interactions

Avoid grapefruit juice; take with or without food.

๐Ÿท Alcohol Interaction

May increase risk of liver toxicity; avoid excessive alcohol.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to dasatinib or any excipients; pregnancy; severe hepatic impairment.

๐Ÿ“Š Monitoring Parameters

Complete blood count (CBC), liver function tests, renal function, ECG for QT interval, pleural effusion symptoms.

๐Ÿคฑ Lactation Safety

Not recommended; excreted in animal milk, unknown in humans.

๐Ÿ’Š Overdose Management

No specific antidote; supportive care, monitor for myelosuppression and bleeding.

โฐ Missed Dose

Take as soon as remembered unless within 12 hours of next dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jul 01, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for daslemia 100 tablet

View All

Alternative brands with exact same active ingredient (Dasatinib (100mg)):

Medical Note: Always consult your doctor before switching medications.

๐Ÿ˜Š Was this information helpful?

Browse Medicines A-Z

Search our extensive medical database alphabetically.

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory
SaathiMed App
SaathiMed App Consult doctors & order medicines faster
Install