curekelafine 25mg/500mg tablet - Pyrimethamine (25mg) + Sulphadoxine (500mg) medicine

curekelafine 25mg/500mg tablet

4.5 (12 reviews)
๐Ÿญ Unicure India Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Aug 23, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Aug 23, 2026

What is curekelafine 25mg/500mg tablet used for?

Curekelafine (Pyrimethamine + Sulphadoxine) is used to treat ANTI MALARIALS. It contains Pyrimethamine (25mg) + Sulphadoxine (500mg), which Pyrimethamine inhibits dihydrofolate reductase; Sulphadoxine inhibits dihydropte. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Pyrimethamine + Sulphadoxine
  • Manufacturer: Unicure India Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š curekelafine 25mg/500mg tablet Uses & Benefits

Treatment of uncomplicated falciparum malaria; prophylaxis in chloroquine-resistant areas

Off-label uses: Toxoplasmosis (pyrimethamine alone)

๐Ÿ“‹ Drug Information

Generic Name(s)Pyrimethamine + Sulphadoxine
Brand NameCurekelafine
ManufacturerUnicure India Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI MALARIALS
Action ClassAntimalarial
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionWell absorbed orally
DistributionWidely distributed, crosses placenta and enters breast milk
Protein BindingPyrimethamine: 87%; Sulphadoxine: 90%
MetabolismHepatic
Half-LifePyrimethamine: 80-95 hours; Sulphadoxine: 100-200 hours
ExcretionRenal
BioavailabilityHigh
Onset of ActionWithin 1-2 hours
Peak Plasma TimePyrimethamine: 2-6 hours; Sulphadoxine: 2-8 hours
Duration of ActionLong (weeks)

How It Works

Pyrimethamine inhibits dihydrofolate reductase; Sulphadoxine inhibits dihydropteroate synthetase, synergistically blocking folate synthesis in Plasmodium

Mechanism Steps

1Pyrimethamine binds to dihydrofolate reductase, inhibiting conversion of dihydrofolate to tetrahydrofolate
2Sulphadoxine inhibits dihydropteroate synthetase, blocking incorporation of para-aminobenzoic acid into dihydropteroate
3Dual blockade of folate synthesis leads to depletion of tetrahydrofolate

๐Ÿ’ก How to Take curekelafine 25mg/500mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of curekelafine 25mg/500mg tablet

โœ… Common Side Effects

  • Nausea
  • Vomiting
  • Headache
  • Dizziness
  • Rash

๐Ÿšจ Serious Side Effects

  • Stevens-Johnson syndrome
  • Toxic epidermal necrolysis
  • Agranulocytosis
  • Aplastic anemia
  • Hepatotoxicity

โš ๏ธ Rare Side Effects

  • Megaloblastic anemia
  • Pulmonary infiltrates
  • Peripheral neuropathy

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Major Increased bleeding risk
Methotrexate Major Increased methotrexate toxicity
Phenytoin Major Increased phenytoin levels
Sulfonylureas Major Increased hypoglycemic effect
Chloramphenicol Moderate Increased bone marrow suppression
Oral contraceptives Moderate Reduced contraceptive efficacy
Thiazide diuretics Moderate Increased risk of thrombocytopenia
Vitamin C Minor Possible decreased absorption
Folic acid Minor Antagonizes effect

๐Ÿšจ Major Interactions

  • Warfarin
  • Methotrexate
  • Phenytoin
  • Sulfonylureas

โšก Moderate Interactions

  • Chloramphenicol
  • Oral contraceptives
  • Thiazide diuretics

โ„น๏ธ Minor Interactions

  • Vitamin C
  • Folic acid

๐Ÿฝ๏ธ Food Interactions

No significant food interactions

๐Ÿท Alcohol Interaction

Avoid alcohol due to increased hepatotoxicity risk

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to sulfonamides or pyrimethamine; severe hepatic or renal impairment; megaloblastic anemia; pregnancy (first trimester)

๐Ÿ“Š Monitoring Parameters

Complete blood count, liver function tests, renal function tests, folate levels

๐Ÿคฑ Lactation Safety

Caution; excreted in breast milk

๐Ÿ’Š Overdose Management

Gastric lavage, activated charcoal, supportive care; folinic acid for pyrimethamine toxicity

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose; do not double dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Last reviewed on: Aug 23, 2026

๐Ÿ”— View Profile

โญ User Reviews

Trusted Reviewer Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

Verified User Jul 10, 2026

Found this to be a helpful product. Good results.

Regular Customer Jul 10, 2026

Found this to be a helpful product. Good results.

Regular Customer Jul 10, 2026

Good quality medicine. Satisfied with the outcome.

Trusted Reviewer Jul 10, 2026

Effective and reliable. Worked as expected.

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