ctzone p 500mg/400mg tablet - Citicoline (500mg) + Piracetam (400mg) medicine

ctzone p 500mg/400mg tablet

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🏭 Mits Healthcare Pvt Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 23, 2026
📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Reviewed by
SaathiMed Expert Panel | Sep 23, 2026

What is ctzone p 500mg/400mg tablet used for?

This medicine contains Citicoline (500mg) + Piracetam (400mg) and is used to treat NEURO CNS. Citicoline provides choline for acetylcholine synthesis and cytidine for membrane phospholipids; Pir. Always consult your doctor before use.

  • Generic Name: Citicoline + Piracetam
  • Manufacturer: Mits Healthcare Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: Category C
  • Prescription Required: Yes
💡 Did You Know? India has the highest number of USFDA-compliant plants outside the USA.

💊 ctzone p 500mg/400mg tablet Uses & Benefits

Cognitive impairment, stroke recovery, dementia, traumatic brain injury.

Off-label uses: Alzheimer's disease, age-related memory decline, ADHD.

📋 Drug Information

Generic Name(s)Citicoline + Piracetam
Brand NameAzedra Plus Tablet
ManufacturerMits Healthcare Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassNootropic
Route of AdministrationOral
StorageStore at room temperature (20-25°C), protect from moisture.
Shelf LifeAs per manufacturer

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionRapidly absorbed after oral administration.
DistributionWidely distributed in body tissues, crosses blood-brain barrier.
Protein BindingCiticoline: <1%; Piracetam: negligible.
MetabolismCiticoline: hydrolyzed to choline and cytidine; Piracetam: not significantly metabolized.
Half-LifeCiticoline: 3.5-4.5 hours; Piracetam: 4-6 hours.
ExcretionPrimarily renal excretion.
BioavailabilityCiticoline: ~90%; Piracetam: ~100%.
Onset of ActionWithin 1-2 hours.
Peak Plasma TimeCiticoline: 1-2 hours; Piracetam: 1-1.5 hours.
Duration of Action6-8 hours.

How It Works

Citicoline provides choline for acetylcholine synthesis and cytidine for membrane phospholipids; Piracetam enhances neuronal membrane fluidity and neurotransmission.

Mechanism Steps

1Citicoline is hydrolyzed to choline and cytidine.
2Choline is used for acetylcholine synthesis.
3Cytidine is converted to uridine, enhancing membrane phospholipid synthesis.
4Piracetam modulates glutamatergic neurotransmission.
5Piracetam increases membrane fluidity and improves neuronal efficiency.

💡 How to Take ctzone p 500mg/400mg tablet

Follow your doctor's prescription exactly.

⚠️ Side Effects of ctzone p 500mg/400mg tablet

✅ Common Side Effects

Headache
Nausea
Diarrhea
Insomnia
Agitation

🚨 Serious Side Effects

Bleeding
Seizures
Severe allergic reaction

⚠️ Rare Side Effects

Angioedema
Hepatotoxicity
Thrombocytopenia

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Warfarin Major Increased bleeding risk
Antiplatelet drugs Major Increased bleeding risk
Levodopa Moderate Possible reduced efficacy of levodopa
Antipsychotics Moderate May worsen extrapyramidal symptoms
Caffeine Minor Additive CNS stimulation

🚨 Major Interactions

  • Warfarin
  • Antiplatelet drugs
  • Anticoagulants

⚡ Moderate Interactions

  • Levodopa
  • Antipsychotics
  • MAOIs

🍷 Alcohol Interaction

Avoid alcohol; may increase CNS depression.

🛡️ Safety & Warnings

🚫 Contraindications

Hypersensitivity, severe renal impairment, hemorrhagic stroke, pregnancy.

🤱 Lactation Safety

Not recommended; excreted in breast milk.

💊 Overdose Management

Symptomatic and supportive treatment; gastric lavage if recent ingestion.

⏰ Missed Dose

Take as soon as remembered; skip if near next dose.

🔄 Substitutes for ctzone p 500mg/400mg tablet

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

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