cilnikem-beta 5 tablet - Nebivolol (5mg) + Cilnidipine (10mg) medicine

cilnikem-beta 5 tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Alkem Laboratories Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 28, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 28, 2026

What is cilnikem-beta 5 tablet used for?

Cilacar NB 5 Tablet (Nebivolol + Cilnidipine) is used to treat CARDIAC. It contains Nebivolol (5mg) + Cilnidipine (10mg), which Nebivolol: Selective beta-1 blocker with nitric oxide-mediated vasodilation; Cil. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Nebivolol + Cilnidipine
  • Manufacturer: Alkem Laboratories Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

๐Ÿ’Š cilnikem-beta 5 tablet Uses & Benefits

Hypertension

Off-label uses: Chronic stable angina, Heart failure (nebivolol)

๐Ÿ“‹ Drug Information

Generic Name(s)Nebivolol + Cilnidipine
Brand NameCilacar NB 5 Tablet
ManufacturerAlkem Laboratories Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassAntihypertensive (Beta-blocker + Calcium channel blocker)
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionNebivolol: Rapidly absorbed; Cilnidipine: Well absorbed after oral administration.
DistributionNebivolol: Widely distributed; Cilnidipine: High volume of distribution.
Protein BindingNebivolol: ~98% bound to albumin; Cilnidipine: >99% bound to plasma proteins.
MetabolismNebivolol: Extensively metabolized via CYP2D6; Cilnidipine: Metabolized by CYP3A4.
Half-LifeNebivolol: 10-12 hours; Cilnidipine: 5-6 hours.
ExcretionNebivolol: Renal (38% unchanged) and fecal; Cilnidipine: Renal and fecal.
BioavailabilityNebivolol: 12-96% (first-pass effect); Cilnidipine: ~13%.
Onset of ActionNebivolol: 1-2 hours; Cilnidipine: 1-2 hours.
Peak Plasma TimeNebivolol: 1.5-4 hours; Cilnidipine: 1-2 hours.
Duration of ActionNebivolol: 24 hours; Cilnidipine: 24 hours.

How It Works

Nebivolol: Selective beta-1 blocker with nitric oxide-mediated vasodilation; Cilnidipine: L-type and N-type calcium channel blocker.

Mechanism Steps

1Nebivolol selectively blocks beta-1 adrenergic receptors in the heart, reducing heart rate and contractility.
2Nebivolol also stimulates nitric oxide release from endothelium, causing vasodilation.
3Cilnidipine blocks L-type calcium channels in vascular smooth muscle, leading to vasodilation.

๐Ÿ’ก How to Take cilnikem-beta 5 tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of cilnikem-beta 5 tablet

โœ… Common Side Effects

  • Headache
  • Dizziness
  • Fatigue
  • Edema
  • Bradycardia

๐Ÿšจ Serious Side Effects

  • Heart block
  • Severe hypotension
  • Bronchospasm
  • Hepatic injury

โš ๏ธ Rare Side Effects

  • Thrombocytopenia
  • Stevens-Johnson syndrome
  • Lupus-like syndrome

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
CYP2D6 inhibitors Major Increased nebivolol levels
CYP3A4 inhibitors Major Increased cilnidipine levels
Other antihypertensives Major Additive hypotension
Digoxin Moderate Increased bradycardia risk
Warfarin Moderate Increased INR
Insulin/oral hypoglycemics Moderate Masked hypoglycemia symptoms
Cimetidine Minor Slight increase in nebivolol levels
Grapefruit juice Minor Increased cilnidipine absorption

๐Ÿšจ Major Interactions

  • CYP2D6 inhibitors (e.g., quinidine, fluoxetine)
  • CYP3A4 inhibitors (e.g., ketoconazole, ritonavir)
  • Other antihypertensives (additive hypotension)

โšก Moderate Interactions

  • Digoxin
  • Warfarin
  • Insulin/oral hypoglycemics

โ„น๏ธ Minor Interactions

  • Cimetidine
  • Grapefruit juice

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase cilnidipine levels.

๐Ÿท Alcohol Interaction

May enhance hypotensive effect; avoid excessive alcohol.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Sick sinus syndrome, heart block (2nd/3rd degree), cardiogenic shock, severe bradycardia, hypersensitivity.

๐Ÿ“Š Monitoring Parameters

Blood pressure, heart rate, ECG, renal function, blood glucose (in diabetics).

๐Ÿคฑ Lactation Safety

Not recommended; avoid breastfeeding.

๐Ÿ’Š Overdose Management

Symptomatic and supportive; monitor ECG, blood pressure; consider atropine for bradycardia.

โฐ Missed Dose

Take as soon as remembered; skip if near next dose; do not double.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 28, 2026

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