celavi-trio tablet - Olmesartan Medoxomil (20mg) + Cilnidipine (10mg) medicine

celavi-trio tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Ajanta Pharma Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jul 2, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jul 02, 2026

What is celavi-trio tablet used for?

Cilidin Trio 20mg/10mg/12.5mg Tablet (Olmesartan Medoxomil + Cilnidipine) is used to treat CARDIAC. It contains Olmesartan Medoxomil (20mg) + Cilnidipine (10mg), which Olmesartan blocks angiotensin II AT1 receptors; Cilnidipine blocks L-type and N-. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Olmesartan Medoxomil + Cilnidipine
  • Manufacturer: Ajanta Pharma Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š celavi-trio tablet Uses & Benefits

Hypertension

Off-label uses: Diabetic nephropathy, Chronic kidney disease

๐Ÿ“‹ Drug Information

Generic Name(s)Olmesartan Medoxomil + Cilnidipine
Brand NameCilidin Trio 20mg/10mg/12.5mg Tablet
ManufacturerAjanta Pharma Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassAngiotensin II Receptor Blocker (ARB) + Calcium Channel Blocker (CCB)
Route of AdministrationOral
StorageStore at 20-25ยฐC, protect from light and moisture
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionOlmesartan: Well absorbed, absolute bioavailability ~26%; Cilnidipine: Well absorbed, bioavailability ~13%
DistributionOlmesartan: Vd ~17 L; Cilnidipine: Vd ~3.5 L/kg
Protein BindingOlmesartan: >99%; Cilnidipine: >99%
MetabolismOlmesartan: Not significantly metabolized; Cilnidipine: Metabolized by CYP3A4
Half-LifeOlmesartan: ~13 h; Cilnidipine: ~5-10 h
ExcretionOlmesartan: 35-50% urine, 50-65% feces; Cilnidipine: 70% feces, 30% urine
BioavailabilityOlmesartan: 26%; Cilnidipine: 13%
Onset of ActionOlmesartan: 1-2 weeks for full effect; Cilnidipine: 2-4 h
Peak Plasma TimeOlmesartan: 1-2 h; Cilnidipine: 1-3 h
Duration of ActionOlmesartan: 24 h; Cilnidipine: 24 h

How It Works

Olmesartan blocks angiotensin II AT1 receptors; Cilnidipine blocks L-type and N-type calcium channels

Mechanism Steps

1Olmesartan selectively blocks AT1 receptors, preventing angiotensin II-mediated vasoconstriction and aldosterone secretion.
2Cilnidipine blocks L-type calcium channels in vascular smooth muscle and N-type calcium channels in sympathetic nerve endings.
3L-type blockade causes vasodilation and reduced peripheral resistance.

๐Ÿ’ก How to Take celavi-trio tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of celavi-trio tablet

โœ… Common Side Effects

  • Dizziness
  • Headache
  • Peripheral edema
  • Fatigue
  • Cough

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Hyperkalemia
  • Acute renal failure
  • Hypotension
  • Hepatotoxicity

โš ๏ธ Rare Side Effects

  • Rhabdomyolysis
  • Stevens-Johnson syndrome
  • Interstitial nephritis

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Lithium Major Increased lithium toxicity risk
NSAIDs Major Reduced antihypertensive effect, increased renal impairment risk
Potassium-sparing diuretics Major Hyperkalemia risk
CYP3A4 inhibitors Major Increased cilnidipine levels
Antidiabetic agents Moderate Enhanced hypoglycemic effect
Beta-blockers Moderate Additive bradycardia
Digoxin Moderate Increased digoxin levels
Antacids Minor Reduced absorption
Cimetidine Minor Increased cilnidipine levels

๐Ÿšจ Major Interactions

  • Lithium
  • NSAIDs
  • Potassium-sparing diuretics
  • CYP3A4 inhibitors (e.g., ketoconazole)

โšก Moderate Interactions

  • Antidiabetic agents
  • Beta-blockers
  • Digoxin

โ„น๏ธ Minor Interactions

  • Antacids
  • Cimetidine

๐Ÿฝ๏ธ Food Interactions

Avoid grapefruit juice (increases cilnidipine levels); high-fat meal reduces absorption

๐Ÿท Alcohol Interaction

May enhance hypotensive effect; avoid excessive alcohol

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity, pregnancy, bilateral renal artery stenosis, severe hepatic impairment, hypotension

๐Ÿ“Š Monitoring Parameters

Blood pressure, serum potassium, renal function, liver function

๐Ÿคฑ Lactation Safety

Not recommended; excreted in milk in animal studies

๐Ÿ’Š Overdose Management

Symptomatic treatment; monitor BP, ECG; gastric lavage if recent

โฐ Missed Dose

Take as soon as remembered; skip if near next dose; do not double

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jul 02, 2026

๐Ÿ”— View Profile

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