actibile 300 tablet - Ursodeoxycholic Acid (300mg) medicine

Actibile 300 Tablet: Complete Guide to Uses, Dosage, and Safety

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🏭 Zydus Cadila 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 25, 2026
⚠️ Hepatotoxicity Risk 🤰 Pregnancy Category Not applicable. The old letter-based pregnancy categories have been replaced. This medicine is used in some pregnancy-related liver conditions under specialist supervision. It should only be used during pregnancy if clearly needed and prescribed by a doctor. 📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Evidence: Well-established for gallstone dissolution and primary biliary cholangitis; limited for other uses.
Reviewed by
SaathiMed Expert Panel | Sep 25, 2026

When to Call Your Doctor IMMEDIATELY

  • Yellowing of the skin or eyes (jaundice)
  • Dark urine or pale stools
  • Severe abdominal pain, especially in the upper right abdomen
  • Persistent vomiting or severe diarrhea
  • Swelling of the face, lips, or throat
  • Difficulty breathing or rash
  • Unusual fatigue or weakness

If experiencing severe symptoms, call emergency services immediately.

What is actibile 300 tablet used for?

This medicine contains Ursodeoxycholic Acid 300 mg, an oral tablet used to dissolve cholesterol gallstones and treat certain liver diseases. It works by reducing cholesterol in bile and protecting liver cells. It is taken with food, and regular monitoring is required.

  • Generic Name: Ursodeoxycholic Acid
  • Manufacturer: Zydus Cadila
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 actibile 300 tablet के बारे में (Hindi Summary)

उपयोग: यह दवा अर्सोडीऑक्सीकोलिक एसिड 300 मिलीग्राम की गोली है, जिसका उपयोग पित्त की थैली में बनी कोलेस्ट्रॉल की पथरी को घोलने और कुछ लिवर रोगों जैसे प्राइमरी बिलियरी कोलैंजाइटिस के इलाज में किया जाता है। यह पित्त में कोलेस्ट्रॉल की मात्रा कम करके और लिवर की कोशिकाओं की रक्षा करके काम करती है। इसे भोजन के साथ लेना चाहिए और डॉक्टर की सलाह के अनुसार नियमित रूप से लेना चाहिए।

साइड इफेक्ट्स: इस दवा के सामान्य दुष्प्रभावों में दस्त, जी मिचलाना, पेट में हल्की असुविधा और कब्ज शामिल हैं। ये आमतौर पर हल्के होते हैं और कुछ समय में ठीक हो जाते हैं। कभी-कभी उल्टी या दाने हो सकते हैं। यदि आपको आंखों या त्वचा का पीलापन, गहरे रंग का पेशाब, गंभीर पेट दर्द, या लगातार उल्टी हो, तो तुरंत डॉक्टर से संपर्क करें।

सुरक्षा सलाह: इस दवा को डॉक्टर के बताए अनुसार ही लें। इसे भोजन के साथ पूरे पानी के साथ निगलें। बिना डॉक्टर की सलाह के इसे चबाएं या तोड़ें नहीं। नियमित रूप से लिवर फंक्शन टेस्ट कराते रहें। शराब का सेवन न करें क्योंकि इससे लिवर पर बुरा असर पड़ सकता है। गर्भावस्था, स्तनपान या गर्भधारण की योजना बनाते समय डॉक्टर से सलाह लें। एंटासिड या अन्य दवाओं के साथ लेने से पहले डॉक्टर से पूछें।

💡 Did You Know? India has the highest number of USFDA-compliant plants outside the USA.

💊 actibile 300 tablet Uses & Benefits

[{"condition":"Cholesterol gallstones","description":"Used to dissolve small, non-calcified cholesterol-rich gallstones in patients who cannot or should not undergo gallbladder surgery.","evidence":"Well-established"},{"condition":"Primary biliary cholangitis","description":"Improves liver enzyme levels and slows disease progression in adults with this chronic autoimmune liver disease.","evidence":"Well-established"},{"condition":"Intrahepatic cholestasis of pregnancy","description":"Helps relieve itching and improves liver enzyme abnormalities in pregnant women with this condition.","evidence":"Moderate"},{"condition":"Primary sclerosing cholangitis","description":"Sometimes used to improve liver enzymes, although benefit on long-term outcomes is uncertain.","evidence":"Limited"},{"condition":"Cystic fibrosis-related liver disease","description":"May be used to improve bile flow and liver function in some patients with cystic fibrosis.","evidence":"Limited"}]

Off-label uses: [{"condition":"Non-alcoholic fatty liver disease","description":"Occasionally prescribed to improve liver enzymes, but evidence for routine use is not strong.","evidence":"Limited"},{"condition":"Biliary dyspepsia","description":"Sometimes used for indigestion symptoms thought to be related to bile flow, but evidence is weak.","evidence":"Limited"}]

Primary treatment for: Cholesterol gallstones and primary biliary cholangitis

Also treats: Intrahepatic cholestasis of pregnancy, Primary sclerosing cholangitis, Cystic fibrosis-related liver disease

📋 Drug Information

Generic Name(s)Ursodeoxycholic Acid
Brand NameActibile 300 Tablet
ManufacturerZydus Cadila
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassGASTRO INTESTINAL
Action ClassHepatoprotectives
Route of AdministrationOral
StorageStore at room temperature between 15°C and 30°C. Keep in the original container, away from moisture and direct sunlight. Do not refrigerate unless specifically instructed.
Shelf LifeTypically 24 months from the date of manufacture. Check the expiry date on the pack.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Always take this medicine with food to improve absorption and reduce stomach upset.
2
Separate this medicine from aluminum-based antacids by at least two hours.
3
Monitor liver function tests regularly during treatment.
4
Advise patients to avoid alcohol to reduce liver stress.
5
For gallstone dissolution, ensure the stones are small and non-calcified before starting therapy.
6
Counsel patients that gallstone dissolution may take several months of continuous treatment.
7
Report persistent diarrhea or severe abdominal pain immediately.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

✅
Gallstone pain (biliary colic)
This medicine is used to dissolve cholesterol gallstones, but it does not provide immediate pain relief.
Likely Use
✅
Itching due to cholestasis
This medicine can help relieve itching in cholestatic liver diseases.
Likely Use
✅
Elevated liver enzymes
This medicine is used to improve liver enzyme levels in certain liver conditions.
Likely Use
❌
Fever
This medicine is not a fever reducer.
Not Primary
❌
Acute abdominal pain
This medicine is not for acute pain relief. Seek medical attention.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionThis medicine is absorbed from the small intestine after oral administration. Absorption is more efficient when the tablet is taken with food because food stimulates bile flow and improves dissolution.
DistributionIt is taken up extensively by the liver on first pass, and a portion enters the systemic circulation and is distributed to tissues. It is highly bound to plasma proteins, mainly albumin.
Protein BindingApproximately 96 to 99 percent bound to plasma proteins, primarily albumin.
MetabolismThis medicine is metabolized in the liver and by intestinal bacteria. It undergoes conjugation with glycine and taurine, and is also converted to other bile acids by bacterial enzymes in the gut.
Half-LifeNot established from the available information.
ExcretionIt is excreted mainly in the feces as bile acids and their metabolites. A small amount is excreted in the urine.
BioavailabilityNot established from the available information.
Onset of ActionThe onset of action is gradual. Improvement in liver enzyme levels may be noticed within a few weeks, while gallstone dissolution may take several months of continuous treatment.
Peak Plasma TimeNot established from the available information.
Duration of ActionThe effect persists as long as the medicine is taken regularly. Gallstone dissolution requires months of continuous therapy.

How It Works

This medicine works by replacing a portion of the natural bile acid pool with ursodeoxycholic acid, which is more water-soluble and less detergent to liver cells. It reduces the amount of cholesterol that the liver secretes into bile and shifts bile composition toward a state where cholesterol is less likely to crystallize into stones. It also protects liver cells from the toxic effects of retained bile acids and stimulates bile flow through the bile ducts.

Mechanism Steps

1
Uptake by the liver: After being absorbed from the intestine, this medicine is taken up efficiently by liver cells from the portal blood.
2
Conjugation and secretion into bile: Inside the liver, it is conjugated with glycine or taurine and then secreted into bile, where it becomes part of the bile acid pool.
3
Reduced cholesterol secretion: Its presence in bile reduces the amount of cholesterol that the liver releases into bile, lowering the chance of cholesterol crystals forming.
4
Gallstone dissolution: With continued use, cholesterol in existing gallstones gradually leaches out, causing the stones to shrink and sometimes disappear completely.
5
Liver cell protection: By displacing more toxic bile acids, this medicine reduces injury to liver cells and improves liver enzyme levels in cholestatic conditions.

💡 How to Take actibile 300 tablet

Strength: Ursodeoxycholic Acid 300 mg immediate-release tablet

1Take the tablet with a full glass of water.
2Take it with food to improve absorption and reduce stomach upset.
3Swallow the tablet whole. Do not crush, chew, or break it unless your doctor advises.
4Take it at the same times each day to maintain steady levels.
5If you take antacids or bile acid sequestrants, separate them by at least two hours.
6Do not stop taking this medicine without consulting your doctor.

Dosage Information

Adult DosageThe usual adult dose of this medicine for dissolving gallstones is 8 to 10 mg per kg of body weight per day, divided into two or three doses, taken with food. For primary biliary cholangitis, the typical dose is 13 to 15 mg per kg per day, often divided into two to four doses. Your doctor will determine the exact dose based on your weight, the condition being treated, and your liver function. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician.
Elderly DosageNo specific dose adjustment is established for elderly patients. However, because liver and kidney function may decline with age, your doctor will individualize the dose and monitor you closely.
Renal ImpairmentNo specific dose adjustment is established for patients with kidney impairment. Consult your doctor for individualized dosing.
Hepatic ImpairmentThis medicine is used in liver diseases, but in severe liver impairment, the dose may need to be adjusted or the medicine may not be suitable. Your doctor will determine the appropriate dose based on your liver function tests.
Maximum Daily DoseThe maximum daily dose is not established from the available information. Doses are individualized by a qualified clinician.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With meals
Take with food
Improves absorption and reduces stomach upset.
High-fiber meals
Avoid taking at the same time
Fiber can bind the medicine and reduce absorption.
Grapefruit
No specific restriction
No clinically significant interaction established.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of actibile 300 tablet

✅ Common Side Effects

Loose stools or mild diarrhea (Common (up to 10%))
Usually settles with continued use. Stay hydrated and consult your doctor if it persists or becomes severe.
Nausea (Common (up to 10%))
Taking the tablet with food may help. Consult your doctor if nausea is persistent.
Abdominal discomfort (Uncommon (1-10%))
Try taking the medicine with meals. Report persistent or severe pain to your doctor.
Constipation (Uncommon (1-10%))
Increase fiber and fluid intake. Consult your doctor if it does not improve.
Vomiting (Uncommon (1-10%))
Take with food and small sips of water. Seek medical advice if vomiting is severe or persistent.

🚨 Serious Side Effects

Worsening of liver inflammation (Rare (<0.1%))
Seek medical attention if you notice yellowing of eyes or skin, dark urine, or worsening fatigue.
Severe diarrhea with dehydration (Rare (<0.1%))
Stop the medicine and seek medical help if diarrhea is severe or you feel dizzy or weak.
Allergic reaction with facial swelling (Rare (<0.1%))
Seek emergency care immediately if you develop swelling of the face, lips, or throat, or difficulty breathing.
Calcification of gallstones (Rare (<0.1%))
This may make stones harder to dissolve. Your doctor will monitor with imaging if needed.

⚠️ Rare Side Effects

Severe skin rash or itching
Stop the medicine and consult your doctor promptly.
Low white blood cell count
Report unusual infections or fever to your doctor.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Aluminum antacids Major
Cholestyramine Major
Ciprofloxacin Moderate
Cyclosporine Moderate
Rosuvastatin Moderate
Nitrendipine Moderate
Oral contraceptives Moderate
Activated charcoal Minor
Sucralfate Minor
Colestipol Major

🚨 Major Interactions

  • Aluminum-based antacids
  • Cholestyramine and colestipol
  • Ciprofloxacin
  • Nitrendipine

⚡ Moderate Interactions

  • Cyclosporine
  • Rosuvastatin
  • Oral contraceptives

🍷 Alcohol Interaction

Alcohol can worsen liver disease and may increase the risk of liver-related side effects. It is best to avoid alcohol while taking this medicine, especially if you have an underlying liver condition.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Complete blockage of the bile duct","Acute inflammation of the gallbladder or bile ducts","Calcified gallstones that cannot dissolve","Known allergy to ursodeoxycholic acid or any ingredient","Severe liver failure"]

⚠️ Warnings & Precautions

["Take with food to improve absorption and reduce stomach upset.","Do not use for gallstones that are calcified or larger than 15 mm, as they are unlikely to dissolve.","Monitor liver function regularly during treatment.","Avoid alcohol to reduce liver stress.","Inform your doctor if you are pregnant, planning pregnancy, or breastfeeding.","Do not stop the medicine without consulting your doctor.","Report persistent diarrhea or severe abdominal pain immediately."]

🤱 Lactation Safety

It is not known whether this medicine passes into breast milk in significant amounts. Consult your doctor before breastfeeding while taking this medicine.

💊 Overdose Management

Overdose with this medicine is unlikely to cause serious harm because it is a naturally occurring bile acid. However, if a large amount is taken, seek medical attention. Treatment is supportive and symptomatic. Contact a poison control center or emergency department if you suspect an overdose.

⏰ Missed Dose

If you miss a dose, take it as soon as you remember, provided it is not almost time for your next dose. If it is nearly time for the next dose, skip the missed dose and continue with your regular schedule. Do not take a double dose to make up for a missed one.

Additional Safety Advice

General Safety

Take this medicine exactly as prescribed by your doctor. Swallow the tablet whole with a glass of water, and take it with food to improve absorption and reduce stomach upset. Do not crush, chew, or break the tablet unless your doctor specifically tells you to. Keep all your follow-up appointments because your doctor will need to check your liver function and monitor how well the medicine is working. Tell your doctor about all other medicines, supplements, and herbal products you are taking, especially antacids, cholesterol-lowering drugs, and antibiotics. Avoid alcohol while taking this medicine because it can worsen liver problems. If you are pregnant, planning pregnancy, or breastfeeding, speak to your doctor before taking this medicine. Do not share this medicine with anyone else, even if they have similar symptoms.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients may have reduced liver and kidney function. Your doctor will individualize the dose and monitor you closely for side effects. Regular liver function tests are important.

🤰 Pregnancy Planning (TTC)

If you are planning pregnancy, consult your doctor before taking this medicine. It may be used in certain pregnancy-related liver conditions under specialist supervision. Your doctor will weigh the benefits and risks.

🏥 Post-Surgery Considerations

If you have undergone gallbladder surgery, this medicine may no longer be needed for gallstone dissolution. Consult your doctor for guidance. After liver surgery, your doctor will determine if this medicine is appropriate.

🦷 Dental Procedures

There are no specific precautions for dental procedures while taking this medicine. However, inform your dentist about all medicines you are taking.

💚 Lifestyle Tips for Better Results

🏃
Maintain a healthy weight to reduce the risk of gallstones.
🥗
Eat a balanced diet low in saturated fats and cholesterol.
😴
Stay well hydrated by drinking plenty of water.
💧
Avoid alcohol to protect your liver.
🧘
Get regular exercise to support overall liver health.
🌞
Follow up regularly with your doctor for monitoring.

🏋️ Exercise Considerations

There are no specific exercise restrictions while taking this medicine. However, if you experience dizziness, fatigue, or abdominal discomfort, avoid strenuous activities until you feel better. Consult your doctor before starting any new exercise program.

🥗 Diet Recommendations

Include plenty of fruits and vegetables.
Choose whole grains over refined grains.
Limit fried and processed foods.
Reduce cholesterol-rich foods like red meat and full-fat dairy.
Stay well hydrated.

💼 Impact on Daily Work & Life

This medicine is unlikely to affect your ability to drive or operate machinery. However, if you experience dizziness, diarrhea, or fatigue, use caution. Most people can continue their normal daily activities while taking this medicine.

🛑 When to Stop This Medicine

Do not stop taking this medicine without consulting your doctor. If you experience severe side effects such as persistent diarrhea, jaundice, or allergic reactions, contact your doctor immediately. Your doctor will decide whether to adjust the dose or stop the medicine based on your condition and test results.

📅 Long-Term Use Effects

Long-term use of this medicine is generally well tolerated. Regular monitoring of liver function is required. In some cases, gallstones may calcify and become resistant to dissolution. If you have been on this medicine for a long time, your doctor will periodically assess whether continued treatment is beneficial. Do not stop the medicine without medical advice.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Surgical removal of gallbladder (cholecystectomy)

Definitive treatment for symptomatic gallstones.

Evidence: Well-established
Extracorporeal shock wave lithotripsy

Non-invasive procedure to break up gallstones, suitable for selected patients.

Evidence: Moderate
Dietary modifications

Low-fat diet can reduce gallbladder symptoms but does not dissolve stones.

Evidence: Limited

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

There are no specific vaccine interactions established with this medicine. However, if you have liver disease, discuss vaccination against hepatitis A and B with your doctor.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate unless specified

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✈️ Traveling with This Medicine

Carry this medicine in its original packaging with a copy of your prescription. Store it at room temperature, away from direct sunlight and moisture. If traveling across time zones, adjust your dosing schedule gradually as advised by your doctor. Keep enough supply for the entire trip. Check customs regulations for carrying prescription medicines. Do not pack it in checked luggage; keep it in your carry-on bag.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 52-year-old woman with small cholesterol gallstones who could not undergo surgery
She was prescribed this medicine at 10 mg per kg per day, taken with meals. After six months of regular use, an ultrasound showed that her gallstones had shrunk significantly. She experienced mild loose stools initially, which settled after a few weeks. She emphasized taking the medicine with food and keeping all follow-up appointments.
💡 Lesson: Consistent daily dosing with food and regular monitoring can lead to successful gallstone dissolution over time.
👤 A 45-year-old man with primary biliary cholangitis and elevated liver enzymes
He started this medicine at 13 mg per kg per day divided into two doses. Within three months, his liver enzyme levels improved markedly, and his itching reduced. He reported no major side effects and continued the medicine as prescribed. He learned the importance of avoiding alcohol and attending regular liver function tests.
💡 Lesson: This medicine can significantly improve liver enzyme levels and quality of life in chronic cholestatic liver disease when taken regularly.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: For liver enzyme improvement, it may take a few weeks. For gallstone dissolution, it may take several months of continuous treatment.

Q: Can I take this medicine with food?

A: Yes, it should be taken with food to improve absorption and reduce stomach upset.

Q: What should I do if I miss a dose?

A: Take it as soon as you remember if it is not almost time for your next dose. Otherwise, skip the missed dose and continue with your regular schedule. Do not double dose.

Q: Is this medicine safe during pregnancy?

A: It should only be used during pregnancy if clearly needed and prescribed by a doctor. Consult your doctor for personalized advice.

Q: Can I stop taking this medicine suddenly?

A: No, do not stop without consulting your doctor. Stopping suddenly may worsen your condition.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?

🔄 Substitutes for actibile 300 tablet

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: This medicine provides immediate pain relief for gallstones.
    Fact: This medicine does not relieve pain immediately. It works slowly to dissolve stones over months.
  • Myth: This medicine can dissolve all types of gallstones.
    Fact: It is only effective for small, non-calcified cholesterol gallstones. Calcified or large stones do not dissolve.
  • Myth: You can stop this medicine once you feel better.
    Fact: Stopping suddenly can cause the condition to worsen. Always consult your doctor before stopping.

🔄 Alternative Options

Generic Alternatives

  • Ursodeoxycholic Acid 300 mg tablet (various manufacturers)

Brand Alternatives

  • Actibile 300 Tablet

📊 Comparison with Similar Medicines

[{"medicine":"Ursodeoxycholic Acid","class":"Bile acid","primary_use":"Gallstone dissolution, cholestatic liver disease","route":"Oral"},{"medicine":"Chenodeoxycholic acid","class":"Bile acid","primary_use":"Gallstone dissolution","route":"Oral"},{"medicine":"Obeticholic acid","class":"FXR agonist","primary_use":"Primary biliary cholangitis","route":"Oral"}]

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