abline 500mg/75mg tablet - Methylcobalamin (500mg) + Pregabalin (75mg) medicine

abline 500mg/75mg tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Aanika Pharma ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is abline 500mg/75mg tablet used for?

Axogurd-SR Tablet (Methylcobalamin + Pregabalin) is used to treat NEURO CNS. It contains Methylcobalamin (500mg) + Pregabalin (75mg), which Methylcobalamin: Coenzyme for myelin synthesis; Pregabalin: Binds to alpha2-delt. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Methylcobalamin + Pregabalin
  • Manufacturer: Aanika Pharma
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

๐Ÿ’Š abline 500mg/75mg tablet Uses & Benefits

Diabetic neuropathy, postherpetic neuralgia, fibromyalgia, neuropathic pain associated with spinal cord injury.

Off-label uses: Generalized anxiety disorder, social anxiety disorder, restless legs syndrome.

๐Ÿ“‹ Drug Information

Generic Name(s)Methylcobalamin + Pregabalin
Brand NameAxogurd-SR Tablet
ManufacturerAanika Pharma
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassNeurotropic vitamin + Gabapentinoid
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionMethylcobalamin: Well absorbed orally; Pregabalin: Rapidly absorbed after oral administration with peak plasma concentrations within 1 hour.
DistributionMethylcobalamin: Distributed to tissues including CNS; Pregabalin: Crosses blood-brain barrier, distributed throughout body.
Protein BindingMethylcobalamin: Low (<10%); Pregabalin: <1% bound to plasma proteins.
MetabolismMethylcobalamin: Metabolized in the liver; Pregabalin: Negligible metabolism (<2% of dose).
Half-LifeMethylcobalamin: Approximately 6 hours; Pregabalin: Approximately 6.3 hours.
ExcretionMethylcobalamin: Renal excretion; Pregabalin: Primarily excreted unchanged in urine (90-99%).
BioavailabilityMethylcobalamin: Variable, approximately 50%; Pregabalin: >90%.
Onset of ActionMethylcobalamin: Days to weeks; Pregabalin: Within 1 hour.
Peak Plasma TimeMethylcobalamin: 2-3 hours; Pregabalin: 1 hour.
Duration of ActionMethylcobalamin: Several hours; Pregabalin: 6-8 hours.

How It Works

Methylcobalamin: Coenzyme for myelin synthesis; Pregabalin: Binds to alpha2-delta subunit of voltage-gated calcium channels, reducing calcium influx and neurotransmitter release.

Mechanism Steps

1Methylcobalamin acts as a cofactor for methionine synthase, promoting myelin synthesis.
2Pregabalin binds to the alpha2-delta subunit of voltage-gated calcium channels in the CNS.
3Binding reduces calcium influx at nerve terminals.

๐Ÿ’ก How to Take abline 500mg/75mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of abline 500mg/75mg tablet

โœ… Common Side Effects

  • Dizziness
  • Somnolence
  • Dry mouth
  • Edema
  • Blurred vision
  • Weight gain
  • Constipation

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Hypersensitivity reactions
  • Suicidal thoughts
  • Rhabdomyolysis
  • PR interval prolongation

โš ๏ธ Rare Side Effects

  • Stevens-Johnson syndrome
  • Hepatotoxicity
  • Pancreatitis
  • Blood dyscrasias

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
CNS depressants Major Increased sedation and respiratory depression
Thalidomide Major Increased risk of peripheral neuropathy
ACE inhibitors Major Increased risk of angioedema
Oral hypoglycemics Moderate May enhance hypoglycemic effect
Antihypertensives Moderate Additive hypotensive effect
Antacids Minor Reduced absorption of pregabalin
H2 blockers Minor Possible reduced absorption of pregabalin

๐Ÿšจ Major Interactions

  • Central nervous system depressants
  • Thalidomide
  • Angiotensin-converting enzyme inhibitors

โšก Moderate Interactions

  • Oral hypoglycemics
  • Antihypertensives

โ„น๏ธ Minor Interactions

  • Antacids
  • H2 blockers

๐Ÿฝ๏ธ Food Interactions

High-fat meal may delay absorption of pregabalin

๐Ÿท Alcohol Interaction

Additive CNS depression; avoid concurrent use.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to any component; severe renal impairment (CrCl <30 mL/min) for pregabalin.

๐Ÿ“Š Monitoring Parameters

Renal function, liver function, CBC, signs of hypersensitivity, CNS depression, suicidal ideation.

๐Ÿคฑ Lactation Safety

Pregabalin excreted in breast milk; caution advised.

๐Ÿ’Š Overdose Management

Supportive care; activated charcoal if recent ingestion; hemodialysis may remove pregabalin.

โฐ Missed Dose

Take as soon as remembered unless near next dose; skip missed dose if close to next dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

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