listap 150 sr tablet - Epalrestat (150mg) medicine

Epstat 150mg Tablet SR: Comprehensive Guide to Uses, Side Effects, and Safety

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🏭 Vivid Biotek Pvt Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 24, 2026
⚠️ Hepatotoxicity Risk 📋 Prescription Required 💊 Generic Available
Medically Reviewed
12 min read
Evidence: Moderate for diabetic neuropathy in some regions; limited in others.
Reviewed by
SaathiMed Expert Panel | Sep 24, 2026

When to Call Your Doctor IMMEDIATELY

  • Yellowing of skin or eyes
  • Dark urine or pale stools
  • Severe abdominal pain
  • Persistent nausea and vomiting
  • Difficulty breathing or swelling of face, lips, or throat
  • Unusual bleeding or bruising
  • Severe dizziness or fainting

If experiencing severe symptoms, call emergency services immediately.

What is listap 150 sr tablet used for?

This medicine contains Epalrestat 150 mg, an aldose reductase inhibitor used to manage diabetic peripheral neuropathy. It works by reducing sorbitol accumulation in nerves, helping to alleviate tingling, numbness, and pain. It is taken orally once daily with meals, and dose adjustments may be needed for liver or kidney problems.

  • Generic Name: Epalrestat (150mg)
  • Manufacturer: Vivid Biotek Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 listap 150 sr tablet के बारे में (Hindi Summary)

उपयोग: यह दवा एपलरेस्टैट 150 मिलीग्राम युक्त है और मधुमेह के कारण होने वाली तंत्रिका समस्या (डायबिटिक न्यूरोपैथी) के इलाज में उपयोग की जाती है। यह हाथ-पैरों में झनझनाहट, सुन्नपन, जलन और दर्द को कम करने में मदद करती है। यह दवा एल्डोज रिडक्टेज एंजाइम को रोककर काम करती है, जिससे तंत्रिका कोशिकाओं में सोर्बिटोल का जमाव कम होता है और तंत्रिका क्षति धीमी होती है। इसे आमतौर पर दिन में एक बार भोजन के साथ लिया जाता है। यह दवा डॉक्टर के पर्चे के बिना नहीं लेनी चाहिए।

साइड इफेक्ट्स: इस दवा के कुछ सामान्य दुष्प्रभाव हो सकते हैं जैसे मतली, उल्टी, दस्त, पेट में असहजता, सिरदर्द और चक्कर आना। ये आमतौर पर हल्के होते हैं और कुछ समय में ठीक हो जाते हैं। दुर्लभ मामलों में यह लिवर की समस्या, त्वचा पर चकत्ते, या सांस लेने में कठिनाई पैदा कर सकती है। अगर आपको पीलिया, गहरे रंग का पेशाब, या लगातार पेट दर्द हो, तो तुरंत डॉक्टर से संपर्क करें।

सुरक्षा सलाह: इस दवा को लेने से पहले अपने डॉक्टर को अपनी सभी स्वास्थ्य समस्याओं और दवाओं के बारे में बताएं। गर्भावस्था या स्तनपान के दौरान इस दवा का उपयोग डॉक्टर की सलाह के बिना न करें। शराब का सेवन न करें क्योंकि इससे लिवर की समस्या बढ़ सकती है। दवा को डॉक्टर के बताए अनुसार ही लें, खुराक न बदलें। यदि खुराक छूट जाए तो याद आते ही ले लें, लेकिन अगली खुराक का समय नजदीक हो तो छूटी हुई खुराक न लें। दवा को ठंडी और सूखी जगह पर रखें। नियमित रूप से ब्लड शुगर की जांच कराएं।

💡 Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

💊 listap 150 sr tablet Uses & Benefits

[{"condition":"Diabetic peripheral neuropathy","description":"This medicine is used to improve symptoms such as tingling, numbness, burning, and pain in the hands and feet caused by nerve damage due to diabetes.","evidence":"Well-established in some regions; evidence varies"},{"condition":"Diabetic autonomic neuropathy","description":"May be used to help manage symptoms related to autonomic nerve damage, such as gastrointestinal issues, though evidence is limited.","evidence":"Limited"}]

Off-label uses: [{"condition":"Other neuropathic pain conditions","description":"Occasionally prescribed off-label for neuropathic pain not related to diabetes, but evidence is insufficient.","evidence":"Limited"}]

Primary treatment for: Diabetic peripheral neuropathy

Also treats: Diabetic autonomic neuropathy, Other neuropathic pain conditions

📋 Drug Information

Generic Name(s)Epalrestat (150mg)
Brand Namelistap 150 sr tablet
ManufacturerVivid Biotek Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI DIABETIC
Action ClassAldose reductase inhibitor
Route of AdministrationOral
StorageStore at room temperature (15-30°C) in a cool, dry place away from direct sunlight. Keep in the original container.
Shelf Life24 months from the date of manufacture.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Take this medicine with meals to reduce stomach upset.
2
Monitor your blood sugar levels regularly while on this medicine.
3
Avoid alcohol consumption as it may increase liver toxicity.
4
Do not stop taking this medicine without consulting your doctor.
5
Report any signs of liver problems like yellowing of eyes or dark urine immediately.
6
Keep all follow-up appointments for monitoring liver and kidney function.
7
Inform your doctor if you experience dizziness or vision changes.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

Tingling in hands and feet
This medicine is commonly prescribed for this.
Likely Use
Burning sensation in feet
This medicine may help relieve this symptom.
Likely Use
Fever
This medicine is not a primary fever reducer.
Not Primary
Headache
This medicine is not used for headache relief.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionEpalrestat is absorbed from the gastrointestinal tract after oral administration. The exact bioavailability and absorption rate are not established from the available information.
DistributionNot established from the available information.
Protein BindingNot established from the available information.
MetabolismEpalrestat is metabolized in the liver, primarily through oxidation and conjugation reactions. The specific enzymes involved are not fully characterized.
Half-LifeNot established from the available information.
ExcretionEpalrestat and its metabolites are excreted mainly via the kidneys in urine and to a lesser extent in feces.
BioavailabilityNot established from the available information.
Onset of ActionThe onset of action for symptom relief may take several weeks to months, as it works by preventing further nerve damage rather than providing immediate pain relief.
Peak Plasma TimeNot established from the available information.
Duration of ActionNot established from the available information.

How It Works

This medicine works by inhibiting the enzyme aldose reductase, which is involved in the polyol pathway. Under high blood sugar conditions, this pathway becomes overactive, leading to the accumulation of sorbitol and fructose inside nerve cells. This accumulation causes osmotic stress and oxidative damage, contributing to nerve dysfunction. By blocking aldose reductase, this medicine reduces sorbitol production and helps protect nerve cells from damage.

Mechanism Steps

1
Inhibition of aldose reductase: This medicine binds to and inhibits the aldose reductase enzyme, blocking the conversion of glucose to sorbitol.
2
Reduced sorbitol accumulation: With less sorbitol produced, osmotic stress inside nerve cells is decreased, preventing swelling and damage.
3
Decreased oxidative stress: By limiting the polyol pathway, this medicine reduces the production of reactive oxygen species that harm nerves.
4
Improved nerve function: Over time, these effects help improve nerve conduction and reduce symptoms like tingling, numbness, and pain.

💡 How to Take listap 150 sr tablet

Strength: Sustained-release tablet, 150 mg

1Take this medicine exactly as prescribed by your doctor.
2Swallow the tablet whole with a glass of water. Do not crush, chew, or break the sustained-release tablet.
3Take it with meals to reduce stomach upset.
4Take it at the same time each day to maintain consistent levels.
5Do not take more than the prescribed dose.
6If you miss a dose, follow the missed dose instructions.
7Do not stop taking this medicine without consulting your doctor.

Dosage Information

Adult DosageThe usual adult dose of this medicine is 150 mg taken orally once daily, preferably with meals to reduce stomach upset. However, the dose may be adjusted by your doctor based on your condition, response to treatment, and kidney or liver function. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function. Do not change the dose without consulting your doctor.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician.
Elderly DosageElderly patients may be more sensitive to the effects of this medicine. Dose adjustments may be necessary based on kidney and liver function. Consult your doctor for appropriate dosing.
Renal ImpairmentDose adjustment may be needed in patients with kidney impairment. Consult your doctor for appropriate dosing.
Hepatic ImpairmentDose adjustment may be needed in patients with liver impairment. Consult your doctor for appropriate dosing.
Maximum Daily Dose150 mg per day, unless otherwise directed by your doctor.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With meals
Take with food
Reduces stomach upset and improves tolerability.
Alcohol
Avoid
Increases risk of liver problems and side effects.
Grapefruit
Caution
May affect drug metabolism; monitor for side effects.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of listap 150 sr tablet

✅ Common Side Effects

Nausea (Common (5-10%))
Take with food to reduce nausea. If it persists, consult your doctor.
Vomiting (Common (5-10%))
Stay hydrated and inform your doctor if vomiting is severe or persistent.
Diarrhea (Common (5-10%))
Drink plenty of fluids. If diarrhea lasts more than a few days, consult your doctor.
Stomach discomfort (Common (5-10%))
Take with meals. Avoid spicy or fatty foods.
Headache (Common (5-10%))
Rest and stay hydrated. If headache is severe or persistent, consult your doctor.

🚨 Serious Side Effects

Liver dysfunction (Rare (<0.1%))
Seek immediate medical attention if you notice yellowing of skin or eyes, dark urine, or severe abdominal pain.
Severe allergic reaction (Rare (<0.1%))
Seek emergency help if you experience swelling of face, lips, throat, or difficulty breathing.
Blood dyscrasias (Rare (<0.1%))
Report unusual bleeding, bruising, or persistent fever to your doctor immediately.

⚠️ Rare Side Effects

Skin rash
Discontinue and consult your doctor if rash develops.
Itching
Consult your doctor if itching is bothersome.
Dizziness
Avoid driving or operating machinery until you know how this medicine affects you.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Insulin Moderate
Sulfonylureas Moderate
Methotrexate Moderate
Isoniazid Moderate
Warfarin Minor
Diuretics Minor
ACE inhibitors Minor
NSAIDs Minor
Grapefruit juice Minor
Other aldose reductase inhibitors Major

🚨 Major Interactions

  • Other aldose reductase inhibitors

⚡ Moderate Interactions

  • Antidiabetic drugs (e.g., insulin, sulfonylureas)
  • Hepatotoxic drugs (e.g., methotrexate, isoniazid)

🍷 Alcohol Interaction

Avoid consuming alcohol while taking this medicine, as it can increase the risk of liver damage and may worsen side effects such as nausea and dizziness.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Hypersensitivity to Epalrestat or any component of the tablet","Pregnancy and breastfeeding (unless advised by doctor)","Severe liver disease","Severe kidney disease"]

⚠️ Warnings & Precautions

["Use with caution in patients with liver or kidney impairment.","May cause dizziness; avoid driving or operating machinery until you know how it affects you.","Avoid alcohol consumption.","Monitor blood sugar regularly as this medicine is used in diabetic patients.","Do not stop taking this medicine without consulting your doctor.","Inform your doctor if you are pregnant, planning to become pregnant, or breastfeeding."]

🤱 Lactation Safety

It is not known whether Epalrestat passes into breast milk. Consult your doctor before breastfeeding while taking this medicine.

💊 Overdose Management

If you suspect an overdose, seek immediate medical attention. Symptoms of overdose may include severe nausea, vomiting, dizziness, and liver toxicity. Treatment is supportive and symptomatic.

⏰ Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule. Do not double the dose.

Additional Safety Advice

General Safety

Before starting this medicine, tell your doctor if you have any liver or kidney disease, as dose adjustments may be needed. Do not take this medicine if you are pregnant, planning to become pregnant, or breastfeeding without consulting your doctor, as the safety in these conditions is not well established. Avoid consuming alcohol while taking this medicine, as it may increase the risk of liver problems and worsen side effects. Take this medicine exactly as prescribed by your doctor, and do not change the dose or stop taking it without medical advice. If you miss a dose, take it as soon as you remember, but if it is almost time for your next dose, skip the missed dose and continue with your regular schedule. Do not double the dose to make up for a missed one. Keep this medicine out of reach of children and store it in a cool, dry place away from direct sunlight. Regularly monitor your blood sugar levels and attend follow-up appointments as scheduled. If you experience any unusual symptoms such as severe abdominal pain, yellowing of the eyes or skin, or difficulty breathing, seek immediate medical attention.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients may be more sensitive to the effects of this medicine. Dose adjustments may be needed based on kidney and liver function. Regular monitoring is advised.

🤰 Pregnancy Planning (TTC)

If you are planning to become pregnant, consult your doctor before taking this medicine. The safety of this medicine during pregnancy is not well established.

🏥 Post-Surgery Considerations

Inform your surgeon and anesthesiologist that you are taking this medicine before any surgery. It may need to be stopped temporarily.

🦷 Dental Procedures

Inform your dentist that you are taking this medicine before any dental procedure. No specific precautions are known, but it is important for your dentist to know your medication history.

💚 Lifestyle Tips for Better Results

🏃
Maintain a healthy weight to reduce nerve stress.
🥗
Regular low-impact exercise like walking or swimming.
😴
Practice good foot care and inspect feet daily.
💧
Include anti-inflammatory foods in your diet.
🧘
Get adequate sleep to support nerve health.
🌞
Avoid smoking as it worsens nerve damage.

🏋️ Exercise Considerations

Exercise is generally safe while taking this medicine, but if you experience dizziness, avoid strenuous activities until you know how the medicine affects you. Always warm up and cool down.

🥗 Diet Recommendations

Include omega-3 rich foods like fish and flaxseeds.
Reduce processed and high-sugar foods.
Stay well hydrated.
Eat plenty of fruits and vegetables.
Limit alcohol intake.

💼 Impact on Daily Work & Life

This medicine may cause dizziness in some people. Avoid driving or operating heavy machinery until you know how it affects you. Otherwise, it should not significantly impact your daily activities.

🛑 When to Stop This Medicine

Do not stop taking this medicine without consulting your doctor. If you experience serious side effects like liver problems or severe allergic reactions, seek immediate medical advice. Your doctor will decide if and when to stop the medicine.

📅 Long-Term Use Effects

Long-term use of this medicine may require regular monitoring of liver and kidney function. It is generally well-tolerated, but rare liver toxicity can occur. Periodic blood tests are advised. Do not stop the medicine without consulting your doctor, as symptoms may return.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Tight blood sugar control

Maintaining optimal blood sugar levels is the cornerstone of managing diabetic neuropathy.

Evidence: Well-established
Physical therapy

Can help improve mobility and reduce pain.

Evidence: Moderate
Alpha-lipoic acid

An antioxidant that may help with neuropathic symptoms.

Evidence: Moderate

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

No specific vaccine interactions are known. However, inform your doctor about all medicines before receiving any vaccine.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate unless specified

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✈️ Traveling with This Medicine

When traveling, carry this medicine in its original packaging along with a copy of your prescription. Store it in a cool, dry place away from direct sunlight. If crossing time zones, continue taking your dose at the same time each day as close as possible. Check customs regulations for carrying prescription medicines. Always carry enough supply for the duration of your trip.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 55-year-old man with type 2 diabetes and peripheral neuropathy
He had been experiencing tingling and burning in his feet for over a year. His doctor prescribed this medicine along with his regular diabetes medications. After about 8 weeks, he noticed a significant reduction in the burning sensation and improved sleep. He emphasized taking the tablet with breakfast to avoid stomach upset.
💡 Lesson: Consistent use and good blood sugar control are key to managing neuropathy symptoms.
👤 A 62-year-old woman with diabetic neuropathy and mild kidney impairment
She was started on this medicine at a lower dose due to her kidney function. She experienced mild nausea initially but it subsided after taking it with food. Her symptoms improved gradually over 3 months. Regular monitoring of kidney function was done.
💡 Lesson: Dose adjustments and monitoring are important in patients with kidney problems.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: It may take several weeks to months to notice improvement in symptoms. Continue taking it as prescribed.

Q: Can I take it with other diabetes medicines?

A: Yes, but inform your doctor as dose adjustments may be needed to avoid low blood sugar.

Q: Is it safe for long-term use?

A: It can be used long-term under medical supervision with regular monitoring of liver and kidney function.

Q: What should I do if I miss a dose?

A: Take it as soon as you remember, but if it's almost time for the next dose, skip the missed dose. Do not double dose.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?

🔄 Substitutes for listap 150 sr tablet

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: Epalrestat can cure diabetic neuropathy completely.
    Fact: Epalrestat helps manage symptoms and slow progression but does not cure the condition. Good blood sugar control remains essential.
  • Myth: Epalrestat can be taken without a doctor's prescription.
    Fact: Epalrestat is a prescription medicine and should only be taken under medical supervision.
  • Myth: Epalrestat works immediately.
    Fact: It may take several weeks to months to notice improvement.

🔄 Alternative Options

Generic Alternatives

  • Epalrestat 150 mg tablet

Brand Alternatives

  • Epstat 150mg Tablet SR

📊 Comparison with Similar Medicines

[{"medicine":"Epalrestat","class":"Aldose reductase inhibitor","primary_use":"Diabetic neuropathy","route":"Oral"},{"medicine":"Pregabalin","class":"Anticonvulsant","primary_use":"Neuropathic pain","route":"Oral"},{"medicine":"Gabapentin","class":"Anticonvulsant","primary_use":"Neuropathic pain","route":"Oral"}]

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