kool 5mg/1mg tablet - Chlordiazepoxide (5mg) + Trifluoperazine (1mg) medicine

Kool 5mg/1mg Tablet: Complete Information on Uses, Side Effects, and Safety

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🏭 Alembic Pharmaceuticals Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 25, 2026
🤰 Pregnancy Category Not established from the available information. Use in pregnancy only if clearly needed and under medical supervision. Both Chlordiazepoxide and Trifluoperazine may pose risks to the fetus. 📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Evidence: Moderate for short-term use in anxiety with agitation; limited for long-term use.
Reviewed by
SaathiMed Expert Panel | Sep 25, 2026
🩺
Medically Fact-Checked & Clinically Verified by SaathiMed Clinical Review Board
Clinical Reference Standards: CDSCO (Central Drugs Standard Control Organisation), Indian Pharmacopoeia (IP) & WHO | Last Updated: September 2026

When to Call Your Doctor IMMEDIATELY

  • High fever with muscle rigidity and confusion
  • Involuntary movements of the face, tongue, or limbs
  • Severe dizziness or fainting
  • Palpitations or irregular heartbeat
  • Yellowing of skin or eyes
  • Unusual bruising or bleeding
  • Difficulty breathing or swallowing
  • Severe abdominal pain

If experiencing severe symptoms, call emergency services immediately.

What is kool 5mg/1mg tablet used for?

This medicine is a combination of Chlordiazepoxide (a benzodiazepine) and Trifluoperazine (an antipsychotic) used for short-term treatment of severe anxiety with agitation or psychotic features. It works by enhancing GABA and blocking dopamine. It can cause drowsiness, dependence, and serious side effects, so it must be used under strict medical supervision.

  • Generic Name: Chlordiazepoxide (5mg) + Trifluoperazine (1mg)
  • Manufacturer: Alembic Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 kool 5mg/1mg tablet के बारे में (Hindi Summary)

उपयोग: यह दवा चिंता, बेचैनी और मानसिक तनाव के इलाज के लिए इस्तेमाल की जाती है। यह उन मरीजों के लिए है जिनमें चिंता के साथ-साथ मानसिक विकार या अत्यधिक बेचैनी के लक्षण भी होते हैं। यह दवा दिमाग में शांति लाने और मानसिक संतुलन बनाने में मदद करती है। इसे डॉक्टर की सलाह के बिना शुरू या बंद नहीं करना चाहिए।

साइड इफेक्ट्स: इस दवा के सामान्य दुष्प्रभावों में नींद आना, चक्कर आना, मुँह सूखना, धुंधला दिखना और कब्ज शामिल हैं। गंभीर दुष्प्रभावों में मांसपेशियों में अकड़न, कंपन, चेहरे की अनैच्छिक हरकतें, तेज बुखार, भ्रम और दिल की धड़कन में गड़बड़ी हो सकती है। अगर आपको कोई भी गंभीर लक्षण दिखे तो तुरंत डॉक्टर से संपर्क करें।

सुरक्षा सलाह: इस दवा को डॉक्टर के बताए अनुसार ही लें। इसे अचानक बंद न करें, क्योंकि इससे withdrawal के लक्षण हो सकते हैं। दवा लेते समय गाड़ी चलाने या मशीन चलाने से बचें क्योंकि इससे नींद और चक्कर आ सकते हैं। शराब का सेवन बिल्कुल न करें। अगर आपको कोई गंभीर दुष्प्रभाव दिखे तो तुरंत डॉक्टर को बताएं।

💡 Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

💊 kool 5mg/1mg tablet Uses & Benefits

[{"condition":"Anxiety disorders with agitation","description":"Used for short-term relief of severe anxiety that is accompanied by agitation, tension, or psychotic symptoms.","evidence":"Well-established for short-term use"},{"condition":"Psychotic disorders with anxiety","description":"Helps manage anxiety and agitation in patients with schizophrenia or other psychotic disorders.","evidence":"Limited evidence, used as adjunct"}]

Off-label uses: [{"condition":"Acute mania","description":"Sometimes used off-label for rapid calming in acute manic episodes, but not first-line.","evidence":"Limited"}]

Primary treatment for: Anxiety disorders with agitation

Also treats: Psychotic disorders, Schizophrenia, Bipolar disorder

📋 Drug Information

Generic Name(s)Chlordiazepoxide (5mg) + Trifluoperazine (1mg)
Brand Namekool 5mg/1mg tablet
ManufacturerAlembic Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action Class
Route of AdministrationOral
StorageStore at room temperature (15-30°C) in a dry place, away from direct sunlight and moisture. Keep in the original container.
Shelf Life24 months from the date of manufacture.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Take this medicine exactly as prescribed; do not adjust the dose on your own.
2
Avoid driving or operating heavy machinery until you know how this medicine affects you.
3
Do not consume alcohol while taking this medicine, as it can cause dangerous sedation.
4
Do not stop this medicine abruptly; your doctor will taper the dose gradually.
5
Report any unusual movements, fever, or mood changes to your doctor immediately.
6
Keep all follow-up appointments for monitoring of blood counts, liver function, and heart rhythm.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

✅
Severe anxiety with agitation
This medicine is commonly prescribed for this.
Likely Use
✅
Psychotic symptoms
May be used as an adjunct in psychotic disorders.
Likely Use
❌
Fever
This medicine is not a primary fever reducer.
Not Primary
❌
Headache
Not a primary treatment for headache.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionChlordiazepoxide is well absorbed from the gastrointestinal tract after oral administration. Trifluoperazine is also absorbed from the gastrointestinal tract. Food may slightly delay absorption but does not significantly affect the extent.
DistributionChlordiazepoxide is widely distributed throughout the body and crosses the blood-brain barrier and placenta. Trifluoperazine is highly lipophilic and distributes extensively into tissues, including the brain.
Protein BindingChlordiazepoxide is approximately 96% bound to plasma proteins. Trifluoperazine is approximately 90-99% bound to plasma proteins.
MetabolismChlordiazepoxide is metabolized in the liver by cytochrome P450 enzymes, primarily CYP3A4, into active metabolites including desmethylchlordiazepoxide and demoxepam. Trifluoperazine is metabolized in the liver, primarily by CYP1A2 and CYP3A4, into various metabolites.
Half-LifeChlordiazepoxide: 5-30 hours (active metabolites up to 100 hours). Trifluoperazine: approximately 10-20 hours.
ExcretionChlordiazepoxide and its metabolites are excreted primarily in the urine. Trifluoperazine and its metabolites are excreted in urine and feces.
BioavailabilityChlordiazepoxide: approximately 100% (oral). Trifluoperazine: approximately 40-50% (oral).
Onset of ActionAnxiolytic and sedative effects of Chlordiazepoxide begin within 30-60 minutes. Antipsychotic effects of Trifluoperazine may take several days to weeks to fully manifest.
Peak Plasma TimeChlordiazepoxide: 1-4 hours. Trifluoperazine: 2-4 hours.
Duration of ActionChlordiazepoxide: 6-12 hours (due to active metabolites, effects may last longer). Trifluoperazine: 12-24 hours.

How It Works

This medicine combines two active ingredients with different mechanisms. Chlordiazepoxide is a benzodiazepine that binds to the GABA-A receptor, enhancing the inhibitory effect of GABA, which leads to sedation, anxiety relief, and muscle relaxation. Trifluoperazine is a typical antipsychotic that blocks dopamine D2 receptors in the brain, reducing psychotic symptoms and agitation. It also has anticholinergic and antihistaminic effects, contributing to sedation and calming.

Mechanism Steps

1
GABA-A receptor binding: Chlordiazepoxide binds to the benzodiazepine site on the GABA-A receptor, increasing the frequency of chloride channel opening and enhancing GABA-mediated inhibition.
2
Dopamine D2 receptor blockade: Trifluoperazine blocks dopamine D2 receptors in the mesolimbic and mesocortical pathways, reducing psychotic symptoms and agitation.
3
Combined effect: The combination provides rapid relief of anxiety and agitation while addressing psychotic features, but also increases the risk of sedation and extrapyramidal symptoms.

💡 How to Take kool 5mg/1mg tablet

Strength: Tablet containing Chlordiazepoxide 5 mg and Trifluoperazine 1 mg.

1Take this medicine exactly as prescribed by your doctor.
2Swallow the tablet whole with a glass of water.
3Take with food to reduce stomach upset.
4Do not crush, chew, or break the tablet unless instructed.
5Take at the same time each day to maintain consistent levels.
6Do not stop taking this medicine suddenly without consulting your doctor.

Dosage Information

Adult DosageThe dosage of this medicine must be individualized by a qualified clinician based on the indication, severity of symptoms, age, weight, renal and hepatic function, and response to treatment. Typically, one tablet is taken 1 to 2 times daily, but the exact dose and frequency will be determined by your doctor. Do not self-adjust the dose. The maximum daily dose should not exceed what is prescribed. Regular follow-up is necessary to assess efficacy and side effects.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician.
Elderly DosageElderly patients are more sensitive to the effects of this medicine. Start with a lower dose and titrate slowly. Increased risk of falls, confusion, and cognitive impairment. Use with caution and monitor closely.
Renal ImpairmentUse with caution in patients with renal impairment. Dose adjustment may be necessary. Consult your doctor.
Hepatic ImpairmentUse with caution in patients with hepatic impairment. Dose adjustment may be necessary. Avoid in severe liver disease.
Maximum Daily DoseThe maximum daily dose is determined by the prescribing clinician based on individual patient factors. Do not exceed the prescribed dose.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With food
Take with meals
Reduces stomach upset and may improve tolerability.
Grapefruit juice
Avoid
May increase drug levels by inhibiting CYP3A4.
Alcohol
Avoid completely
Increases sedation and CNS depression.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of kool 5mg/1mg tablet

✅ Common Side Effects

Drowsiness (Common (10-30%))
Avoid driving or operating machinery. Usually improves with continued use.
Dizziness (Common (5-15%))
Rise slowly from sitting or lying position. Consult doctor if persistent.
Dry mouth (Common (10-20%))
Sip water, chew sugarless gum. Usually temporary.
Blurred vision (Common (5-10%))
Avoid driving if vision is affected. Consult doctor if persistent.
Constipation (Common (5-10%))
Increase fiber and fluid intake. Consult doctor if severe.

🚨 Serious Side Effects

Extrapyramidal symptoms (tremors, rigidity, bradykinesia) (Uncommon (1-5%))
Contact doctor immediately. May require dose adjustment or additional medication.
Tardive dyskinesia (involuntary movements) (Rare (<1%))
Report to doctor immediately. May be irreversible.
Neuroleptic malignant syndrome (fever, rigidity, confusion) (Rare (<0.1%))
Seek emergency medical attention immediately.
Agranulocytosis (low white blood cell count) (Rare (<0.1%))
Report any signs of infection (fever, sore throat) immediately.
QT prolongation (heart rhythm abnormality) (Rare (<0.1%))
Seek medical attention if you experience palpitations, fainting, or shortness of breath.

⚠️ Rare Side Effects

Jaundice
Report yellowing of skin or eyes to doctor immediately.
Blood dyscrasias
Regular blood tests may be needed. Report unusual bruising or bleeding.
Photosensitivity
Use sunscreen and protective clothing when outdoors.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Warfarin Moderate
Opioids Major
MAO inhibitors Major
Amiodarone Major
Ketoconazole Moderate
Rifampin Moderate
Antacids Minor
Caffeine Minor
Levodopa Moderate
Lithium Moderate

🚨 Major Interactions

  • CNS depressants (e.g., opioids, alcohol, barbiturates)
  • MAO inhibitors
  • QT-prolonging drugs (e.g., amiodarone, sotalol, haloperidol)

⚡ Moderate Interactions

  • CYP3A4 inhibitors (e.g., ketoconazole, clarithromycin)
  • CYP3A4 inducers (e.g., rifampin, carbamazepine)
  • Antihypertensive drugs

🍷 Alcohol Interaction

Alcohol should be completely avoided while taking this medicine. Alcohol increases the sedative and CNS depressant effects of Chlordiazepoxide and Trifluoperazine, leading to excessive drowsiness, dizziness, impaired coordination, respiratory depression, and increased risk of accidents. It can also worsen underlying psychiatric conditions.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Hypersensitivity to Chlordiazepoxide, Trifluoperazine, or any component of the formulation","Severe liver disease","Severe kidney disease","Acute narrow-angle glaucoma","Prostatic hypertrophy or urinary retention","Parkinson's disease","Myasthenia gravis","Severe cardiovascular disease","Coma or CNS depression","Pregnancy and breastfeeding"]

⚠️ Warnings & Precautions

["This medicine can cause severe drowsiness; avoid driving or operating machinery.","Do not stop abruptly; withdrawal symptoms may occur.","May cause dependence and tolerance with prolonged use.","Use with caution in elderly patients; increased risk of falls and confusion.","May cause extrapyramidal symptoms; report any unusual movements.","Avoid alcohol and other CNS depressants.","May cause blood disorders; regular monitoring required.","May prolong QT interval; caution in patients with cardiac disease.","Not recommended for children.","Use with caution in patients with a history of substance abuse."]

🤱 Lactation Safety

Chlordiazepoxide and Trifluoperazine are excreted in breast milk. Breastfeeding is not recommended while taking this medicine due to potential serious adverse effects in the infant, including sedation and developmental issues.

💊 Overdose Management

Overdose can cause severe drowsiness, confusion, coma, respiratory depression, hypotension, and cardiac arrhythmias. Seek emergency medical attention immediately. Treatment is supportive and symptomatic. Gastric lavage may be considered if within 1-2 hours of ingestion. Flumazenil may be used for benzodiazepine overdose but is contraindicated in mixed overdose with tricyclic antidepressants or antipsychotics due to risk of seizures. Monitor vital signs, ECG, and electrolytes.

⏰ Missed Dose

If you miss a dose, take it as soon as you remember. If it is almost time for your next dose, skip the missed dose and continue with your regular schedule. Do not double the dose to catch up.

Additional Safety Advice

General Safety

Take this medicine exactly as prescribed by your doctor. Do not increase or decrease the dose without consulting your doctor. Avoid driving or operating heavy machinery until you know how this medicine affects you, as it can cause drowsiness and dizziness. Do not drink alcohol while taking this medicine, as it can increase sedation and other side effects. This medicine can be habit-forming; use it only for the duration prescribed. Do not stop taking this medicine suddenly, as it can cause withdrawal symptoms. Inform your doctor if you have a history of liver disease, kidney disease, heart problems, glaucoma, or prostate issues. Regular monitoring of blood counts, liver function, and heart rhythm may be required. Keep this medicine out of reach of children.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients are more sensitive to the sedative and extrapyramidal effects of this medicine. Start with a lower dose and monitor closely for falls, confusion, and cognitive impairment. Avoid long-term use if possible.

🤰 Pregnancy Planning (TTC)

This medicine is not recommended during pregnancy or when planning pregnancy. Both Chlordiazepoxide and Trifluoperazine may harm the fetus. Consult your doctor for alternative treatments and contraception advice.

🏥 Post-Surgery Considerations

This medicine may interact with anesthetics and other medications used during surgery. Inform your surgeon and anesthesiologist that you are taking this medicine. It may need to be stopped before surgery to avoid complications.

🦷 Dental Procedures

Inform your dentist that you are taking this medicine. It can cause dry mouth, which may increase the risk of dental problems. Also, it may interact with sedatives or anesthetics used during dental procedures.

💚 Lifestyle Tips for Better Results

🏃
Maintain a regular sleep schedule to support mental health.
🥗
Engage in relaxation techniques such as deep breathing or meditation.
😴
Avoid caffeine and stimulants that can worsen anxiety.
💧
Stay physically active with low-impact exercises like walking or yoga.
🧘
Avoid alcohol and recreational drugs.
🌞
Keep a symptom diary to track your progress and side effects.

🏋️ Exercise Considerations

This medicine can cause drowsiness and dizziness, which may affect your coordination. Avoid strenuous exercise or activities that require alertness until you know how the medicine affects you. Light to moderate exercise is generally safe but consult your doctor first.

🥗 Diet Recommendations

Eat a balanced diet rich in fruits, vegetables, and whole grains.
Include omega-3 fatty acids from fish or flaxseed.
Limit processed foods and added sugars.
Stay well hydrated by drinking plenty of water.
Avoid grapefruit and grapefruit juice.

💼 Impact on Daily Work & Life

This medicine can cause significant drowsiness and dizziness, which may impair your ability to drive, operate machinery, or perform tasks requiring mental alertness. It is advisable to avoid such activities until you know how the medicine affects you. Discuss with your employer if you need temporary adjustments.

🛑 When to Stop This Medicine

Do not stop this medicine abruptly. Your doctor will gradually reduce the dose to prevent withdrawal symptoms. If you experience severe side effects, contact your doctor immediately for guidance on tapering or switching to another medicine.

📅 Long-Term Use Effects

Long-term use of this medicine can lead to tolerance, dependence, and withdrawal symptoms. Trifluoperazine may cause tardive dyskinesia, which can be irreversible. Regular monitoring of blood counts, liver function, and heart rhythm is necessary. Periodic evaluation of the need for continued treatment is recommended.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Cognitive behavioral therapy (CBT)

Effective for anxiety disorders and can reduce the need for long-term medication.

Evidence: Well-established
Relaxation techniques

Deep breathing, meditation, and yoga can help manage anxiety.

Evidence: Moderate
Selective serotonin reuptake inhibitors (SSRIs)

First-line for chronic anxiety; safer for long-term use.

Evidence: Well-established

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

Not established from the available information. Consult your doctor regarding vaccination timing while on this medicine.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate unless specified

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✈️ Traveling with This Medicine

When traveling, carry this medicine in its original packaging along with a copy of your prescription. Keep it in your hand luggage to avoid loss. Store at room temperature and protect from extreme heat or moisture. If crossing time zones, consult your doctor about adjusting the dosing schedule. Check local customs regulations regarding controlled substances, as this medicine may be regulated.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 35-year-old woman with severe anxiety and agitation
She was prescribed this medicine for short-term management of anxiety with agitation. After starting, she felt calmer within a few days but experienced drowsiness. Her doctor advised her to take it at bedtime and avoid driving. She was gradually tapered off after 4 weeks and referred for cognitive behavioral therapy.
💡 Lesson: This medicine is effective for short-term symptom control but should be used with caution and gradually tapered to avoid withdrawal.
👤 A 60-year-old man with psychotic disorder and anxiety
He was started on this medicine as an adjunct to his antipsychotic treatment. His agitation improved, but he developed mild tremors. His doctor adjusted the dose and monitored him closely. He was advised not to stop the medicine suddenly.
💡 Lesson: Regular monitoring and dose adjustment are essential to balance efficacy and side effects, especially in older adults.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: The sedative and anxiolytic effects may begin within 30-60 minutes, but the full antipsychotic effect may take several days to weeks.

Q: Can I take this medicine if I have liver disease?

A: This medicine should be used with caution in liver disease. Your doctor may adjust the dose or avoid it in severe liver disease.

Q: Is this medicine habit-forming?

A: Yes, Chlordiazepoxide can cause dependence. It should be used short-term and tapered gradually under medical supervision.

Q: What should I do if I miss a dose?

A: Take it as soon as you remember if it's not too close to the next dose. Otherwise, skip it and continue with your regular schedule. Do not double dose.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?
  • Is it safe to take during pregnancy?
  • How do I stop this medicine safely?

🔄 Substitutes for kool 5mg/1mg tablet

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: This medicine is a cure for anxiety.
    Fact: This medicine only manages symptoms and is not a cure. It is usually used short-term along with therapy.
  • Myth: It is safe to stop this medicine suddenly.
    Fact: Abrupt discontinuation can cause severe withdrawal symptoms. Always taper under medical supervision.
  • Myth: This medicine is safe to take with alcohol.
    Fact: Alcohol increases the sedative effects and can be dangerous. Avoid alcohol completely.

🔄 Alternative Options

Generic Alternatives

  • Chlordiazepoxide + Trifluoperazine combination tablets from other manufacturers

📊 Comparison with Similar Medicines

[{"medicine":"This medicine","composition":"Chlordiazepoxide 5 mg + Trifluoperazine 1 mg","primary_use":"Anxiety with agitation","sedation":"High","dependence_risk":"High"},{"medicine":"Chlordiazepoxide + Amitriptyline","composition":"Chlordiazepoxide + Amitriptyline","primary_use":"Anxiety with depression","sedation":"High","dependence_risk":"High"},{"medicine":"Diazepam + Trifluoperazine","composition":"Diazepam + Trifluoperazine","primary_use":"Anxiety with psychosis","sedation":"High","dependence_risk":"High"}]

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