irinores 40mg injection - Irinotecan (40mg) medicine

Ertikan 40mg Injection (Irinotecan): Comprehensive Medicine Guide

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🏭 Resonance Laboratories Pvt Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 26, 2026
⚠️ Hepatotoxicity Risk ⚠️ Nephrotoxicity Risk 🤰 Pregnancy Category This medicine can cause fetal harm when administered to a pregnant woman. It is not recommended during pregnancy. Women of childbearing potential should use effective contraception during treatment and for a period after the last dose. If pregnancy occurs during treatment, immediate medical advice should be sought. 📋 Prescription Required 💊 Generic Available
Medically Reviewed
12 min read
Evidence: Well-established for colorectal cancer; limited for other uses.
Reviewed by
SaathiMed Expert Panel | Sep 26, 2026
🩺
Medically Fact-Checked & Clinically Verified by SaathiMed Clinical Review Board
Clinical Reference Standards: CDSCO (Central Drugs Standard Control Organisation), Indian Pharmacopoeia (IP) & WHO | Last Updated: September 2026

When to Call Your Doctor IMMEDIATELY

  • Fever of 100.4°F (38°C) or higher, with or without chills
  • Severe diarrhoea (more than 6 stools per day) or diarrhoea with blood
  • Signs of dehydration: dizziness, decreased urination, dry mouth
  • Unusual bleeding or bruising
  • Shortness of breath, chest pain, or swelling in legs
  • Yellowing of skin or eyes, dark urine
  • Severe abdominal pain

If experiencing severe symptoms, call emergency services immediately.

What is irinores 40mg injection used for?

This medicine contains Irinotecan 40 mg and is a chemotherapy injection used mainly for advanced colorectal cancer. It works by blocking an enzyme that cancer cells need to divide. It is given intravenously by a healthcare professional and can cause side effects like diarrhoea, low blood counts, and hair loss.

  • Generic Name: Irinotecan (40mg)
  • Manufacturer: Resonance Laboratories Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 irinores 40mg injection के बारे में (Hindi Summary)

उपयोग: यह दवा इरिनोटेकान 40 मिलीग्राम इंजेक्शन के रूप में एक कीमोथेरेपी दवा है। इसका उपयोग मुख्य रूप से उन्नत कोलोरेक्टल कैंसर (आंत के कैंसर) के इलाज के लिए किया जाता है। यह कैंसर कोशिकाओं को बढ़ने और विभाजित होने से रोकती है। यह दवा केवल डॉक्टर या नर्स द्वारा नस के माध्यम से दी जाती है। इसे घर पर स्वयं न लें। यह दवा अन्य कैंसर जैसे अग्नाशय और फेफड़ों के कैंसर में भी कभी-कभी उपयोग की जाती है।

साइड इफेक्ट्स: आम दुष्प्रभावों में दस्त, मतली, उल्टी, पेट दर्द, भूख न लगना, मुँह के छाले, बालों का झड़ना, थकान और रक्त कोशिकाओं की कमी शामिल हैं। गंभीर दुष्प्रभावों में गंभीर दस्त, बुखार के साथ कम श्वेत रक्त कोशिकाएं, रक्तस्राव, और एलर्जी प्रतिक्रिया शामिल हैं। कोई भी दुष्प्रभाव होने पर तुरंत डॉक्टर को बताएं।

सुरक्षा सलाह: यह दवा केवल योग्य स्वास्थ्य पेशेवर द्वारा ही दी जानी चाहिए। इसे स्वयं न लें। उपचार के दौरान गर्भनिरोधक उपाय करें। स्तनपान न कराएं। पर्याप्त पानी पिएं। बुखार, ठंड लगना, गंभीर दस्त, या सांस लेने में कठिनाई होने पर तुरंत डॉक्टर से संपर्क करें।

💡 Did You Know? India has the highest number of USFDA-compliant plants outside the USA.

💊 irinores 40mg injection Uses & Benefits

[{"condition":"Metastatic colorectal cancer","description":"Used as part of combination chemotherapy or as a single agent for advanced colorectal cancer after other treatments have failed.","evidence":"Well-established"},{"condition":"Metastatic pancreatic cancer","description":"Sometimes used in combination regimens for advanced pancreatic cancer, though this is not a primary approved use in all regions.","evidence":"Limited"},{"condition":"Small cell lung cancer","description":"May be used in some chemotherapy regimens for extensive-stage small cell lung cancer.","evidence":"Limited"},{"condition":"Gastric cancer","description":"Occasionally used in combination therapy for advanced gastric or gastroesophageal junction cancer.","evidence":"Limited"}]

Off-label uses: [{"condition":"Ewing sarcoma","description":"Sometimes used in combination regimens for Ewing sarcoma, a rare bone cancer.","evidence":"Limited"},{"condition":"Brain tumors","description":"Investigated in some high-grade gliomas, but not standard of care.","evidence":"Limited"}]

Primary treatment for: Metastatic colorectal cancer

Also treats: Metastatic pancreatic cancer, Small cell lung cancer, Gastric cancer

📋 Drug Information

Generic Name(s)Irinotecan (40mg)
Brand Nameirinores 40mg injection
ManufacturerResonance Laboratories Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI NEOPLASTICS
Action ClassTopoisomerase Inhibitor
Route of AdministrationParenteral (intravenous infusion)
StorageStore vials in a refrigerator at 2°C to 8°C (36°F to 46°F). Protect from light. Do not freeze. Once diluted for infusion, the solution should be used within a specified time as per institutional guidelines.
Shelf LifeThe shelf life of the unopened vial is typically 24 months from the date of manufacture. Check the expiry date on the packaging.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Administer this medicine only in a facility equipped to manage severe allergic reactions and extravasation.
2
Pre-medicate with antiemetics as prescribed to reduce nausea and vomiting.
3
Instruct patients to report diarrhoea immediately, especially if it occurs more than 24 hours after infusion.
4
Monitor complete blood counts before each cycle and adjust dose based on toxicity.
5
Consider UGT1A1 genotyping in patients with a history of severe toxicity.
6
Advise patients to use effective contraception during and after treatment.
7
Avoid live vaccines during treatment.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

✅
Advanced colorectal cancer
This medicine is commonly prescribed for this condition.
Likely Use
❌
Fever
This medicine is not a fever reducer; fever may indicate infection and requires immediate medical attention.
Not Primary
❌
Diarrhoea
Diarrhoea is a side effect of this medicine, not a reason to use it.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionThis medicine is administered intravenously, so absorption from the gastrointestinal tract is not applicable. The drug is directly introduced into the bloodstream.
DistributionIrinotecan and its active metabolite SN-38 distribute widely into body tissues. Plasma protein binding of irinotecan is moderate, and SN-38 is highly bound to albumin.
Protein BindingIrinotecan is approximately 30-68% bound to plasma proteins, while SN-38 is about 95% bound to human serum albumin.
MetabolismIrinotecan is metabolized primarily in the liver by carboxylesterases to SN-38. SN-38 is further glucuronidated by UGT1A1 to an inactive glucuronide. Irinotecan is also metabolized by CYP3A4 to inactive metabolites.
Half-LifeThe elimination half-life of irinotecan is approximately 6 to 12 hours, and that of SN-38 is about 10 to 20 hours.
ExcretionIrinotecan and its metabolites are excreted mainly in bile and urine. About 20-50% of the dose is excreted in urine, and the remainder in feces via bile.
BioavailabilityNot applicable for intravenous administration, as the drug is given directly into the bloodstream.
Onset of ActionThe cytotoxic effects begin after the drug is converted to SN-38, which occurs within hours of infusion. However, clinical effects such as tumor shrinkage are seen over weeks.
Peak Plasma TimePeak plasma concentration is reached at the end of the intravenous infusion.
Duration of ActionThe cytotoxic effect persists as long as SN-38 remains in the body, typically for several days after a dose. The dosing schedule is usually every 1 to 3 weeks to allow recovery of normal tissues.

How It Works

Irinotecan is a prodrug that is converted in the body to its active metabolite, SN-38. SN-38 binds to and inhibits topoisomerase I, an enzyme that relieves torsional stress in DNA during replication. By blocking topoisomerase I, SN-38 causes single-strand DNA breaks to accumulate, which leads to arrest of DNA replication and cell death, particularly in rapidly dividing cancer cells.

Mechanism Steps

1
Prodrug conversion: Irinotecan is converted by carboxylesterases in the liver and other tissues to the active metabolite SN-38.
2
Topoisomerase I inhibition: SN-38 binds to the topoisomerase I-DNA complex and prevents the enzyme from re-ligating the DNA strand.
3
DNA damage: This leads to single-strand DNA breaks that accumulate during DNA replication.
4
Cell cycle arrest and apoptosis: The DNA damage triggers cell cycle arrest and programmed cell death, primarily in rapidly dividing cancer cells.

💡 How to Take irinores 40mg injection

Strength: Injection: 40 mg per vial (as irinotecan hydrochloride).

1This medicine is given by a healthcare professional in a clinic or hospital setting.
2It is administered as an intravenous infusion over 90 minutes.
3You will be monitored for allergic reactions during and after the infusion.
4Drink plenty of fluids before and after the infusion to stay hydrated.
5Follow your doctor's instructions for pre-medications to prevent nausea and vomiting.
6Report any side effects to your healthcare team immediately.

Dosage Information

Adult DosageThe dose of this medicine is highly individualized and depends on the type of cancer, the treatment regimen, and the patient's overall health. It is usually given as an intravenous infusion over 90 minutes. Common regimens include 350 mg/m² every 3 weeks as a single agent, or 180 mg/m² every 2 weeks in combination with other chemotherapy drugs. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function, and blood counts.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatric oncologist.
Elderly DosageElderly patients (65 years and older) may be more sensitive to the effects of this medicine, especially diarrhoea and bone marrow suppression. Doses may need to be reduced or given less frequently. Close monitoring is required.
Renal ImpairmentNo specific dose adjustment is recommended for patients with mild to moderate renal impairment. However, caution is advised in severe renal impairment, and close monitoring is necessary.
Hepatic ImpairmentPatients with liver impairment may require dose reduction. For patients with bilirubin levels above the normal range, a reduced dose is often recommended. Consult the prescribing information for specific guidelines.
Maximum Daily DoseThe maximum recommended dose varies by regimen. As a single agent, the maximum is 350 mg/m² every 3 weeks. In combination regimens, the dose is lower. Do not exceed the dose prescribed by your doctor.

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

Grapefruit
Avoid
May increase drug levels and toxicity.
St. John's Wort
Avoid
May decrease drug efficacy.
Alcohol
Avoid
May worsen liver toxicity and dehydration.

⏰ What to Do If You Miss a Dose

📌 You miss an appointment for your infusion
→ Contact your treatment center as soon as possible to reschedule.
💡 Do not attempt to self-administer the missed dose.

⚠️ Side Effects of irinores 40mg injection

✅ Common Side Effects

Diarrhoea (Very common (>10%))
Drink plenty of fluids. Your doctor may prescribe loperamide. If diarrhoea is severe or persists beyond 24 hours, contact your doctor immediately.
Nausea and vomiting (Common (1-10%))
Take anti-nausea medicines as prescribed. Eat small, frequent meals. Inform your doctor if vomiting is severe.
Low white blood cell count (neutropenia) (Very common (>10%))
Your doctor will monitor your blood counts. Report any fever, sore throat, or signs of infection immediately.
Hair loss (Common (1-10%))
Hair usually grows back after treatment ends. Consider a wig or head covering if desired.
Fatigue (Common (1-10%))
Get plenty of rest. Pace your activities. Inform your doctor if fatigue is overwhelming.

🚨 Serious Side Effects

Severe diarrhoea with dehydration (Common (1-10%))
Seek immediate medical attention if you have more than 6 stools per day, blood in stool, or signs of dehydration such as dizziness, decreased urination, or dry mouth.
Febrile neutropenia (Common (1-10%))
Go to the emergency room immediately if you have a fever of 100.4°F (38°C) or higher, with or without chills.
Severe allergic reaction (anaphylaxis) (Rare (<0.1%))
Seek emergency help if you experience rash, itching, swelling of the face, lips, tongue, or throat, difficulty breathing, or a sudden drop in blood pressure.
Liver toxicity (Uncommon (0.1-1%))
Report yellowing of the skin or eyes, dark urine, or severe abdominal pain to your doctor immediately.
Interstitial lung disease (Rare (<0.1%))
Seek immediate medical attention if you develop new or worsening shortness of breath, cough, or fever.

⚠️ Rare Side Effects

Kidney failure
Report decreased urine output, swelling in legs, or confusion to your doctor immediately.
Blood clots
Seek emergency care if you have chest pain, shortness of breath, or swelling and pain in one leg.
Severe skin reactions
Report any severe rash, blistering, or peeling skin to your doctor immediately.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Ketoconazole Major
Rifampin Major
Warfarin Moderate
Atazanavir Major
Phenytoin Major
Carbamazepine Major
Clarithromycin Major
Gemfibrozil Major
Live vaccines Major
Diuretics Moderate

🚨 Major Interactions

  • Strong CYP3A4 inhibitors (e.g., ketoconazole, clarithromycin)
  • Strong CYP3A4 inducers (e.g., rifampin, carbamazepine, phenytoin)
  • UGT1A1 inhibitors (e.g., atazanavir, gemfibrozil)
  • Live vaccines

⚡ Moderate Interactions

  • Warfarin
  • Diuretics
  • Other myelosuppressive agents

🍷 Alcohol Interaction

Alcohol may worsen liver toxicity and increase the risk of dehydration from diarrhoea. It is best to avoid alcohol while receiving this medicine.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Severe bone marrow suppression","Severe liver impairment","Known severe hypersensitivity to irinotecan or any component of the formulation","Pregnancy (unless potential benefit justifies risk)","Breastfeeding"]

⚠️ Warnings & Precautions

["This medicine should be administered only under the supervision of a qualified oncologist.","Severe diarrhoea can occur and may be life-threatening. Early recognition and treatment are essential.","Febrile neutropenia is a serious complication. Monitor for fever and signs of infection.","Patients with UGT1A1*28 polymorphism may be at higher risk of severe toxicity.","Avoid live vaccines during treatment.","Use effective contraception during and after treatment.","Caution in patients with liver or kidney impairment.","Elderly patients may be more susceptible to toxicity."]

🤱 Lactation Safety

It is not known whether irinotecan is excreted in human milk. Because of the potential for serious adverse reactions in nursing infants, breastfeeding should be discontinued during treatment and for a period after the last dose, as advised by the doctor.

💊 Overdose Management

There is no known antidote for irinotecan overdose. Management should be symptomatic and supportive, including monitoring of blood counts, liver and kidney function, and treatment of diarrhoea and dehydration. In case of overdose, contact a poison control center or emergency room immediately.

⏰ Missed Dose

This medicine is given by a healthcare professional in a clinic or hospital setting. If you miss an appointment for your dose, contact your doctor or treatment center as soon as possible to reschedule. Do not attempt to self-administer a missed dose.

Additional Safety Advice

General Safety

This medicine must be given only by a qualified healthcare professional in a properly equipped facility. Do not attempt to administer it yourself. Inform your doctor if you have liver disease, kidney disease, bone marrow problems, or a history of severe diarrhoea. Use effective contraception during treatment and for a period after the last dose, as advised by your doctor. Avoid live vaccines while on this medicine. Drink plenty of fluids to prevent dehydration, especially if you have diarrhoea. Do not breastfeed while receiving this medicine. Keep all appointments for blood tests and follow-up visits. Tell your doctor immediately if you experience fever, chills, severe diarrhoea, unusual bleeding, or difficulty breathing.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Patients over 65 years of age may be more sensitive to the side effects of this medicine, especially diarrhoea and bone marrow suppression. Close monitoring and dose adjustments may be necessary.

🤰 Pregnancy Planning (TTC)

This medicine can cause harm to the fetus. Women of childbearing potential should use effective contraception during treatment and for a period after the last dose. Men should also use contraception. Discuss pregnancy planning with your doctor before starting treatment.

🏥 Post-Surgery Considerations

If you have recently had surgery, inform your doctor. This medicine may affect wound healing and increase the risk of bleeding or infection. Your doctor will decide the appropriate timing to start treatment after surgery.

🦷 Dental Procedures

Inform your dentist that you are receiving this medicine before any dental procedure. You may be at increased risk of bleeding or infection. Your dentist may recommend postponing non-urgent procedures until your blood counts recover.

💚 Lifestyle Tips for Better Results

🏃
Stay well hydrated by drinking plenty of fluids.
🥗
Eat small, frequent meals to manage nausea.
😴
Get adequate rest and pace your activities.
💧
Avoid people with infections to reduce risk of illness.
🧘
Practice good hand hygiene.
🌞
Use sunscreen and protective clothing when outdoors.

🏋️ Exercise Considerations

Mild to moderate exercise may help reduce fatigue, but avoid strenuous activities if you feel weak or dizzy. Consult your doctor before starting any exercise program.

🥗 Diet Recommendations

Eat a balanced diet rich in fruits and vegetables.
Include lean proteins to support healing.
Avoid raw or undercooked foods to prevent infections.
Limit spicy and greasy foods if you have diarrhoea.
Drink oral rehydration solutions if you have diarrhoea.

💼 Impact on Daily Work & Life

This medicine may cause fatigue, nausea, and other side effects that can affect your ability to work. Discuss with your employer about flexible hours or remote work options. Avoid driving or operating heavy machinery if you feel unwell.

🛑 When to Stop This Medicine

Do not stop this medicine without consulting your doctor. Treatment may be stopped or adjusted based on your response, side effects, or other medical conditions. Your doctor will decide the appropriate duration of therapy.

📅 Long-Term Use Effects

Long-term effects of this medicine may include persistent fatigue, increased risk of infections, and potential organ toxicity. Regular monitoring of blood counts, liver and kidney function is essential. Some patients may experience delayed effects such as secondary cancers, though this is rare. Discuss any long-term concerns with your oncologist.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Other chemotherapy regimens

Depending on your cancer type and prior treatments, other chemotherapy drugs or combinations may be options.

Evidence: Well-established
Targeted therapy

For some colorectal cancers, targeted therapies such as cetuximab or bevacizumab may be used.

Evidence: Well-established
Immunotherapy

In selected patients with certain genetic markers, immunotherapy may be an option.

Evidence: Limited

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

Live vaccines should be avoided during treatment with this medicine due to the risk of serious infections. Inactivated vaccines may be given, but their effectiveness may be reduced. Consult your doctor before receiving any vaccine.

📦 Storage Guide

✅ DO

Store in refrigerator at 2°C to 8°C

❌ DON'T

Do not freeze

✅ DO

Keep in original carton to protect from light

❌ DON'T

Do not use if the solution is discolored or contains particles

✅ DO

Follow institutional guidelines for diluted solution storage

❌ DON'T

Do not store diluted solution for longer than recommended

✈️ Traveling with This Medicine

This medicine is given in a healthcare setting, so travel is not applicable for administration. However, if you are traveling between treatment cycles, carry a copy of your prescription and medical records. Keep the medicine in its original packaging and store it in a cool, dry place. Check with your doctor about any travel restrictions and ensure you have access to medical care at your destination.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 58-year-old man with metastatic colorectal cancer
He received this medicine as part of a combination chemotherapy regimen. He experienced moderate diarrhoea after the first cycle, which was managed with loperamide and fluids. His doctor adjusted the dose for subsequent cycles. He advises other patients to keep a diary of bowel movements and report changes promptly.
💡 Lesson: Early reporting and management of diarrhoea can prevent serious complications and allow treatment to continue.
👤 A 62-year-old woman with advanced pancreatic cancer
She was treated with this medicine in combination with other drugs. She experienced fatigue and hair loss but found that resting and using a wig helped her cope. She emphasizes the importance of staying hydrated and eating small, frequent meals.
💡 Lesson: Supportive care and lifestyle adjustments can help manage side effects and improve quality of life during chemotherapy.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: The effects of this medicine on cancer cells begin soon after infusion, but measurable tumor shrinkage may take several weeks to months. Your doctor will monitor your response with regular scans and tests.

Q: Can I drive after receiving this medicine?

A: This medicine can cause fatigue, dizziness, or blurred vision. It is best to arrange for someone else to drive you to and from your treatment sessions and avoid driving if you feel unwell.

Q: Is it safe to take during pregnancy?

A: No, this medicine can harm the developing baby. It is not recommended during pregnancy. Use effective contraception during treatment and for a period after the last dose.

Q: What should I do if I experience diarrhoea?

A: Start taking loperamide as directed by your doctor and drink plenty of fluids. If diarrhoea is severe or persists beyond 24 hours, contact your doctor immediately.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine if I have liver problems?
  • Will this medicine affect my fertility?
  • Can I work while on this medicine?
  • How long will I need to take this medicine?
  • What should I do if I miss a dose?
  • Can I take other medicines while on this?

🔄 Substitutes for irinores 40mg injection

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: This medicine can be taken at home like a pill.
    Fact: This medicine is an injection that must be given by a healthcare professional in a clinic or hospital setting.
  • Myth: This medicine cures all types of cancer.
    Fact: This medicine is approved for specific cancers, mainly colorectal cancer, and is used as part of a comprehensive treatment plan.
  • Myth: Side effects mean the medicine is not working.
    Fact: Side effects are common with chemotherapy and do not indicate whether the medicine is working. Your doctor will monitor your response with tests.

🔄 Alternative Options

Generic Alternatives

  • Irinotecan generic injection

Brand Alternatives

  • Ertikan
  • Irinotel
  • Campto

📊 Comparison with Similar Medicines

[{"medicine":"Irinotecan","class":"Topoisomerase I inhibitor","route":"Intravenous","main_use":"Colorectal cancer"},{"medicine":"Topotecan","class":"Topoisomerase I inhibitor","route":"Intravenous or oral","main_use":"Ovarian, lung, cervical cancers"},{"medicine":"Oxaliplatin","class":"Platinum-based","route":"Intravenous","main_use":"Colorectal cancer"}]

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