dpm injection - Diazepam (NA) medicine

dpm injection - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Arrow Pharma ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 28, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 28, 2026

What is dpm injection used for?

Alzepam (Diazepam) is used to treat NEURO CNS. It contains Diazepam (NA), which Enhances GABA-A receptor activity by increasing frequency of chloride channel op. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Diazepam
  • Manufacturer: Arrow Pharma
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

๐Ÿ’Š dpm injection Uses & Benefits

Anxiety disorders, alcohol withdrawal, muscle spasms, seizure disorders, preoperative sedation.

Off-label uses: Panic disorder, insomnia, restless legs syndrome, spasticity in multiple sclerosis.

๐Ÿ“‹ Drug Information

Generic Name(s)Diazepam
Brand NameAlzepam
ManufacturerArrow Pharma
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassBenzodiazepines
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF) in a dry place, protect from light.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionWell absorbed orally with peak plasma concentrations within 1-2 hours.
DistributionHighly lipophilic, crosses blood-brain barrier and placenta; distributed into breast milk.
Protein Binding98% bound to plasma proteins.
MetabolismHepatic via CYP2C19 and CYP3A4 to active metabolites (nordiazepam, temazepam, oxazepam).
Half-Life20-50 hours (parent); active metabolites have longer half-lives.
ExcretionPrimarily renal as metabolites; less than 10% unchanged.
Bioavailability90-100% (oral).
Onset of Action30-60 minutes (oral).
Peak Plasma Time1-2 hours.
Duration of Action12-24 hours (depending on dose and tolerance).

How It Works

Enhances GABA-A receptor activity by increasing frequency of chloride channel opening.

Mechanism Steps

1Binds to benzodiazepine site on GABA-A receptor
2Increases affinity of GABA for receptor
3Enhances chloride ion influx

๐Ÿ’ก How to Take dpm injection

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of dpm injection

โœ… Common Side Effects

  • Drowsiness
  • Dizziness
  • Fatigue
  • Ataxia
  • Slurred speech

๐Ÿšจ Serious Side Effects

  • Respiratory depression
  • Paradoxical reactions (agitation, aggression)
  • Dependence
  • Withdrawal seizures

โš ๏ธ Rare Side Effects

  • Jaundice
  • Blood dyscrasias
  • Anaphylaxis
  • Hypotension

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Alcohol Major Increased sedation and respiratory depression
Opioids Major Additive CNS depression, risk of respiratory depression
Ketoconazole Major Increased diazepam levels due to CYP3A4 inhibition
Omeprazole Major Increased diazepam levels due to CYP2C19 inhibition
Rifampin Moderate Decreased diazepam levels due to enzyme induction
Oral contraceptives Moderate May prolong half-life of diazepam
Antacids Minor May delay absorption
Cimetidine Minor May increase diazepam levels

๐Ÿšจ Major Interactions

  • CNS depressants (alcohol, opioids, barbiturates)
  • CYP3A4 inhibitors (ketoconazole, ritonavir)
  • CYP2C19 inhibitors (omeprazole, fluvoxamine)

โšก Moderate Interactions

  • CYP3A4 inducers (rifampin, carbamazepine)
  • CYP2C19 inducers (rifampin)
  • Oral contraceptives

โ„น๏ธ Minor Interactions

  • Antacids
  • Cimetidine
  • Disulfiram

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase absorption; food delays absorption.

๐Ÿท Alcohol Interaction

Additive CNS depression; avoid concurrent use.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity, severe respiratory insufficiency, sleep apnea, myasthenia gravis, narrow-angle glaucoma.

๐Ÿ“Š Monitoring Parameters

CNS depression, respiratory rate, blood pressure, liver function tests, signs of dependence.

๐Ÿคฑ Lactation Safety

Excreted in breast milk; avoid or monitor infant for sedation.

๐Ÿ’Š Overdose Management

Supportive care; flumazenil as antidote (use with caution in benzodiazepine-dependent patients).

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose; do not double.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 28, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for dpm injection

View All

Alternative brands with exact same active ingredient (Diazepam (NA)):

Medical Note: Always consult your doctor before switching medications.

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