divi a 500mg injection - Metamizole (500mg) medicine

Divi A 500mg Injection (Metamizole): Comprehensive Medicine Guide

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🏭 Flagship Biotech International 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 25, 2026
⚠️ Nephrotoxicity Risk 🤰 Pregnancy Category Not recommended during pregnancy, especially in the first and third trimesters. Metamizole crosses the placenta and may cause fetal harm. Use only if clearly needed and under medical supervision. 📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Evidence: Well-established for acute severe pain and fever in countries where it is approved.
Reviewed by
SaathiMed Expert Panel | Sep 25, 2026

When to Call Your Doctor IMMEDIATELY

  • Fever, sore throat, or mouth ulcers (may indicate agranulocytosis).
  • Difficulty breathing, swelling of face or throat (anaphylaxis).
  • Severe skin rash with blisters or peeling (Stevens-Johnson syndrome).
  • Decreased urine output or swelling in legs (kidney injury).
  • Yellowing of eyes or skin (liver toxicity).
  • Unusual bleeding or bruising (blood disorder).
  • Severe abdominal pain or blood in vomit/stool (GI bleeding).

If experiencing severe symptoms, call emergency services immediately.

What is divi a 500mg injection used for?

This medicine is a 500mg injection of Metamizole, a strong pain reliever and fever reducer. It is given by a healthcare professional for moderate to severe pain or high fever when oral medicines are not suitable. It works by blocking pain and fever signals in the body. It is not recommended for routine use due to rare but serious blood-related side effects.

  • Generic Name: Metamizole (500mg)
  • Manufacturer: Flagship Biotech International
  • Form: Allopathy
  • Pregnancy Category: Consult doctor
  • Prescription Required: Yes

🇮🇳 divi a 500mg injection के बारे में (Hindi Summary)

उपयोग: यह दवा मेटामिज़ोल का 500 मिलीग्राम इंजेक्शन है, जिसका उपयोग तेज दर्द और तेज बुखार के इलाज के लिए किया जाता है। यह आमतौर पर तब दी जाती है जब मरीज मुंह से दवा नहीं ले सकता या अन्य दर्द निवारक दवाएं काम नहीं कर रही हों। यह दवा डॉक्टर या नर्स द्वारा इंजेक्शन के रूप में दी जाती है। यह दर्द और बुखार को कम करने में मदद करती है।

साइड इफेक्ट्स: आम दुष्प्रभावों में इंजेक्शन वाली जगह पर दर्द, लालिमा, मतली, चक्कर आना और सिरदर्द शामिल हैं। गंभीर दुष्प्रभावों में एग्रानुलोसाइटोसिस (खून की गंभीर बीमारी), एलर्जी, और किडनी की समस्या हो सकती है। अगर आपको बुखार, गले में खराश, या मुंह में छाले हों तो तुरंत डॉक्टर को बताएं।

सुरक्षा सलाह: यह दवा केवल डॉक्टर की देखरेख में ही दी जानी चाहिए। खुद से इंजेक्शन न लगवाएं। अगर आपको खून की बीमारी, किडनी या लिवर की समस्या है, या दर्द निवारक दवाओं से एलर्जी है, तो डॉक्टर को बताएं। इलाज के दौरान शराब न पिएं। बिना डॉक्टर की सलाह के लंबे समय तक इसका इस्तेमाल न करें।

💡 Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

💊 divi a 500mg injection Uses & Benefits

[{"condition":"Acute severe pain","description":"Used for rapid relief of moderate to severe pain when oral administration is not possible, such as in postoperative pain or trauma.","evidence":"Well-established"},{"condition":"High fever","description":"Effective in reducing high fever that does not respond to other antipyretics, especially in emergency settings.","evidence":"Well-established"},{"condition":"Colicky pain","description":"Due to its antispasmodic properties, it is used for renal or biliary colic.","evidence":"Moderate"},{"condition":"Cancer pain","description":"May be used as an adjunct for cancer-related pain when other analgesics are inadequate.","evidence":"Limited"}]

Off-label uses: [{"condition":"Migraine","description":"Sometimes used off-label for acute migraine attacks, but not first-line.","evidence":"Limited"}]

Primary treatment for: Acute severe pain

Also treats: High fever, Colicky pain, Postoperative pain, Cancer pain

📋 Drug Information

Generic Name(s)Metamizole (500mg)
Brand Namedivi a 500mg injection
ManufacturerFlagship Biotech International
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassPAIN ANALGESICS
Action ClassNSAID's-Non-Selective COX 1&2 Inhibitors (Others)
Route of AdministrationParenteral (intramuscular or intravenous)
StorageStore below 25°C, protected from light. Do not freeze. Keep out of reach of children.
Shelf Life24 months from the date of manufacture.
WHO GuidelineNot established from the available information.
ICMR GuidelineNot established from the available information.

👨‍⚕️ Doctor's Practical Tips

Evidence-based practical advice from experienced clinicians

1
Always administer this medicine slowly intravenously to avoid sudden drop in blood pressure.
2
Monitor patients for at least 30 minutes after injection for any signs of allergic reaction.
3
Avoid using this medicine for more than 3-5 days without reassessing the patient.
4
Check complete blood counts if the patient develops any signs of infection during treatment.
5
Use with caution in elderly patients and those with kidney or liver problems.
6
Do not mix this medicine with other drugs in the same syringe.

🔍 Is This Medicine Right for Your Symptom?

Educational reference. Always consult a doctor for diagnosis.

✅
Severe pain
This medicine is commonly prescribed for moderate to severe pain.
Likely Use
✅
High fever
This medicine is effective for reducing high fever.
Likely Use
❌
Mild headache
This medicine is not typically used for mild pain.
Not Primary
❌
Common cold
This medicine is not a treatment for cold symptoms.
Not Primary

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionFollowing intramuscular administration, metamizole is rapidly absorbed, with peak plasma concentrations reached within 30-60 minutes. Intravenous administration provides immediate plasma levels.
DistributionMetamizole and its metabolites are distributed widely in the body. The active metabolite MAA has a volume of distribution of approximately 0.7 L/kg. It crosses the placenta and is excreted in breast milk.
Protein BindingThe active metabolite MAA is approximately 58% bound to plasma proteins.
MetabolismMetamizole is extensively metabolized in the liver via hydrolysis to MAA, which is further metabolized to 4-formylaminoantipyrine (FAA) and 4-acetylaminoantipyrine (AAA). These metabolites are then excreted.
Half-LifeThe elimination half-life of the active metabolite MAA is approximately 2.7 to 3.5 hours. In elderly patients or those with hepatic impairment, the half-life may be prolonged.
ExcretionMetabolites are primarily excreted in the urine (approximately 90%) and to a lesser extent in feces.
BioavailabilityIntramuscular bioavailability is high, approximately 85-90%. Intravenous administration provides 100% bioavailability.
Onset of ActionPain relief begins within 20-30 minutes after intramuscular injection and within 5-10 minutes after intravenous administration.
Peak Plasma TimePeak plasma concentration of the active metabolite MAA occurs approximately 30-60 minutes after intramuscular injection and immediately after intravenous injection.
Duration of ActionThe analgesic effect lasts approximately 4-6 hours after a single dose.

How It Works

Metamizole is a prodrug that is hydrolyzed to 4-methylaminoantipyrine (MAA), which inhibits cyclooxygenase (COX) enzymes, particularly COX-2, leading to decreased synthesis of prostaglandins. It also activates the endogenous opioid system and inhibits prostaglandin synthesis in the central nervous system, contributing to analgesia and antipyresis. Additionally, it has antispasmodic effects on smooth muscle.

Mechanism Steps

1
Prodrug conversion: Metamizole is rapidly hydrolyzed in the body to its active metabolite, 4-methylaminoantipyrine (MAA).
2
COX inhibition: MAA inhibits cyclooxygenase enzymes, reducing the production of prostaglandins, which are mediators of pain and fever.
3
Central analgesia: It also acts on the central nervous system to modulate pain perception, possibly involving opioid receptors.
4
Antispasmodic effect: It relaxes smooth muscle, which is beneficial in treating colicky pain.

💡 How to Take divi a 500mg injection

Strength: 500 mg injection (2 mL ampoule).

1This medicine is given by a healthcare professional.
2For intramuscular injection, the usual site is the upper outer quadrant of the buttock.
3For intravenous injection, it should be given slowly over 5-10 minutes to avoid hypotension.
4Do not mix with other drugs in the same syringe.
5After injection, remain under observation for at least 30 minutes to monitor for allergic reactions.

Dosage Information

Adult DosageThe usual adult dose is 500 mg to 1000 mg (1-2 ampoules) given intramuscularly or intravenously every 6-8 hours as needed, not exceeding 4000 mg per day. For intravenous use, inject slowly over 5-10 minutes. Dose must be individualized by a qualified clinician based on indication, age, weight, renal and hepatic function.
Pediatric DosagePediatric dosing is not established from available information. Consult a pediatrician. In some countries, metamizole is used in children over 3 months at a dose of 10-20 mg/kg per dose, but this must be determined by a pediatrician.
Elderly DosageElderly patients may require lower doses due to reduced renal and hepatic function. Start with the lowest effective dose and monitor closely.
Renal ImpairmentUse with caution in patients with renal impairment. Dose reduction may be necessary. Avoid in severe renal impairment (eGFR <30 mL/min).
Hepatic ImpairmentUse with caution in patients with hepatic impairment. Dose reduction may be necessary. Avoid in severe hepatic impairment.
Maximum Daily Dose4000 mg per day (8 ampoules of 500 mg).

Dosage Timeline

🌅 Morning ❌ ☀️ Afternoon ❌ 🌆 Evening ❌ 🌙 Night ❌

🍽️ Food Timing Guide

With food
No specific food restrictions for injection.
This medicine is given parenterally, so food does not affect its absorption.
Alcohol
Avoid
Increases risk of liver toxicity and gastrointestinal bleeding.

⏰ What to Do If You Miss a Dose

📌 Less than half the dosing interval has passed
→ Take the missed dose as soon as you remember.
💡 Continue with the regular schedule.
📌 More than half the dosing interval has passed
→ Skip the missed dose.
💡 Do not double dose to catch up.

⚠️ Side Effects of divi a 500mg injection

✅ Common Side Effects

Injection site pain (Common (5-10%))
Apply a cold compress to the site. It usually resolves within a few hours.
Nausea (Common (5-10%))
Take small sips of water. If persistent, consult your doctor.
Dizziness (Common (5-10%))
Lie down until it passes. Avoid driving or operating machinery.
Headache (Common (5-10%))
Rest in a quiet, dark room. Consult doctor if severe.

🚨 Serious Side Effects

Agranulocytosis (Rare (<0.1%))
Seek immediate medical attention if you develop fever, sore throat, or mouth ulcers.
Anaphylaxis (Rare (<0.1%))
Call emergency services if you experience difficulty breathing, swelling of face or throat, or a severe rash.
Stevens-Johnson syndrome (Very rare (<0.01%))
Seek immediate medical attention if you develop a painful rash with blisters or peeling skin.
Acute kidney injury (Rare (<0.1%))
Report decreased urine output or swelling to your doctor immediately.

⚠️ Rare Side Effects

Thrombocytopenia
Report unusual bruising or bleeding to your doctor.
Leukopenia
Regular blood tests may be needed. Report any signs of infection.
Hepatotoxicity
Report yellowing of skin or eyes, dark urine, or abdominal pain.

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Warfarin Major
Methotrexate Major
Cyclosporine Major
Aspirin Moderate
ACE inhibitors Moderate
Diuretics Moderate
Lithium Moderate
SSRIs Moderate
Corticosteroids Moderate
Phenytoin Minor

🚨 Major Interactions

  • Warfarin
  • Methotrexate
  • Cyclosporine

⚡ Moderate Interactions

  • Aspirin
  • ACE inhibitors
  • Diuretics

🍷 Alcohol Interaction

Avoid alcohol consumption while receiving this medicine. Alcohol can increase the risk of stomach bleeding, liver damage, and may worsen side effects such as dizziness and drowsiness.

🔎 Check Your Other Medicines

Educational tool. Always confirm with your doctor or pharmacist.

🛡️ Safety & Warnings

🚫 Contraindications

["Hypersensitivity to metamizole or other pyrazolones.","History of agranulocytosis or bone marrow suppression.","Genetic deficiency of glucose-6-phosphate dehydrogenase (G6PD).","Acute hepatic porphyria.","Third trimester of pregnancy and lactation.","Severe renal or hepatic impairment.","Children under 3 months or under 5 kg body weight."]

⚠️ Warnings & Precautions

["Risk of agranulocytosis: Inform patients to report early signs of infection.","Anaphylactic reactions: Have emergency equipment ready.","Hypotension: Can occur with rapid intravenous injection. Inject slowly.","Renal impairment: Use with caution and monitor.","Hepatic impairment: Use with caution and monitor.","Elderly: Increased risk of side effects. Use lower doses.","Avoid in patients with active peptic ulcer or bleeding disorders."]

🤱 Lactation Safety

Metamizole and its metabolites are excreted in breast milk. Breastfeeding is not recommended during treatment. If treatment is essential, consider pumping and discarding milk during therapy and for 48 hours after the last dose.

💊 Overdose Management

Overdose may cause nausea, vomiting, abdominal pain, dizziness, drowsiness, and in severe cases, seizures, coma, and acute renal failure. There is no specific antidote. Treatment is supportive and symptomatic. Gastric lavage may be considered if oral ingestion is recent. Monitor vital signs, renal and hepatic function. Hemodialysis may be effective in removing metabolites.

⏰ Missed Dose

This medicine is usually given as a single dose or as needed under medical supervision. If you miss a scheduled dose, contact your healthcare provider for instructions. Do not self-administer an extra dose.

Additional Safety Advice

General Safety

This medicine must only be administered by a healthcare professional. Do not self-administer. Inform your doctor if you have a history of blood disorders, kidney or liver disease, or allergies to pain relievers. Avoid alcohol during treatment as it may increase the risk of stomach bleeding and liver toxicity. Do not use for prolonged periods without medical supervision. If you experience fever, sore throat, or mouth sores, seek immediate medical attention as these may be signs of a serious blood disorder. Keep all follow-up appointments for blood tests if advised.

👴 Special Considerations for Elderly

💡 For Patients Above 65

Elderly patients are at higher risk of side effects, especially agranulocytosis, kidney injury, and gastrointestinal bleeding. Lower doses may be needed. Monitor renal and hepatic function closely.

🤰 Pregnancy Planning (TTC)

This medicine is not recommended during pregnancy, especially in the first and third trimesters. If you are planning pregnancy, discuss alternative pain management options with your doctor. Use effective contraception while on this medicine.

🏥 Post-Surgery Considerations

This medicine may be used for postoperative pain. It should be administered under medical supervision. Monitor for signs of infection, bleeding, and allergic reactions. Ensure adequate hydration.

🦷 Dental Procedures

Inform your dentist if you are receiving this medicine, as it may increase bleeding risk during dental procedures. Your dentist may recommend postponing elective procedures until you have completed treatment.

💚 Lifestyle Tips for Better Results

🏃
Stay well hydrated to help your kidneys flush out the medicine.
🥗
Avoid alcohol to reduce the risk of liver and stomach problems.
😴
Eat a balanced diet to support your immune system.
💧
Get plenty of rest to help your body recover.
🧘
Report any unusual symptoms to your doctor promptly.
🌞
Do not share this medicine with others.

🏋️ Exercise Considerations

Avoid strenuous exercise or activities that could cause injury while you are experiencing pain. If you feel dizzy or drowsy after the injection, do not drive or operate heavy machinery. Gentle movement may be beneficial once acute pain subsides, but consult your doctor before resuming exercise.

🥗 Diet Recommendations

Drink plenty of water to stay hydrated.
Avoid alcohol completely during treatment.
Eat light, easily digestible meals if you have nausea.
Include fruits and vegetables rich in antioxidants to support recovery.

💼 Impact on Daily Work & Life

This medicine may cause dizziness or drowsiness, so avoid driving or operating machinery until you know how it affects you. You may need to take rest after the injection. It is usually given in a hospital or clinic setting, so you may need to arrange for transportation home.

🛑 When to Stop This Medicine

This medicine is usually given for a short duration. Stop using it and consult your doctor immediately if you experience any signs of allergic reaction, infection, or unusual bleeding. Do not stop prescribed treatment without consulting your doctor.

📅 Long-Term Use Effects

Long-term use of this medicine is not recommended due to the risk of agranulocytosis, which can occur at any time. Prolonged use may also lead to kidney or liver damage. Regular monitoring of blood counts, liver, and kidney function is advised if long-term therapy is necessary. The risk of agranulocytosis may increase with duration of use, so the lowest effective dose for the shortest duration should be used.

🌿 Non-Medicine Approaches

These can complement medicine but do not replace prescribed treatment.

Paracetamol

Safer alternative for mild to moderate pain and fever.

Evidence: Well-established
NSAIDs (e.g., ibuprofen, diclofenac)

Effective for pain and inflammation but carry GI and renal risks.

Evidence: Well-established
Opioids (e.g., tramadol, morphine)

For severe pain, but have risk of dependence.

Evidence: Well-established
Physical therapy

Can complement medicine for chronic pain.

Evidence: Well-established

💉 Vaccination Considerations

💉 If You're Getting Vaccinated

No specific interactions with vaccines are known. However, if you have a fever, vaccination may be postponed until you recover. Consult your doctor.

📦 Storage Guide

✅ DO

Store at room temperature (15-30°C)

❌ DON'T

Do not refrigerate or freeze

✅ DO

Keep in original container

❌ DON'T

Do not transfer to unmarked containers

✅ DO

Keep away from direct sunlight

❌ DON'T

Do not store in bathroom cabinet

✅ DO

Check expiry date before use

❌ DON'T

Do not use if solution is discolored or contains particles

✈️ Traveling with This Medicine

When traveling with this medicine, carry it in its original packaging with the prescription label intact. Keep a copy of your prescription and a letter from your doctor explaining the medical need. Store it in a cool, dry place away from direct sunlight. If traveling by air, keep it in your carry-on luggage. Check the customs regulations of your destination country regarding injectable medicines. For time zone changes, consult your doctor for dose adjustment if you are on a scheduled regimen.

💰 Cost Analysis & Savings

👥 Real Patient Stories

Educational, anonymized scenarios. Individual results may vary.

👤 A 60-year-old man with severe postoperative pain after knee surgery.
He was given this medicine intramuscularly every 8 hours. His pain significantly reduced within 30 minutes of injection. He experienced mild nausea but it subsided. He was monitored for blood counts and kidney function, which remained normal.
💡 Lesson: This medicine provides rapid pain relief but requires monitoring for side effects, especially in elderly patients.
👤 A 35-year-old woman with high fever unresponsive to oral paracetamol.
She received an intravenous dose of this medicine. Her fever dropped within 20 minutes. She developed a mild rash which was managed with antihistamines. She was advised not to use this medicine again due to allergic reaction.
💡 Lesson: Allergic reactions can occur even with first use. Immediate medical attention is necessary if any rash or swelling appears.

💬 Questions Patients Often Ask

Q: How long does it take to work?

A: This medicine starts working within 20-30 minutes after intramuscular injection and within 5-10 minutes after intravenous injection.

Q: How long does the effect last?

A: The pain-relieving effect lasts approximately 4-6 hours.

Q: Can I take this medicine at home?

A: No, this medicine must be administered by a healthcare professional in a clinical setting.

Q: What should I do if I experience side effects?

A: Report any side effects to your doctor immediately. Seek emergency care if you have difficulty breathing, swelling, or severe rash.

🤔 Common Patient Concerns

💭 These are the concerns patients most commonly raise

  • Can I take this medicine long-term?
  • Will it affect my kidney function?
  • Can I drive after taking this medicine?
  • Does it interact with my blood pressure medicine?
  • What if I miss a dose?
  • Can I drink alcohol while taking this?
  • Is it safe during pregnancy?
  • Can it cause blood cancer?

🔄 Substitutes for divi a 500mg injection

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

🛑 Myths vs. Facts

  • Myth: Metamizole is a safe alternative to morphine.
    Fact: Metamizole is effective for pain but carries a rare risk of agranulocytosis, so it is not entirely safe and is not a direct substitute for morphine.
  • Myth: Metamizole can be used for any type of pain.
    Fact: It is indicated for moderate to severe pain and fever, but not for mild pain or routine use.
  • Myth: Metamizole is banned worldwide.
    Fact: It is banned in some countries like the USA, but available in many others including India, Mexico, and parts of Europe.

🔄 Alternative Options

Generic Alternatives

  • Metamizole 500mg injection

Brand Alternatives

  • Divi A 500mg injection

📊 Comparison with Similar Medicines

[{"medicine":"Metamizole","class":"Pyrazolone","uses":"Severe pain, fever","route":"Parenteral","key_side_effects":"Agranulocytosis, allergic reactions"},{"medicine":"Paracetamol","class":"Analgesic/antipyretic","uses":"Mild to moderate pain, fever","route":"Oral, rectal, IV","key_side_effects":"Hepatotoxicity in overdose"},{"medicine":"Diclofenac","class":"NSAID","uses":"Moderate to severe pain, inflammation","route":"Oral, IM, IV","key_side_effects":"GI bleeding, renal impairment"}]

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