dermosav plus cream - Ciprofloxacin (1% w/w) + Metronidazole (1% w/w) medicine

dermosav plus cream - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Bennet Mypher Pharmaceuticals LLP ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 29, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 29, 2026

What is dermosav plus cream used for?

Clobest-CM Cream (Ciprofloxacin + Metronidazole) is used to treat DERMA. It contains Ciprofloxacin (1% w/w) + Metronidazole (1% w/w), which Ciprofloxacin inhibits bacterial DNA gyrase and topoisomerase IV; Metronidazole . Always consult your doctor before use. Take as prescribed.

  • Generic Name: Ciprofloxacin + Metronidazole
  • Manufacturer: Bennet Mypher Pharmaceuticals LLP
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š dermosav plus cream Uses & Benefits

Topical treatment of infected wounds, ulcers, and skin infections with mixed aerobic/anaerobic flora

Off-label uses: Pressure ulcers, Diabetic foot ulcers

๐Ÿ“‹ Drug Information

Generic Name(s)Ciprofloxacin + Metronidazole
Brand NameClobest-CM Cream
ManufacturerBennet Mypher Pharmaceuticals LLP
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassDERMA
Action ClassAntibiotic + Antiprotozoal
Route of AdministrationTopical
StorageStore at 20-25ยฐC; protect from light
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionMinimal systemic absorption following topical application
DistributionLimited to local tissues; negligible systemic distribution
Protein BindingCiprofloxacin: 20-40%; Metronidazole: <20%
MetabolismCiprofloxacin: Hepatic (partial); Metronidazole: Hepatic (oxidation and glucuronidation)
Half-LifeCiprofloxacin: 4 hours; Metronidazole: 8 hours (systemic, but topical absorption minimal)
ExcretionCiprofloxacin: Renal (fecal); Metronidazole: Renal (60-80%)
BioavailabilityNegligible via topical route
Onset of ActionWithin 24-48 hours
Peak Plasma TimeNot applicable (topical)
Duration of Action12-24 hours

How It Works

Ciprofloxacin inhibits bacterial DNA gyrase and topoisomerase IV; Metronidazole disrupts DNA synthesis in anaerobic bacteria and protozoa

Mechanism Steps

1Ciprofloxacin enters bacterial cells and binds to DNA gyrase and topoisomerase IV
2Inhibition of DNA replication and transcription leads to bacterial cell death
3Metronidazole enters anaerobic cells and is reduced to active metabolites

๐Ÿ’ก How to Take dermosav plus cream

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of dermosav plus cream

โœ… Common Side Effects

  • Application site irritation
  • Itching
  • Redness

๐Ÿšจ Serious Side Effects

  • Severe allergic reaction
  • Tendon rupture (rare with topical)

โš ๏ธ Rare Side Effects

  • Peripheral neuropathy
  • Disulfiram-like reaction with alcohol

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Major Increased INR and bleeding risk
Tizanidine Major Hypotension, sedation
Theophylline Major Increased theophylline levels, toxicity
NSAIDs Moderate Increased CNS stimulation risk
Oral hypoglycemics Moderate Hypoglycemia risk
Corticosteroids Moderate Increased tendon rupture risk
Caffeine Minor Reduced caffeine clearance
Antacids (systemic) Minor Reduced ciprofloxacin absorption (if oral)

๐Ÿšจ Major Interactions

  • Warfarin
  • Tizanidine
  • Theophylline

โšก Moderate Interactions

  • NSAIDs
  • Oral hypoglycemics
  • Corticosteroids

โ„น๏ธ Minor Interactions

  • Caffeine
  • Antacids (systemic)

๐Ÿฝ๏ธ Food Interactions

No significant food interactions for topical use

๐Ÿท Alcohol Interaction

Avoid alcohol during metronidazole therapy (disulfiram-like reaction)

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to quinolones or metronidazole; application to open wounds or mucous membranes

๐Ÿ“Š Monitoring Parameters

Local skin reactions, signs of superinfection

๐Ÿคฑ Lactation Safety

Caution; avoid application to breast area

๐Ÿ’Š Overdose Management

Unlikely with topical use; if ingested, symptomatic treatment

โฐ Missed Dose

Apply as soon as remembered; skip if almost time for next dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 29, 2026

๐Ÿ”— View Profile

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