creslip 40mg/10mg tablet - Telmisartan (40mg) + Atorvastatin (10mg) medicine

creslip 40mg/10mg tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Cipla Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jul 3, 2026
โš ๏ธ Hepatotoxicity Risk ๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jul 03, 2026

What is creslip 40mg/10mg tablet used for?

Arbitel-AV Tablet (Telmisartan + Atorvastatin) is used to treat CARDIAC. It contains Telmisartan (40mg) + Atorvastatin (10mg), which Telmisartan blocks angiotensin II AT1 receptors, causing vasodilation and reduce. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Telmisartan + Atorvastatin
  • Manufacturer: Cipla Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š creslip 40mg/10mg tablet Uses & Benefits

Hypertension with dyslipidemia, cardiovascular risk reduction.

Off-label uses: Diabetic nephropathy, migraine prophylaxis (telmisartan), familial hypercholesterolemia (atorvastatin).

๐Ÿ“‹ Drug Information

Generic Name(s)Telmisartan + Atorvastatin
Brand NameArbitel-AV Tablet
ManufacturerCipla Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassAngiotensin II Receptor Blocker + HMG-CoA Reductase Inhibitor
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionTelmisartan: Rapidly absorbed; Atorvastatin: Rapidly absorbed after oral administration.
DistributionTelmisartan: High volume of distribution; Atorvastatin: Extensive distribution into tissues.
Protein BindingTelmisartan: >99.5%; Atorvastatin: 98-99%
MetabolismTelmisartan: Glucuronidation; Atorvastatin: CYP3A4 to active metabolites.
Half-LifeTelmisartan: ~24 hours; Atorvastatin: ~14 hours (parent drug), active metabolites: 20-30 hours.
ExcretionTelmisartan: Mainly feces (97%); Atorvastatin: Biliary (70% as metabolites) and renal (2%).
BioavailabilityTelmisartan: 42-58%; Atorvastatin: 14% (oral), increased with food.
Onset of ActionTelmisartan: 2-4 hours; Atorvastatin: 1-2 weeks for lipid effects.
Peak Plasma TimeTelmisartan: 0.5-1 hour; Atorvastatin: 1-2 hours.
Duration of ActionTelmisartan: 24 hours; Atorvastatin: 24 hours (lipid lowering).

How It Works

Telmisartan blocks angiotensin II AT1 receptors, causing vasodilation and reduced aldosterone secretion. Atorvastatin inhibits HMG-CoA reductase, reducing cholesterol synthesis.

Mechanism Steps

1Telmisartan binds to AT1 receptor, blocking angiotensin II.
2Vasodilation occurs, reducing peripheral resistance.
3Aldosterone secretion decreases, reducing sodium and water retention.

๐Ÿ’ก How to Take creslip 40mg/10mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of creslip 40mg/10mg tablet

โœ… Common Side Effects

  • Headache
  • Dizziness
  • Diarrhea
  • Muscle pain
  • Upper respiratory infection

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Rhabdomyolysis
  • Hepatotoxicity
  • Renal impairment
  • Hypotension

โš ๏ธ Rare Side Effects

  • Pancreatitis
  • Interstitial lung disease
  • Stevens-Johnson syndrome
  • Myasthenia gravis exacerbation

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Moderate Increased INR and bleeding risk
Ketoconazole Major Increased atorvastatin levels and myopathy risk
Cyclosporine Major Increased atorvastatin levels and myopathy risk
Gemfibrozil Major Increased risk of myopathy/rhabdomyolysis
Rifampin Major Decreased atorvastatin efficacy
Digoxin Major Increased digoxin levels
Antacids Moderate Reduced telmisartan absorption
Colchicine Moderate Increased risk of myopathy
Fibrates Moderate Increased risk of myopathy
Niacin Moderate Increased risk of myopathy
Grapefruit juice Minor Increased atorvastatin levels
Oral contraceptives Minor Increased contraceptive levels

๐Ÿšจ Major Interactions

  • CYP3A4 inhibitors (e.g., ketoconazole, itraconazole)
  • Cyclosporine
  • Gemfibrozil
  • Rifampin
  • Digoxin

โšก Moderate Interactions

  • Warfarin
  • Antacids
  • Colchicine
  • Fibrates
  • Niacin

โ„น๏ธ Minor Interactions

  • Grapefruit juice
  • Oral contraceptives
  • Digoxin

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase atorvastatin levels; avoid high-fat meals with telmisartan.

๐Ÿท Alcohol Interaction

May increase risk of liver damage and hypotension.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Pregnancy, lactation, hypersensitivity, active liver disease, severe renal impairment, concomitant use with strong CYP3A4 inhibitors.

๐Ÿ“Š Monitoring Parameters

Blood pressure, lipid profile, liver enzymes, renal function, muscle symptoms.

๐Ÿคฑ Lactation Safety

Contraindicated; avoid breastfeeding.

๐Ÿ’Š Overdose Management

Symptomatic and supportive; monitor BP, ECG, liver function; consider gastric lavage.

โฐ Missed Dose

Take as soon as remembered; skip if near next dose; do not double.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jul 03, 2026

๐Ÿ”— View Profile

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