cilnicue-t tablet - Cilnidipine (10mg) + Telmisartan (40mg) medicine

cilnicue-t tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Cue Labs ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 30, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 30, 2026

What is cilnicue-t tablet used for?

Acmetel-LN Tablet (Cilnidipine + Telmisartan) is used to treat CARDIAC. It contains Cilnidipine (10mg) + Telmisartan (40mg), which Cilnidipine: Inhibits calcium influx through L-type and N-type calcium channels,. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Cilnidipine + Telmisartan
  • Manufacturer: Cue Labs
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

๐Ÿ’Š cilnicue-t tablet Uses & Benefits

Hypertension (essential hypertension).

Off-label uses: Chronic kidney disease (with proteinuria), heart failure (limited data).

๐Ÿ“‹ Drug Information

Generic Name(s)Cilnidipine + Telmisartan
Brand NameAcmetel-LN Tablet
ManufacturerCue Labs
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassCalcium channel blocker + Angiotensin II receptor blocker
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionCilnidipine: Well absorbed after oral administration; Telmisartan: Rapidly absorbed, absolute bioavailability is dose-dependent (42% for 40 mg, 58% for 160 mg).
DistributionCilnidipine: Highly protein bound (>99%); Telmisartan: Extensively distributed, Vd ~500 L.
Protein BindingCilnidipine: >99%; Telmisartan: >99.5% (mainly albumin and alpha-1-acid glycoprotein).
MetabolismCilnidipine: Metabolized by CYP3A4; Telmisartan: Metabolized by glucuronidation (no CYP involvement).
Half-LifeCilnidipine: ~5-6 hours; Telmisartan: ~24 hours.
ExcretionCilnidipine: 80% feces, 20% urine; Telmisartan: >97% feces (unchanged).
BioavailabilityCilnidipine: ~13%; Telmisartan: 42-58%.
Onset of ActionCilnidipine: 1-2 hours; Telmisartan: 1-2 hours.
Peak Plasma TimeCilnidipine: 2-3 hours; Telmisartan: 0.5-1 hour.
Duration of ActionCilnidipine: ~24 hours; Telmisartan: >24 hours.

How It Works

Cilnidipine: Inhibits calcium influx through L-type and N-type calcium channels, causing vasodilation and reduced blood pressure; Telmisartan: Blocks angiotensin II type 1 (AT1) receptors, leading to vasodilation and reduced aldosterone secretion.

Mechanism Steps

1Cilnidipine binds to L-type and N-type calcium channels in vascular smooth muscle and sympathetic nerve terminals.
2Inhibition of calcium influx causes vasodilation and reduced peripheral resistance.
3Telmisartan selectively blocks AT1 receptors, preventing angiotensin II-mediated vasoconstriction and aldosterone release.

๐Ÿ’ก How to Take cilnicue-t tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of cilnicue-t tablet

โœ… Common Side Effects

  • Dizziness
  • Headache
  • Peripheral edema
  • Fatigue
  • Diarrhea

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Syncope
  • Acute renal failure
  • Hyperkalemia
  • Hepatotoxicity

โš ๏ธ Rare Side Effects

  • Thrombocytopenia
  • Interstitial pneumonitis
  • Anaphylaxis

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Lithium Major Increased lithium levels and toxicity
Potassium-sparing diuretics Major Increased risk of hyperkalemia
NSAIDs Moderate Reduced antihypertensive effect and increased renal risk
CYP3A4 inhibitors Moderate Increased cilnidipine levels
Digoxin Moderate Increased digoxin levels
Warfarin Minor Minimal effect on INR

๐Ÿšจ Major Interactions

  • Lithium
  • Potassium-sparing diuretics
  • ACE inhibitors
  • Aliskiren

โšก Moderate Interactions

  • NSAIDs
  • CYP3A4 inhibitors (e.g., ketoconazole)
  • CYP3A4 inducers (e.g., rifampin)
  • Digoxin

โ„น๏ธ Minor Interactions

  • Antacids
  • Warfarin

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase cilnidipine levels; high-fat meals may reduce telmisartan absorption.

๐Ÿท Alcohol Interaction

May potentiate hypotensive effects; avoid excessive alcohol.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity; pregnancy; bilateral renal artery stenosis; severe hepatic impairment; concomitant use with aliskiren in diabetes.

๐Ÿ“Š Monitoring Parameters

Blood pressure, heart rate, serum potassium, renal function, liver function.

๐Ÿคฑ Lactation Safety

Not recommended; avoid breastfeeding.

๐Ÿ’Š Overdose Management

Symptomatic and supportive treatment; monitor blood pressure and heart rate; consider gastric lavage if recent ingestion.

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 30, 2026

๐Ÿ”— View Profile

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