caregalin-m tablet - Alpha Lipoic Acid (300mg) + Pregabalin (75mg) medicine

caregalin-m tablet

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🏭 Humane Care Pharmaceuticals Pvt. Ltd. 📦 Varies by brand 💊 Allopathy 📅 Updated: Oct 23, 2026
📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Reviewed by
SaathiMed Expert Panel | Oct 23, 2026
🩺
Medically Fact-Checked & Clinically Verified by SaathiMed Clinical Review Board
Clinical Reference Standards: CDSCO (Central Drugs Standard Control Organisation), Indian Pharmacopoeia (IP) & WHO | Last Updated: September 2026

What is caregalin-m tablet used for?

This medicine contains Alpha Lipoic Acid (300mg) + Pregabalin (75mg) and is used to treat NEURO CNS. Pregabalin binds to alpha2-delta subunit of voltage-gated calcium channels, reducing calcium influx . Always consult your doctor before use.

  • Generic Name: Alpha Lipoic Acid + Pregabalin
  • Manufacturer: Humane Care Pharmaceuticals Pvt. Ltd.
  • Form: Allopathy
  • Pregnancy Category: Category A
  • Prescription Required: Yes
💡 Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

💊 caregalin-m tablet Uses & Benefits

Neuropathic pain associated with diabetic neuropathy, postherpetic neuralgia, fibromyalgia.

Off-label uses: Generalized anxiety disorder, social anxiety disorder (pregabalin); diabetic neuropathy (alpha lipoic acid)

📋 Drug Information

Generic Name(s)Alpha Lipoic Acid + Pregabalin
Brand NameCaregalin-M Tablet
ManufacturerHumane Care Pharmaceuticals Pvt. Ltd.
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassNeuropathic pain modulator
Route of AdministrationOral
StorageStore at room temperature (20-25°C), protect from light and moisture.
Shelf LifeAs per manufacturer

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionPregabalin is rapidly absorbed after oral administration; alpha lipoic acid is absorbed in the gastrointestinal tract.
DistributionPregabalin distributes to tissues including brain; alpha lipoic acid distributes to various tissues.
Protein BindingPregabalin: <1%; Alpha lipoic acid: approximately 80-90%
MetabolismPregabalin: minimal hepatic metabolism; Alpha lipoic acid: extensively metabolized in liver via oxidation and conjugation.
Half-LifePregabalin: ~6.3 hours; Alpha lipoic acid: ~30 minutes
ExcretionPregabalin: primarily renal (90% unchanged); Alpha lipoic acid: renal (metabolites)
BioavailabilityPregabalin: >90%; Alpha lipoic acid: ~30% (oral)
Onset of ActionPregabalin: 1-2 weeks for analgesic effect; Alpha lipoic acid: variable
Peak Plasma TimePregabalin: ~1 hour; Alpha lipoic acid: ~1-2 hours
Duration of ActionPregabalin: 6-12 hours; Alpha lipoic acid: 2-4 hours

How It Works

Pregabalin binds to alpha2-delta subunit of voltage-gated calcium channels, reducing calcium influx and neurotransmitter release; Alpha lipoic acid acts as an antioxidant and improves nerve blood flow.

Mechanism Steps

1Pregabalin binds to alpha2-delta subunit of presynaptic voltage-gated calcium channels.
2Reduces calcium influx into nerve terminals.
3Decreases release of excitatory neurotransmitters (e.g., glutamate, norepinephrine, substance P).
4Alpha lipoic acid scavenges free radicals and reduces oxidative stress.
5Improves endothelial function and nerve blood flow.
6Enhances mitochondrial function and glucose uptake.

💡 How to Take caregalin-m tablet

Follow your doctor's prescription exactly.

⚠️ Side Effects of caregalin-m tablet

✅ Common Side Effects

Dizziness
Somnolence
Dry mouth
Peripheral edema
Blurred vision
Weight gain

🚨 Serious Side Effects

Angioedema
Hypersensitivity reactions
Suicidal ideation
Rhabdomyolysis
Heart failure

⚠️ Rare Side Effects

Stevens-Johnson syndrome
Hepatotoxicity
Pancreatitis
Thrombocytopenia

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
CNS depressants Major Enhanced sedation and respiratory depression
Alcohol Major Increased dizziness and sedation
Thiazolidinediones Major Increased risk of fluid retention and heart failure

🚨 Major Interactions

  • Central nervous system depressants
  • Alcohol
  • Thiazolidinediones

⚡ Moderate Interactions

  • Antidiabetic agents
  • Antihypertensives

🍷 Alcohol Interaction

Increased CNS depression and dizziness

🛡️ Safety & Warnings

🚫 Contraindications

Hypersensitivity to pregabalin or alpha lipoic acid; severe renal impairment (CrCl

🤱 Lactation Safety

Pregabalin excreted in breast milk; avoid breastfeeding. Alpha lipoic acid: limited data.

💊 Overdose Management

Supportive care; consider activated charcoal if recent ingestion; hemodialysis may remove pregabalin.

⏰ Missed Dose

Take as soon as remembered unless near next dose; skip missed dose if close to next dose.

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