caldob cream - Uses, Price, Side Effects & Substitutes
What is caldob cream used for?
Anasure Cream (Lidocaine + Calcium Dobesilate) is used to treat CARDIAC. It contains Lidocaine (3% w/w) + Calcium Dobesilate (0.25% w/w), which Lidocaine blocks voltage-gated sodium channels, inhibiting nerve impulse conduct. Always consult your doctor before use. Take as prescribed.
- Generic Name: Lidocaine + Calcium Dobesilate
- Manufacturer: Comed Chemicals Ltd
- Form: Allopathy
- Pregnancy Category: A
- Prescription Required: Yes
๐ caldob cream Uses & Benefits
Hemorrhoids, anal fissures, local pain relief, varicose veins.
Off-label uses: Post-hemorrhoidectomy pain, Minor skin wounds
๐ Drug Information
| Generic Name(s) | Lidocaine + Calcium Dobesilate |
| Brand Name | Anasure Cream |
| Manufacturer | Comed Chemicals Ltd |
| Packaging / Form | Varies by brand (Allopathy) |
| Therapeutic Class | CARDIAC |
| Action Class | Local anesthetic + Capillary stabilizer |
| Route of Administration | Topical |
| Storage | Store at room temperature (20-25ยฐC), away from moisture and heat. |
| Shelf Life | As per manufacturer |
๐ฌ Pharmacology (PK/PD)
Pharmacokinetics
How It Works
Lidocaine blocks voltage-gated sodium channels, inhibiting nerve impulse conduction; Calcium dobesilate reduces capillary permeability and platelet aggregation.
Mechanism Steps
๐ก How to Take caldob cream
Follow your doctor's prescription exactly.
โ ๏ธ Side Effects of caldob cream
โ Common Side Effects
- Burning sensation
- Stinging
- Erythema
- Pruritus
๐จ Serious Side Effects
- Allergic reactions
- Methemoglobinemia (rare)
- Cardiac arrhythmias (systemic toxicity)
โ ๏ธ Rare Side Effects
- Contact dermatitis
- Hypersensitivity reactions
Consult your doctor if you experience any unusual symptoms.
๐ฌ Drug Interactions
| โ ๏ธ Drug | Severity | Effect |
|---|---|---|
| Class I antiarrhythmics | Major | Additive cardiac depression |
| CYP3A4 inhibitors | Moderate | Increased lidocaine levels |
| Beta-blockers | Moderate | Reduced lidocaine clearance |
๐จ Major Interactions
- Class I antiarrhythmics
- Other local anesthetics
โก Moderate Interactions
- CYP3A4 inhibitors
- Beta-blockers
โน๏ธ Minor Interactions
- Cimetidine
- Antacids
๐ฝ๏ธ Food Interactions
No significant food interactions.
๐ท Alcohol Interaction
No known interaction.
๐ก๏ธ Safety & Warnings
๐ซ Contraindications
Hypersensitivity to lidocaine or calcium dobesilate, severe liver disease, open wounds or broken skin at application site.
๐ Monitoring Parameters
Local skin irritation, signs of systemic toxicity (dizziness, blurred vision, seizures).
๐คฑ Lactation Safety
Lidocaine excreted in breast milk in small amounts; calcium dobesilate unknown. Use with caution.
๐ Overdose Management
Discontinue use; symptomatic and supportive care; severe cases may require cardiac monitoring.
โฐ Missed Dose
Apply as soon as remembered; skip if almost time for next dose.