benicort injection - Betamethasone (4mg/ml) medicine

Benicort Injection - Uses, Price, Side Effects

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๐Ÿญ P & B Pharmaceuticals Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 29, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 29, 2026

What is benicort injection used for?

Benicort Injection contains Betamethasone, a corticosteroid that reduces inflammation and suppresses the immune system. It is used to treat respiratory conditions like asthma and allergic reactions, as well as other inflammatory disorders. It works by blocking the release of substances that cause inflammation.

  • Generic Name: Betamethasone
  • Manufacturer: P & B Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š benicort injection Uses & Benefits

Allergic conditions, asthma, COPD exacerbations, inflammatory disorders, autoimmune diseases.

Off-label uses: COVID-19 (severe cases), certain dermatoses, cerebral edema.

๐Ÿ“‹ Drug Information

Generic Name(s)Betamethasone
Brand NameAlerkim
ManufacturerP & B Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassRESPIRATORY
Action ClassGlucocorticoids
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF); protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionWell absorbed orally; peak plasma concentration within 1-2 hours.
DistributionDistributes widely; crosses placenta and enters breast milk.
Protein BindingApproximately 64% bound to plasma proteins.
MetabolismHepatic via CYP3A4.
Half-Life36-54 hours (plasma); biological half-life 36-54 hours.
ExcretionRenal (primarily as metabolites) and fecal.
BioavailabilityHigh oral bioavailability (approximately 100%).
Onset of ActionWithin hours for anti-inflammatory effects.
Peak Plasma Time1-2 hours.
Duration of ActionDuration of action: 3-4 days (single dose).

How It Works

Agonist at glucocorticoid receptors, leading to anti-inflammatory and immunosuppressive effects.

Mechanism Steps

1Betamethasone binds to glucocorticoid receptor (GR) in cytoplasm.
2Receptor-ligand complex translocates to nucleus.
3Complex binds to glucocorticoid response elements (GREs) on DNA.

๐Ÿ’ก How to Take benicort injection

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โœ… ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of benicort injection

โœ… Common Side Effects

  • Increased appetite
  • Weight gain
  • Insomnia
  • Mood changes
  • Fluid retention
  • Hypertension
  • Hyperglycemia

๐Ÿšจ Serious Side Effects

  • Adrenal suppression
  • Osteoporosis
  • Glaucoma
  • Cataracts
  • Peptic ulcer
  • Pancreatitis
  • Psychiatric disturbances

โš ๏ธ Rare Side Effects

  • Avascular necrosis
  • Cushing's syndrome
  • Growth suppression in children
  • Kaposi's sarcoma
  • Anaphylaxis

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Major Increased bleeding risk
NSAIDs Moderate Increased gastrointestinal side effects
Diuretics Moderate Increased risk of hypokalemia

๐Ÿšจ Major Interactions

  • CYP3A4 inducers (e.g., rifampin, phenytoin, carbamazepine)
  • CYP3A4 inhibitors (e.g., ketoconazole, ritonavir)
  • Anticoagulants (e.g., warfarin)
  • NSAIDs (increased GI bleeding risk)
  • Antidiabetic agents (reduced efficacy)
  • Live vaccines (increased infection risk)

โšก Moderate Interactions

  • Diuretics (increased hypokalemia risk)
  • Cardiac glycosides (increased toxicity risk)
  • Amphotericin B (increased hypokalemia)
  • Cholestyramine (reduced absorption)

โ„น๏ธ Minor Interactions

  • Antacids (slight reduction in absorption)
  • Oral contraceptives (increased corticosteroid levels)

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase levels (CYP3A4 inhibition).

๐Ÿท Alcohol Interaction

May increase risk of GI irritation and bleeding.

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Low
Heart
Low
Pregnancy
Category C

๐Ÿšซ Contraindications

Systemic fungal infections, hypersensitivity to betamethasone, live vaccine administration.

๐Ÿ“Š Monitoring Parameters

Blood glucose, blood pressure, electrolytes, signs of infection, adrenal suppression.

๐Ÿคฑ Lactation Safety

Use with caution; excreted in breast milk.

๐Ÿ’Š Overdose Management

Supportive care; no specific antidote; monitor electrolytes and glucose.

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 29, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for benicort injection

View All

Alternative brands with exact same active ingredient (Betamethasone (4mg/ml)):

Medical Note: Always consult your doctor before switching medications.

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