auctista m 500mg/20mg tablet - Metformin (500mg) + Teneligliptin (20mg) medicine

Auctista M 500mg/20mg Tablet - Uses, Price, Side Effects

4.4 (14 reviews)
๐Ÿญ Bioaltus Pharmaceuticals Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Aug 22, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Aug 22, 2026

What is auctista m 500mg/20mg tablet used for?

Auctista M 500mg/20mg Tablet is a combination medicine used to treat type 2 diabetes mellitus. It contains Metformin and Teneligliptin, which work by improving insulin sensitivity and increasing insulin release, thereby helping to control blood sugar levels. It is usually taken once daily with meals.

  • Generic Name: Metformin + Teneligliptin
  • Manufacturer: Bioaltus Pharmaceuticals Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India has the highest number of USFDA-compliant plants outside the USA.

๐Ÿ’Š auctista m 500mg/20mg tablet Uses & Benefits

Type 2 diabetes mellitus as an adjunct to diet and exercise, when monotherapy with metformin or teneligliptin is inadequate.

Off-label uses: Polycystic ovary syndrome (metformin), gestational diabetes (metformin), prevention of type 2 diabetes (metformin).

๐Ÿ“‹ Drug Information

Generic Name(s)Metformin + Teneligliptin
Brand NameAfoglip M 500 Tablet ER
ManufacturerBioaltus Pharmaceuticals Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI DIABETIC
Action ClassAntidiabetic (Biguanide + DPP-4 inhibitor)
Route of AdministrationOral
StorageStore at room temperature (20-25ยฐC), protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionMetformin: Absorbed mainly from small intestine; Teneligliptin: Rapidly absorbed after oral administration.
DistributionMetformin: Low protein binding, distributed into erythrocytes; Teneligliptin: Extensive distribution.
Protein BindingMetformin: Negligible; Teneligliptin: ~70%
MetabolismMetformin: Not metabolized; Teneligliptin: Minimally metabolized via CYP3A4 and FMO3.
Half-LifeMetformin: ~6.2 hours; Teneligliptin: ~24 hours
ExcretionMetformin: Renal (90% unchanged); Teneligliptin: Renal (70% unchanged) and fecal.
BioavailabilityMetformin: 50-60%; Teneligliptin: ~70%
Onset of ActionMetformin: Within days; Teneligliptin: Within 1-2 hours.
Peak Plasma TimeMetformin: 2-4 hours (ER); Teneligliptin: 1-2 hours
Duration of ActionMetformin: Up to 24 hours; Teneligliptin: >24 hours

How It Works

Metformin: Decreases hepatic glucose production, increases insulin sensitivity; Teneligliptin: Inhibits DPP-4, increasing incretin levels (GLP-1, GIP), enhancing insulin secretion and decreasing glucagon.

Mechanism Steps

1Metformin activates AMPK in hepatocytes, reducing gluconeogenesis and glycogenolysis.
2Metformin increases insulin sensitivity in peripheral tissues (muscle, adipose).
3Metformin decreases intestinal glucose absorption.

๐Ÿ’ก How to Take auctista m 500mg/20mg tablet

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โŒ ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of auctista m 500mg/20mg tablet

โœ… Common Side Effects

  • Nausea
  • Diarrhea
  • Abdominal discomfort
  • Headache
  • Nasopharyngitis
  • Hypoglycemia (when combined with other agents)

๐Ÿšจ Serious Side Effects

  • Lactic acidosis
  • Pancreatitis
  • Severe hypersensitivity reactions
  • Acute renal failure
  • Hepatic injury

โš ๏ธ Rare Side Effects

  • Vitamin B12 deficiency
  • Metallic taste
  • Urticaria
  • Angioedema
  • Stevens-Johnson syndrome

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Insulin Major Increased risk of hypoglycemia
Sulfonylureas Major Increased risk of hypoglycemia
Corticosteroids Moderate Reduced hypoglycemic effect
Diuretics Moderate Possible hyperglycemia

๐Ÿšจ Major Interactions

  • Contrast agents (iodinated)
  • Cimetidine
  • Cationic drugs eliminated by renal tubular secretion

โšก Moderate Interactions

  • Insulin
  • Sulfonylureas
  • Thiazolidinediones
  • Alcohol

โ„น๏ธ Minor Interactions

  • Furosemide
  • Nifedipine
  • Topiramate

๐Ÿฝ๏ธ Food Interactions

Alcohol, High-fat meals may affect absorption

๐Ÿท Alcohol Interaction

Increased risk of lactic acidosis with metformin

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Moderate
Heart
Low
Pregnancy
Category A

๐Ÿšซ Contraindications

Severe renal impairment (eGFR <30 mL/min), metabolic acidosis, acute or chronic metabolic acidosis, diabetic ketoacidosis, hypersensitivity, hepatic impairment, acute myocardial infarction, sepsis.

๐Ÿ“Š Monitoring Parameters

Blood glucose, HbA1c, renal function (eGFR), liver function, vitamin B12 levels (long-term metformin), signs of lactic acidosis.

๐Ÿคฑ Lactation Safety

Metformin excreted in milk; Teneligliptin unknown; avoid breastfeeding.

๐Ÿ’Š Overdose Management

Supportive care; monitor blood glucose and lactate; hemodialysis may remove metformin.

โฐ Missed Dose

Take as soon as remembered unless near next dose; skip missed dose if next dose is due.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Last reviewed on: Aug 22, 2026

๐Ÿ”— View Profile

โญ User Reviews

Happy Patient Jul 10, 2026

Found this to be a helpful product. Good results.

Trusted Reviewer Jul 10, 2026

Found this to be a helpful product. Good results.

Verified User Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

Verified User Jul 10, 2026

Good quality medicine. Satisfied with the outcome.

Certified Buyer Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

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