asevator 10mg tablet - Uses, Price, Side Effects & Substitutes
What is asevator 10mg tablet used for?
Azin 10mg Tablet (Asenapine) is used to treat NEURO CNS. It contains Asenapine (10mg), which Antagonist at dopamine D2 and serotonin 5-HT2A receptors; also has affinity for . Always consult your doctor before use. Take as prescribed.
- Generic Name: Asenapine
- Manufacturer: Ryon Pharma
- Form: Allopathy
- Pregnancy Category: A
- Prescription Required: Yes
๐ asevator 10mg tablet Uses & Benefits
Schizophrenia; acute treatment of manic or mixed episodes associated with bipolar I disorder.
Off-label uses: Treatment-resistant depression; Tourette syndrome; borderline personality disorder.
๐ Drug Information
| Generic Name(s) | Asenapine |
| Brand Name | Azin 10mg Tablet |
| Manufacturer | Ryon Pharma |
| Packaging / Form | Varies by brand (Allopathy) |
| Therapeutic Class | NEURO CNS |
| Action Class | Atypical Antipsychotics |
| Route of Administration | Sublingual (tablet placed under tongue until dissolved). |
| Storage | Store at 20-25ยฐC (68-77ยฐF); protect from moisture. |
| Shelf Life | As per manufacturer |
๐ฌ Pharmacology (PK/PD)
Pharmacokinetics
How It Works
Antagonist at dopamine D2 and serotonin 5-HT2A receptors; also has affinity for other receptors.
Mechanism Steps
๐ก How to Take asevator 10mg tablet
Follow your doctor's prescription exactly.
โ ๏ธ Side Effects of asevator 10mg tablet
โ Common Side Effects
- Somnolence
- Dizziness
- Extrapyramidal symptoms
- Weight gain
- Increased appetite
- Dry mouth
- Constipation
- Dysgeusia
๐จ Serious Side Effects
- Neuroleptic malignant syndrome
- Tardive dyskinesia
- QT prolongation
- Seizures
- Hyperglycemia
- Dyslipidemia
โ ๏ธ Rare Side Effects
- Hepatic failure
- Agranulocytosis
- Pancreatitis
- Priapism
- Allergic reactions
Consult your doctor if you experience any unusual symptoms.
๐ฌ Drug Interactions
| โ ๏ธ Drug | Severity | Effect |
|---|---|---|
| Fluvoxamine | Major | Increased asenapine levels due to CYP1A2 inhibition |
| Carbamazepine | Major | Decreased asenapine levels due to CYP1A2 induction |
| Levodopa | Major | Antagonism of dopaminergic effects |
| Alcohol | Moderate | Increased CNS depression and sedation |
| Grapefruit juice | Minor | Possible increase in asenapine levels |
๐จ Major Interactions
- CYP1A2 inhibitors (e.g., fluvoxamine)
- CYP1A2 inducers (e.g., carbamazepine)
- Dopamine agonists
- Levodopa
โก Moderate Interactions
- Antihypertensives
- CNS depressants (e.g., alcohol, benzodiazepines)
- QTc-prolonging drugs
โน๏ธ Minor Interactions
- CYP2D6 substrates
- CYP3A4 substrates
๐ฝ๏ธ Food Interactions
Grapefruit juice may increase asenapine levels; avoid high-fat meals within 10 minutes of administration.
๐ท Alcohol Interaction
Avoid alcohol; may increase CNS depression and hypotensive effects.
๐ก๏ธ Safety & Warnings
๐ซ Contraindications
Hypersensitivity to asenapine or any excipients; severe hepatic impairment.
๐ Monitoring Parameters
Mental status, blood pressure, heart rate, ECG (QTc interval), liver function tests, blood glucose, lipid profile, weight.
๐คฑ Lactation Safety
Not recommended; excreted in breast milk in animal studies.
๐ Overdose Management
Supportive care; monitor vital signs, ECG, and mental status; no specific antidote.
โฐ Missed Dose
Take as soon as remembered; if close to next dose, skip missed dose; do not double dose.
๐จโโ๏ธ Reviewed by Expert
๐ Substitutes for asevator 10mg tablet
View AllAlternative brands with exact same active ingredient (Asenapine (10mg)):
-
azin 10mg tabletIntas Pharmaceuticals Ltd โน85.00 4.5% CHEAPER
-
welenuf 10mg sublingual tabletTorrent Pharmaceuticals Ltd โน85.00 4.5% CHEAPER
-
asenapt 10 sublingual tabletSun Pharmaceutical Industries Ltd โน89.00 SAME PRICE
Medical Note: Always consult your doctor before switching medications.