asar-ct 40/12.5 tablet - Azilsartan medoxomil (40mg) + Chlorthalidone (12.5mg) medicine

asar-ct 40/12.5 tablet - Uses, Price, Side Effects & Substitutes

No reviews yet
๐Ÿญ Glenmark Pharmaceuticals Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is asar-ct 40/12.5 tablet used for?

Asar-CT 40/12.5 Tablet (Azilsartan medoxomil + Chlorthalidone) is used to treat CARDIAC. It contains Azilsartan medoxomil (40mg) + Chlorthalidone (12.5mg), which Azilsartan blocks AT1 receptor, reducing vasoconstriction and aldosterone secret. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Azilsartan medoxomil + Chlorthalidone
  • Manufacturer: Glenmark Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

๐Ÿ’Š asar-ct 40/12.5 tablet Uses & Benefits

Hypertension (alone or in combination).

Off-label uses: Heart failure (limited data).

๐Ÿ“‹ Drug Information

Generic Name(s)Azilsartan medoxomil + Chlorthalidone
Brand NameAsar-CT 40/12.5 Tablet
ManufacturerGlenmark Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassAngiotensin II receptor blocker (ARB) + Thiazide-like diuretic
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF); protect from moisture and light.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionAzilsartan medoxomil is rapidly absorbed; Chlorthalidone is well absorbed orally.
DistributionAzilsartan: Vd ~16 L; Chlorthalidone: Vd ~3-9 L/kg.
Protein BindingAzilsartan: >99%; Chlorthalidone: 75% bound to albumin.
MetabolismAzilsartan: hydrolyzed to active form, then glucuronidated; Chlorthalidone: minimal hepatic metabolism.
Half-LifeAzilsartan: ~11 hours; Chlorthalidone: 40-60 hours.
ExcretionAzilsartan: 55% feces, 42% urine; Chlorthalidone: primarily urine (50-70% unchanged).
BioavailabilityAzilsartan: ~60%; Chlorthalidone: ~64%.
Onset of ActionAzilsartan: 2-4 weeks for full effect; Chlorthalidone: 2-3 hours.
Peak Plasma TimeAzilsartan: 1.5-3 hours; Chlorthalidone: 2-4 hours.
Duration of ActionAzilsartan: 24 hours; Chlorthalidone: 24-72 hours.

How It Works

Azilsartan blocks AT1 receptor, reducing vasoconstriction and aldosterone secretion; Chlorthalidone inhibits Na+/Cl- cotransporter in distal tubule, increasing diuresis.

Mechanism Steps

1Azilsartan medoxomil is hydrolyzed to active azilsartan.
2Azilsartan selectively blocks AT1 receptor, preventing angiotensin II binding.
3Blockade of AT1 receptor leads to vasodilation, reduced aldosterone secretion, and decreased blood pressure.

๐Ÿ’ก How to Take asar-ct 40/12.5 tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of asar-ct 40/12.5 tablet

โœ… Common Side Effects

  • Dizziness
  • Fatigue
  • Diarrhea
  • Hypokalemia
  • Hyperuricemia

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Acute renal failure
  • Hyperkalemia
  • Hypotension
  • Syncope

โš ๏ธ Rare Side Effects

  • Hepatotoxicity
  • Pancreatitis
  • Stevens-Johnson syndrome
  • Anaphylaxis

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Lithium Major Increased lithium toxicity risk
NSAIDs Major Reduced antihypertensive effect, increased renal impairment risk
ACE inhibitors Major Increased risk of hypotension, hyperkalemia, renal dysfunction
Aliskiren Major Increased risk of hypotension, hyperkalemia, renal dysfunction
Potassium-sparing diuretics Major Increased risk of hyperkalemia
Corticosteroids Moderate Reduced diuretic effect
Amphotericin B Moderate Increased risk of hypokalemia
Loop diuretics Moderate Additive diuretic effect, electrolyte imbalance
Dofetilide Moderate Increased risk of torsades de pointes due to hypokalemia
Antidiabetic agents Minor May alter blood glucose control
Alcohol Minor Additive hypotensive effect
Barbiturates Minor Additive hypotensive effect

๐Ÿšจ Major Interactions

  • Lithium
  • NSAIDs
  • ACE inhibitors
  • Aliskiren
  • Potassium-sparing diuretics

โšก Moderate Interactions

  • Corticosteroids
  • Amphotericin B
  • Loop diuretics
  • Dofetilide

โ„น๏ธ Minor Interactions

  • Antidiabetic agents
  • Alcohol
  • Barbiturates

๐Ÿฝ๏ธ Food Interactions

Avoid high-potassium foods; take with or without food.

๐Ÿท Alcohol Interaction

May potentiate orthostatic hypotension.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Anuria, hypersensitivity to sulfonamides, severe renal impairment (CrCl <30 mL/min), pregnancy.

๐Ÿ“Š Monitoring Parameters

Blood pressure, serum potassium, renal function, blood glucose, uric acid.

๐Ÿคฑ Lactation Safety

Not recommended; Chlorthalidone excreted in milk, Azilsartan unknown.

๐Ÿ’Š Overdose Management

Symptomatic and supportive; monitor electrolytes, BP, renal function; consider gastric lavage.

โฐ Missed Dose

Take as soon as remembered; if near next dose, skip missed dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

๐Ÿ˜Š Was this information helpful?

Browse Medicines A-Z

Search our extensive medical database alphabetically.

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory
SaathiMed App
SaathiMed App Consult doctors & order medicines faster
Install