amoline h 5mg/12.5mg tablet - Amlodipine (5mg) + Hydrochlorothiazide (12.5mg) medicine

amoline h 5mg/12.5mg tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Zeelab Pharmacy Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 28, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 28, 2026

What is amoline h 5mg/12.5mg tablet used for?

Amlong-H Tablet (Amlodipine + Hydrochlorothiazide) is used to treat CARDIAC. It contains Amlodipine (5mg) + Hydrochlorothiazide (12.5mg), which Amlodipine inhibits calcium influx across cell membranes, causing vasodilation; . Always consult your doctor before use. Take as prescribed.

  • Generic Name: Amlodipine + Hydrochlorothiazide
  • Manufacturer: Zeelab Pharmacy Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The first generic medicine was introduced in India in 1970 after the Patents Act was amended.

๐Ÿ’Š amoline h 5mg/12.5mg tablet Uses & Benefits

Hypertension (alone or in combination); not for initial therapy

Off-label uses: Chronic stable angina (amlodipine alone); heart failure (amlodipine alone)

๐Ÿ“‹ Drug Information

Generic Name(s)Amlodipine + Hydrochlorothiazide
Brand NameAmlong-H Tablet
ManufacturerZeelab Pharmacy Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassCARDIAC
Action ClassCalcium channel blocker + Thiazide diuretic
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF); protect from light and moisture
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionAmlodipine: Well absorbed after oral administration; Hydrochlorothiazide: Well absorbed (65-75%)
DistributionAmlodipine: Extensive distribution; Hydrochlorothiazide: Crosses placenta, not blood-brain barrier
Protein BindingAmlodipine: ~93%; Hydrochlorothiazide: ~40-68%
MetabolismAmlodipine: Extensive hepatic metabolism (CYP3A4); Hydrochlorothiazide: Not metabolized
Half-LifeAmlodipine: 30-50 hours; Hydrochlorothiazide: 6-15 hours
ExcretionAmlodipine: 60% urine, 20-25% feces; Hydrochlorothiazide: Primarily urine (unchanged)
BioavailabilityAmlodipine: 64-90%; Hydrochlorothiazide: 65-75%
Onset of ActionAmlodipine: 2-4 hours; Hydrochlorothiazide: 2 hours
Peak Plasma TimeAmlodipine: 6-12 hours; Hydrochlorothiazide: 4 hours
Duration of ActionAmlodipine: 24 hours; Hydrochlorothiazide: 6-12 hours

How It Works

Amlodipine inhibits calcium influx across cell membranes, causing vasodilation; Hydrochlorothiazide inhibits sodium reabsorption in distal tubules, reducing plasma volume

Mechanism Steps

1Amlodipine binds to L-type calcium channels in vascular smooth muscle and cardiac muscle
2Inhibits calcium influx, reducing intracellular calcium
3Causes relaxation of vascular smooth muscle, leading to vasodilation and decreased peripheral resistance

๐Ÿ’ก How to Take amoline h 5mg/12.5mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of amoline h 5mg/12.5mg tablet

โœ… Common Side Effects

  • Edema (ankle swelling)
  • Dizziness
  • Headache
  • Fatigue
  • Nausea
  • Flushing
  • Palpitations
  • Hypokalemia
  • Hyperuricemia
  • Increased urination

๐Ÿšจ Serious Side Effects

  • Severe hypotension
  • Syncope
  • Arrhythmias
  • Acute renal failure
  • Pancreatitis
  • Stevens-Johnson syndrome
  • Toxic epidermal necrolysis
  • Angioedema

โš ๏ธ Rare Side Effects

  • Hepatotoxicity
  • Leukopenia
  • Thrombocytopenia
  • Anaphylaxis
  • Photosensitivity
  • Acute angle-closure glaucoma

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
CYP3A4 inhibitors (e.g., ketoconazole) Major Increased amlodipine levels, risk of toxicity
CYP3A4 inducers (e.g., rifampin) Major Decreased amlodipine efficacy
Lithium Major Increased lithium toxicity risk
Digoxin Major Increased digoxin levels, risk of toxicity
NSAIDs Moderate Reduced antihypertensive effect, increased renal impairment risk
Corticosteroids Moderate Hypokalemia, reduced diuretic effect
Cholestyramine Moderate Reduced hydrochlorothiazide absorption
Alcohol Minor Increased orthostatic hypotension

๐Ÿšจ Major Interactions

  • CYP3A4 inhibitors (e.g., ketoconazole, itraconazole, ritonavir)
  • CYP3A4 inducers (e.g., rifampin, carbamazepine)
  • Lithium
  • Digoxin
  • Other antihypertensives (additive effect)

โšก Moderate Interactions

  • NSAIDs
  • Corticosteroids
  • Amphotericin B
  • Cholestyramine
  • Colestipol

โ„น๏ธ Minor Interactions

  • Calcium supplements
  • Vitamin D
  • Antacids

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase amlodipine levels; avoid high-sodium foods

๐Ÿท Alcohol Interaction

May potentiate orthostatic hypotension; avoid excessive alcohol

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to amlodipine, hydrochlorothiazide, or sulfonamides; anuria; severe renal impairment; hypercalcemia; symptomatic hypotension; cardiogenic shock

๐Ÿ“Š Monitoring Parameters

Blood pressure, heart rate, serum electrolytes (K+, Na+, Ca2+), renal function, hepatic function, blood glucose, uric acid

๐Ÿคฑ Lactation Safety

Amlodipine excreted in milk; hydrochlorothiazide may suppress lactation; avoid or use with caution

๐Ÿ’Š Overdose Management

Gastric lavage, activated charcoal; monitor BP, ECG; treat hypotension with fluids and vasopressors; correct electrolyte imbalances

โฐ Missed Dose

Take as soon as remembered; if close to next dose, skip missed dose; do not double dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 28, 2026

๐Ÿ”— View Profile

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