amitop m 5mg/1500mcg tablet - Amitriptyline (5mg) + Methylcobalamin (1500mcg) medicine

amitop m 5mg/1500mcg tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Tas Med India Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 28, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 28, 2026

What is amitop m 5mg/1500mcg tablet used for?

Amnurite 10 Tablet SR (Amitriptyline + Methylcobalamin) is used to treat NEURO CNS. It contains Amitriptyline (5mg) + Methylcobalamin (1500mcg), which Amitriptyline: Inhibits reuptake of serotonin and norepinephrine; Methylcobalami. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Amitriptyline + Methylcobalamin
  • Manufacturer: Tas Med India Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: A
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š amitop m 5mg/1500mcg tablet Uses & Benefits

Depression, neuropathic pain, diabetic neuropathy, fibromyalgia

Off-label uses: Migraine prophylaxis, chronic pain, insomnia, anxiety disorders

๐Ÿ“‹ Drug Information

Generic Name(s)Amitriptyline + Methylcobalamin
Brand NameAmnurite 10 Tablet SR
ManufacturerTas Med India Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassTricyclic antidepressant + Vitamin B12 analogue
Route of AdministrationOral
StorageStore at 20-25ยฐC, protect from light and moisture
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionAmitriptyline: Well absorbed orally; Methylcobalamin: Absorbed via active transport in ileum
DistributionAmitriptyline: Widely distributed, crosses blood-brain barrier; Methylcobalamin: Distributed to tissues, stored in liver
Protein BindingAmitriptyline: ~96% bound to plasma proteins; Methylcobalamin: Binds to transcobalamin
MetabolismAmitriptyline: Hepatic via CYP2D6, CYP3A4, CYP1A2; Methylcobalamin: Converted to coenzyme forms in cells
Half-LifeAmitriptyline: 13-36 hours; Methylcobalamin: ~6 days
ExcretionAmitriptyline: Renal (metabolites); Methylcobalamin: Biliary and renal
BioavailabilityAmitriptyline: 30-60%; Methylcobalamin: Variable, dose-dependent
Onset of ActionAmitriptyline: 2-4 weeks for antidepressant effect; Methylcobalamin: Days to weeks for neuropathy
Peak Plasma TimeAmitriptyline: 2-8 hours; Methylcobalamin: 3-8 hours
Duration of ActionAmitriptyline: 24 hours; Methylcobalamin: Several days

How It Works

Amitriptyline: Inhibits reuptake of serotonin and norepinephrine; Methylcobalamin: Coenzyme for myelin synthesis and nerve regeneration

Mechanism Steps

1Amitriptyline inhibits reuptake of serotonin and norepinephrine at presynaptic terminals
2Increased synaptic levels of serotonin and norepinephrine enhance neurotransmission
3Downregulation of postsynaptic receptors over time contributes to antidepressant effect

๐Ÿ’ก How to Take amitop m 5mg/1500mcg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of amitop m 5mg/1500mcg tablet

โœ… Common Side Effects

  • Dry mouth
  • Drowsiness
  • Dizziness
  • Constipation
  • Blurred vision
  • Weight gain
  • Urinary retention

๐Ÿšจ Serious Side Effects

  • QT prolongation
  • Arrhythmias
  • Seizures
  • Serotonin syndrome
  • Suicidal thoughts
  • Agranulocytosis

โš ๏ธ Rare Side Effects

  • Hepatotoxicity
  • Paralytic ileus
  • Bone marrow suppression
  • Allergic reactions

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
MAOIs Major Hypertensive crisis, serotonin syndrome
CYP2D6 inhibitors Major Increased amitriptyline toxicity
CYP3A4 inhibitors Major Increased amitriptyline levels
CYP1A2 inhibitors Major Increased amitriptyline levels
Other serotonergic drugs Major Serotonin syndrome
Anticholinergics Major Additive anticholinergic effects
CNS depressants Major Enhanced sedation
Anticoagulants Moderate Increased anticoagulant effect
Antihypertensives Moderate Additive hypotension
Sympathomimetics Moderate Hypertension, arrhythmias
Thyroid medications Moderate Increased cardiac effects
Quinolones Moderate Increased risk of QT prolongation
Cimetidine Minor Increased amitriptyline levels
Methylphenidate Minor Increased amitriptyline levels
Oral contraceptives Minor Reduced amitriptyline efficacy

๐Ÿšจ Major Interactions

  • MAOIs
  • CYP2D6 inhibitors
  • CYP3A4 inhibitors
  • CYP1A2 inhibitors
  • Other serotonergic drugs
  • Anticholinergics
  • CNS depressants

โšก Moderate Interactions

  • Anticoagulants
  • Antihypertensives
  • Sympathomimetics
  • Thyroid medications
  • Quinolones

โ„น๏ธ Minor Interactions

  • Cimetidine
  • Methylphenidate
  • Oral contraceptives

๐Ÿฝ๏ธ Food Interactions

Grapefruit juice may increase amitriptyline levels; high-fiber foods may reduce absorption

๐Ÿท Alcohol Interaction

Increased CNS depression; avoid alcohol

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Recent MI, concurrent MAOI use, narrow-angle glaucoma, urinary retention, hypersensitivity

๐Ÿ“Š Monitoring Parameters

ECG, liver function, serum drug levels, mental status, blood pressure

๐Ÿคฑ Lactation Safety

Amitriptyline excreted in milk; use with caution. Methylcobalamin safe.

๐Ÿ’Š Overdose Management

Activated charcoal, supportive care, physostigmine for anticholinergic symptoms, sodium bicarbonate for arrhythmias

โฐ Missed Dose

Take as soon as remembered unless near next dose; skip if close to next dose. Do not double.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 28, 2026

๐Ÿ”— View Profile

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