amigatin ls 100mg/10mg tablet - Gabapentin (100mg) + Amitriptyline (10mg) medicine

amigatin ls 100mg/10mg tablet - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Crescent Therapeutics Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 30, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 30, 2026

What is amigatin ls 100mg/10mg tablet used for?

Amigaba LS Tablet (Gabapentin + Amitriptyline) is used to treat NEURO CNS. It contains Gabapentin (100mg) + Amitriptyline (10mg), which Gabapentin: Binds to ฮฑ2ฮด subunit of voltage-gated calcium channels, reducing n. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Gabapentin + Amitriptyline
  • Manufacturer: Crescent Therapeutics Ltd
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? India is the largest provider of generic medicines globally, supplying over 50% of global vaccine demand.

๐Ÿ’Š amigatin ls 100mg/10mg tablet Uses & Benefits

Neuropathic pain, fibromyalgia, depression, anxiety, migraine prophylaxis.

Off-label uses: Chronic pain, restless legs syndrome, social anxiety disorder.

๐Ÿ“‹ Drug Information

Generic Name(s)Gabapentin + Amitriptyline
Brand NameAmigaba LS Tablet
ManufacturerCrescent Therapeutics Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassNEURO CNS
Action ClassAnticonvulsant + Tricyclic Antidepressant
Route of AdministrationOral
StorageStore at 20-25ยฐC, protect from light and moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionGabapentin: Absorbed via L-amino acid transporter; Amitriptyline: Well absorbed orally.
DistributionGabapentin: Crosses blood-brain barrier; Amitriptyline: Widely distributed, high protein binding.
Protein BindingGabapentin: <3%; Amitriptyline: 90-95%
MetabolismGabapentin: Not significantly metabolized; Amitriptyline: Hepatic via CYP2D6, CYP3A4, CYP2C19
Half-LifeGabapentin: 5-7 hours; Amitriptyline: 10-28 hours
ExcretionGabapentin: Renal (unchanged); Amitriptyline: Renal (metabolites)
BioavailabilityGabapentin: 60% (dose-dependent); Amitriptyline: 45-60%
Onset of ActionGabapentin: 1-2 weeks; Amitriptyline: 2-4 weeks
Peak Plasma TimeGabapentin: 2-3 hours; Amitriptyline: 2-6 hours
Duration of ActionGabapentin: 6-8 hours; Amitriptyline: 24 hours

How It Works

Gabapentin: Binds to ฮฑ2ฮด subunit of voltage-gated calcium channels, reducing neurotransmitter release. Amitriptyline: Inhibits reuptake of serotonin and norepinephrine, blocks histamine, acetylcholine, and ฮฑ1-adrenergic receptors.

Mechanism Steps

1Gabapentin binds to ฮฑ2ฮด subunit of voltage-gated calcium channels.
2Reduces calcium influx and neurotransmitter release (glutamate, substance P).
3Amitriptyline inhibits serotonin and norepinephrine reuptake.

๐Ÿ’ก How to Take amigatin ls 100mg/10mg tablet

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of amigatin ls 100mg/10mg tablet

โœ… Common Side Effects

  • Drowsiness
  • Dizziness
  • Dry mouth
  • Blurred vision
  • Constipation
  • Weight gain

๐Ÿšจ Serious Side Effects

  • Suicidal thoughts
  • Seizures
  • QT prolongation
  • Serotonin syndrome
  • Agranulocytosis

โš ๏ธ Rare Side Effects

  • Hepatotoxicity
  • Pancreatitis
  • Rhabdomyolysis
  • Stevens-Johnson syndrome

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
MAOIs Major Risk of serotonin syndrome, hypertensive crisis
CNS depressants Major Enhanced sedation, respiratory depression
Anticholinergics Major Additive anticholinergic effects
CYP2D6 inhibitors Moderate Increased amitriptyline levels
CYP3A4 inhibitors Moderate Increased amitriptyline levels
Anticoagulants Moderate Increased bleeding risk
Cimetidine Minor Increased amitriptyline levels
Antacids Minor Decreased gabapentin absorption

๐Ÿšจ Major Interactions

  • MAOIs
  • CNS depressants
  • Anticholinergics

โšก Moderate Interactions

  • CYP2D6 inhibitors
  • CYP3A4 inhibitors
  • Anticoagulants

โ„น๏ธ Minor Interactions

  • Cimetidine
  • Antacids

๐Ÿฝ๏ธ Food Interactions

Gabapentin: High-fat meal may decrease absorption; Amitriptyline: Avoid grapefruit juice.

๐Ÿท Alcohol Interaction

Increased CNS depression; avoid alcohol.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity, recent MI, MAOI use within 14 days, narrow-angle glaucoma, urinary retention, severe hepatic impairment.

๐Ÿ“Š Monitoring Parameters

ECG, liver function, renal function, serum drug levels (amitriptyline), suicidal ideation, sedation.

๐Ÿคฑ Lactation Safety

Not recommended; excreted in breast milk.

๐Ÿ’Š Overdose Management

Supportive care; activated charcoal, ECG monitoring, benzodiazepines for seizures, sodium bicarbonate for arrhythmias.

โฐ Missed Dose

Take as soon as remembered unless near next dose; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 30, 2026

๐Ÿ”— View Profile

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