alersafe m oral suspension - Levocetirizine (2.5mg) + Montelukast (4mg) medicine

Alersafe M Oral Suspension - Uses, Price, Side Effects

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๐Ÿญ Medrix Pharma Pvt Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 28, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Jun 28, 2026

What is alersafe m oral suspension used for?

Alersafe M Oral Suspension is a combination medicine containing Levocetirizine (an antihistamine) and Montelukast (a leukotriene receptor antagonist). It is used to relieve symptoms of allergic rhinitis such as sneezing, runny nose, and itching, and to prevent asthma attacks. Levocetirizine blocks histamine, while Montelukast reduces inflammation in the airways.

  • Generic Name: Levocetirizine + Montelukast
  • Manufacturer: Medrix Pharma Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: B
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š alersafe m oral suspension Uses & Benefits

Seasonal and perennial allergic rhinitis; asthma prophylaxis

Off-label uses: Urticaria, Eosinophilic esophagitis

๐Ÿ“‹ Drug Information

Generic Name(s)Levocetirizine + Montelukast
Brand NameAllercet-M Tablet
ManufacturerMedrix Pharma Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassRESPIRATORY
Action ClassAntihistamine + Leukotriene Receptor Antagonist
Route of AdministrationOral
StorageStore at 20-25ยฐC (68-77ยฐF); protect from light and moisture
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed from the gastrointestinal tract
DistributionDistributed widely; crosses blood-brain barrier minimally for levocetirizine
Protein BindingLevocetirizine: ~90%; Montelukast: >99%
MetabolismLevocetirizine: minimally metabolized; Montelukast: extensively metabolized by CYP3A4 and CYP2C9
Half-LifeLevocetirizine: 7-8 hours; Montelukast: 2.7-5.5 hours
ExcretionLevocetirizine: primarily renal (85%); Montelukast: primarily biliary
BioavailabilityLevocetirizine: ~100%; Montelukast: ~64% (oral)
Onset of ActionLevocetirizine: 1 hour; Montelukast: within hours
Peak Plasma TimeLevocetirizine: 0.9-1.5 hours; Montelukast: 3-4 hours
Duration of ActionLevocetirizine: 24 hours; Montelukast: 24 hours

How It Works

Levocetirizine selectively inhibits peripheral H1 receptors; Montelukast antagonizes leukotriene D4 at CysLT1 receptors

Mechanism Steps

1Levocetirizine binds to H1 receptors, blocking histamine action
2Montelukast binds to CysLT1 receptors, blocking leukotriene D4
3Reduction of nasal congestion, sneezing, and bronchoconstriction

๐Ÿ’ก How to Take alersafe m oral suspension

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โœ… ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of alersafe m oral suspension

โœ… Common Side Effects

  • Headache
  • Drowsiness
  • Dry mouth
  • Cough
  • Pharyngitis

๐Ÿšจ Serious Side Effects

  • Angioedema
  • Anaphylaxis
  • Neuropsychiatric events (agitation, depression)

โš ๏ธ Rare Side Effects

  • Hepatitis
  • Thrombocytopenia
  • Seizures

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Warfarin Moderate Increased risk of bleeding
Theophylline Moderate Increased theophylline levels
Ketoconazole Minor Reduced montelukast metabolism

๐Ÿšจ Major Interactions

  • CYP3A4 inducers (e.g., Rifampin)
  • CYP2C9 inducers (e.g., Phenobarbital)

โšก Moderate Interactions

  • Gemfibrozil
  • Itraconazole
  • Warfarin

โ„น๏ธ Minor Interactions

  • Theophylline
  • Oral contraceptives

๐Ÿฝ๏ธ Food Interactions

Montelukast absorption decreased by high-fat meal; take on empty stomach

๐Ÿท Alcohol Interaction

Levocetirizine may potentiate CNS depression

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Low
Heart
Low
Pregnancy
Category B

๐Ÿšซ Contraindications

Hypersensitivity to any component; severe renal impairment (CrCl <10 mL/min) for levocetirizine

๐Ÿ“Š Monitoring Parameters

Renal function, hepatic function, signs of neuropsychiatric events

๐Ÿคฑ Lactation Safety

Levocetirizine excreted in breast milk; caution advised

๐Ÿ’Š Overdose Management

Symptomatic and supportive; no specific antidote

โฐ Missed Dose

Take as soon as remembered; skip if almost time for next dose; do not double

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 28, 2026

๐Ÿ”— View Profile

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