airtio rotacap - Tiotropium (18mcg) medicine

airtio rotacap - Uses, Price, Side Effects & Substitutes

No reviews yet
๐Ÿญ Glenmark Pharmaceuticals Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is airtio rotacap used for?

Aerotrop Inhalation (Tiotropium) is used to treat RESPIRATORY. It contains Tiotropium (18mcg), which Long-acting muscarinic antagonist (LAMA) that blocks acetylcholine at M3 recepto. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Tiotropium
  • Manufacturer: Glenmark Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

๐Ÿ’Š airtio rotacap Uses & Benefits

Maintenance treatment of COPD (chronic bronchitis and emphysema), reduction of exacerbations in COPD.

Off-label uses: Asthma (not approved in many countries), cystic fibrosis.

๐Ÿ“‹ Drug Information

Generic Name(s)Tiotropium
Brand NameAerotrop Inhalation
ManufacturerGlenmark Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassRESPIRATORY
Action ClassAnticholinergic - COPD
Route of AdministrationInhalation (oral inhalation via HandiHaler device)
StorageStore at 25ยฐC (77ยฐF); excursions permitted to 15-30ยฐC (59-86ยฐF). Protect from moisture.
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionInhaled tiotropium is absorbed slowly from the lungs, reaching peak plasma concentrations within 5-7 minutes.
DistributionApproximately 72% bound to plasma proteins. Volume of distribution is 32 L/kg.
Protein Binding72%
MetabolismMinimally metabolized via cytochrome P450 (CYP2D6 and CYP3A4) to inactive metabolites.
Half-Life5-6 days
ExcretionPrimarily unchanged drug excreted in urine (14%) and feces (86%).
Bioavailability19.5% (inhalation)
Onset of Action30 minutes
Peak Plasma Time5-7 minutes
Duration of Action24 hours

How It Works

Long-acting muscarinic antagonist (LAMA) that blocks acetylcholine at M3 receptors in bronchial smooth muscle, causing bronchodilation.

Mechanism Steps

1Inhaled tiotropium binds to M3 muscarinic receptors on bronchial smooth muscle.
2Blocks acetylcholine from binding, preventing receptor activation.
3Inhibits Gq/11 protein-mediated signaling, reducing intracellular calcium.

๐Ÿ’ก How to Take airtio rotacap

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of airtio rotacap

โœ… Common Side Effects

  • Dry mouth
  • Constipation
  • Cough
  • Pharyngitis
  • Sinusitis

๐Ÿšจ Serious Side Effects

  • Paradoxical bronchospasm
  • Urinary retention
  • Angle-closure glaucoma
  • Atrial fibrillation

โš ๏ธ Rare Side Effects

  • Anaphylaxis
  • Angioedema
  • Rash
  • Urticaria

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Ipratropium Major Additive anticholinergic effects, increased risk of dry mouth, urinary retention.
Quinidine Major Increased tiotropium exposure due to CYP2D6 inhibition.
Ketoconazole Moderate Increased tiotropium exposure due to CYP3A4 inhibition.
Diphenhydramine Moderate Additive anticholinergic effects.

๐Ÿšจ Major Interactions

  • Anticholinergic drugs (e.g., ipratropium, atropine)
  • CYP2D6 inhibitors (e.g., quinidine, fluoxetine)

โšก Moderate Interactions

  • CYP3A4 inhibitors (e.g., ketoconazole, ritonavir)
  • Antihistamines (e.g., diphenhydramine)

โ„น๏ธ Minor Interactions

  • Beta-agonists
  • Corticosteroids

๐Ÿฝ๏ธ Food Interactions

No significant food interactions.

๐Ÿท Alcohol Interaction

No known interaction.

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to tiotropium or any component, history of hypersensitivity to atropine or its derivatives.

๐Ÿ“Š Monitoring Parameters

Lung function (FEV1), exacerbation frequency, signs of anticholinergic effects (e.g., urinary retention, glaucoma).

๐Ÿคฑ Lactation Safety

Not recommended; unknown if excreted in human milk.

๐Ÿ’Š Overdose Management

Supportive treatment; monitor for anticholinergic effects (e.g., dry mouth, blurred vision, tachycardia).

โฐ Missed Dose

Skip missed dose and take next dose at usual time; do not double dose.

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

๐Ÿ”„ Substitutes for airtio rotacap

View All

Alternative brands with exact same active ingredient (Tiotropium (18mcg)):

Medical Note: Always consult your doctor before switching medications.

๐Ÿ˜Š Was this information helpful?

Browse Medicines A-Z

Search our extensive medical database alphabetically.

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory
SaathiMed App
SaathiMed App Consult doctors & order medicines faster
Install