airtio-f instacaps - Formoterol (12mcg) + Tiotropium (18mcg) medicine

airtio-f instacaps - Uses, Price, Side Effects & Substitutes

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๐Ÿญ Glenmark Pharmaceuticals Ltd ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Jun 26, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
Dr. SaathiMed Expert Panel | Jun 26, 2026

What is airtio-f instacaps used for?

Aerotrop-F Inhaler (Formoterol + Tiotropium) is used to treat RESPIRATORY. It contains Formoterol (12mcg) + Tiotropium (18mcg), which Formoterol stimulates beta2-adrenergic receptors causing bronchodilation; Tiotro. Always consult your doctor before use. Take as prescribed.

  • Generic Name: Formoterol + Tiotropium
  • Manufacturer: Glenmark Pharmaceuticals Ltd
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

๐Ÿ’Š airtio-f instacaps Uses & Benefits

Maintenance treatment of COPD, asthma (as add-on therapy)

Off-label uses: Acute bronchospasm (not recommended), Bronchiectasis

๐Ÿ“‹ Drug Information

Generic Name(s)Formoterol + Tiotropium
Brand NameAerotrop-F Inhaler
ManufacturerGlenmark Pharmaceuticals Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassRESPIRATORY
Action ClassLong-acting beta2-agonist (LABA) + Long-acting muscarinic antagonist (LAMA)
Route of AdministrationInhalation
StorageStore at room temperature (20-25ยฐC), protect from moisture and light
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionRapidly absorbed from lungs after inhalation
DistributionDistributes to lungs and systemic circulation
Protein BindingFormoterol: 61-64%; Tiotropium: 72%
MetabolismFormoterol: Hepatic via CYP2D6, CYP2C19, CYP2C9; Tiotropium: Minimal hepatic metabolism
Half-LifeFormoterol: 10 hours; Tiotropium: 5-6 days
ExcretionFormoterol: Urine (60%) and feces (40%); Tiotropium: Urine (74%)
BioavailabilityFormoterol: ~30% (inhalation); Tiotropium: 19.5% (inhalation)
Onset of ActionFormoterol: 1-3 minutes; Tiotropium: 30 minutes
Peak Plasma TimeFormoterol: 0.5-1 hour; Tiotropium: 5 minutes
Duration of ActionFormoterol: 12 hours; Tiotropium: 24 hours

How It Works

Formoterol stimulates beta2-adrenergic receptors causing bronchodilation; Tiotropium blocks muscarinic M3 receptors causing bronchodilation

Mechanism Steps

1Formoterol binds to beta2-adrenergic receptors on airway smooth muscle
2Activates Gs protein, increasing cAMP
3cAMP activates protein kinase A

๐Ÿ’ก How to Take airtio-f instacaps

Follow your doctor's prescription exactly.

โš ๏ธ Side Effects of airtio-f instacaps

โœ… Common Side Effects

  • Dry mouth
  • Cough
  • Headache
  • Throat irritation
  • Dysphonia

๐Ÿšจ Serious Side Effects

  • Paradoxical bronchospasm
  • QTc prolongation
  • Hypokalemia
  • Hyperglycemia
  • Urinary retention

โš ๏ธ Rare Side Effects

  • Anaphylaxis
  • Angioedema
  • Atrial fibrillation
  • Glaucoma exacerbation

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Monoamine oxidase inhibitors Major Increased risk of hypertensive crisis
Tricyclic antidepressants Major Enhanced cardiovascular effects
Beta-blockers Major Antagonism of bronchodilator effect
QTc-prolonging drugs Major Increased risk of arrhythmias
Diuretics Moderate Hypokalemia risk
Corticosteroids Moderate Increased hypokalemia risk
Xanthine derivatives Moderate Additive hypokalemia
Anticholinergics Minor Additive anticholinergic effects
Sympathomimetics Minor Additive sympathomimetic effects

๐Ÿšจ Major Interactions

  • Monoamine oxidase inhibitors
  • Tricyclic antidepressants
  • Beta-blockers
  • QTc-prolonging drugs

โšก Moderate Interactions

  • Diuretics
  • Corticosteroids
  • Xanthine derivatives

โ„น๏ธ Minor Interactions

  • Anticholinergics
  • Sympathomimetics

๐Ÿฝ๏ธ Food Interactions

No significant food interactions

๐Ÿท Alcohol Interaction

No specific interaction reported

๐Ÿ›ก๏ธ Safety & Warnings

๐Ÿšซ Contraindications

Hypersensitivity to any component, severe hypersensitivity to milk proteins (lactose), acute bronchospasm

๐Ÿ“Š Monitoring Parameters

Lung function (FEV1), heart rate, QTc interval, serum potassium

๐Ÿคฑ Lactation Safety

Caution advised; limited data

๐Ÿ’Š Overdose Management

Supportive care; monitor cardiac function, electrolytes; consider beta-blockers for excessive beta-agonist effects

โฐ Missed Dose

Take as soon as remembered; skip if close to next dose; do not double dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

Dr. SaathiMed Expert Panel

MD, PhD - Pharmacology

Reviewed: Jun 26, 2026

๐Ÿ”— View Profile

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