ceftron s 1000mg/500mg injection - Ceftriaxone (1000mg) + Sulbactam (500mg) medicine

ceftron s 1000mg/500mg injection

No reviews yet
🏭 Cablin Healthcare Pvt Ltd 📦 Varies by brand 💊 Allopathy 📅 Updated: Sep 24, 2026
⚠️ Hepatotoxicity Risk 📋 Prescription Required 💊 Generic Available
Medically Reviewed
11 min read
Reviewed by
SaathiMed Expert Panel | Sep 24, 2026

What is ceftron s 1000mg/500mg injection used for?

This medicine contains Ceftriaxone (1000mg) + Sulbactam (500mg) and is used to treat ANTI INFECTIVES. Ceftriaxone inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins (PBPs);. Always consult your doctor before use.

  • Generic Name: Ceftriaxone + Sulbactam
  • Manufacturer: Cablin Healthcare Pvt Ltd
  • Form: Allopathy
  • Pregnancy Category: Category A
  • Prescription Required: Yes
💡 Did You Know? The Indian pharmaceutical market is expected to reach $130 billion by 2030.

💊 ceftron s 1000mg/500mg injection Uses & Benefits

Lower respiratory tract infections, urinary tract infections, skin and soft tissue infections, intra-abdominal infections, septicemia, meningitis, bone and joint infections

Off-label uses: Gonorrhea, Lyme disease, pelvic inflammatory disease

📋 Drug Information

Generic Name(s)Ceftriaxone + Sulbactam
Brand NameAccuzon Plus 1.5gm Injection
ManufacturerCablin Healthcare Pvt Ltd
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassANTI INFECTIVES
Action ClassCephalosporin + Beta-lactamase inhibitor
Route of AdministrationIntravenous (IV) or Intramuscular (IM)
StorageStore at 20-25°C (68-77°F); protect from light; reconstituted solution stable for 24 hours at room temperature or 3 days refrigerated
Shelf LifeAs per manufacturer

🔬 How This Medicine Works (Pharmacology)

Pharmacokinetics

AbsorptionIntramuscular administration: well absorbed; Intravenous: immediate bioavailability
DistributionWidely distributed into tissues and body fluids including CSF (when meninges inflamed)
Protein BindingCeftriaxone: 85-95%; Sulbactam: ~38%
MetabolismCeftriaxone: not metabolized; Sulbactam: minimally metabolized
Half-LifeCeftriaxone: 5.8-8.7 hours; Sulbactam: ~1 hour
ExcretionCeftriaxone: 33-67% renal, rest biliary; Sulbactam: primarily renal
BioavailabilityIM: ~100%
Onset of ActionRapid (within 30 min IV)
Peak Plasma TimeIV: end of infusion; IM: 1-2 hours
Duration of ActionApproximately 24 hours

How It Works

Ceftriaxone inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins (PBPs); Sulbactam irreversibly inhibits beta-lactamases, protecting ceftriaxone from degradation.

Mechanism Steps

1Ceftriaxone binds to penicillin-binding proteins (PBPs) on bacterial cell wall
2Inhibits transpeptidase activity, preventing cross-linking of peptidoglycan
3Activates autolytic enzymes, leading to cell lysis and death
4Sulbactam irreversibly binds to beta-lactamases, preventing hydrolysis of ceftriaxone

💡 How to Take ceftron s 1000mg/500mg injection

Follow your doctor's prescription exactly.

⚠️ Side Effects of ceftron s 1000mg/500mg injection

✅ Common Side Effects

Diarrhea
Injection site reactions
Rash
Eosinophilia

🚨 Serious Side Effects

Anaphylaxis
Stevens-Johnson syndrome
Clostridioides difficile colitis
Hemolytic anemia
Seizures

⚠️ Rare Side Effects

Pseudomembranous colitis
Biliary sludge
Interstitial nephritis
Agranulocytosis

Consult your doctor if you experience any unusual symptoms.

🔬 Drug Interactions

Drug Severity Effect
Warfarin Major Increased bleeding risk
Alcohol Major Disulfiram-like reaction
Aminoglycosides Major Increased nephrotoxicity
Probenecid Moderate Decreased renal excretion of ceftriaxone
Loop diuretics Moderate Increased nephrotoxicity risk
NSAIDs Moderate Increased bleeding risk
Live vaccines Minor Reduced vaccine efficacy
BCG Minor Reduced therapeutic effect

🚨 Major Interactions

  • Warfarin
  • Alcohol (disulfiram-like reaction)
  • Aminoglycosides (nephrotoxicity)

⚡ Moderate Interactions

  • Probenecid
  • Loop diuretics
  • NSAIDs

🍷 Alcohol Interaction

May cause disulfiram-like reaction (nausea, vomiting, headache)

🛡️ Safety & Warnings

🚫 Contraindications

Hypersensitivity to cephalosporins or beta-lactam antibiotics; history of anaphylaxis to penicillins

🤱 Lactation Safety

Excreted in breast milk in low amounts; generally considered compatible

💊 Overdose Management

Supportive care; hemodialysis may remove ceftriaxone but not sulbactam

⏰ Missed Dose

Administer as soon as remembered; if near next dose, skip missed dose; do not double dose

🔄 Substitutes for ceftron s 1000mg/500mg injection

View All

Alternative brands with exact same active ingredient:

Medical Note: Always consult your doctor before switching medications.

😊 Was this information helpful?

Browse Medicines A-Z

A B C D E F G H I J K L M N O P Q R S T U V W X Y Z
Back to Medicines Directory