brimofinet 5 mg/1.5 mg eye drop - Timolol (5mg) + Brimonidine (1.5mg) medicine

Brimofinet 5 mg/1.5 mg Eye Drop - Uses, Price, Side Effects

4.6 (18 reviews)
๐Ÿญ Calix Health Care ๐Ÿ“ฆ Varies by brand ๐Ÿ’Š Allopathy ๐Ÿ“… Updated: Aug 23, 2026
๐Ÿ“‹ Prescription Required ๐Ÿ’Š Generic Available
Medically Reviewed
SaathiMed Expert Panel | Aug 23, 2026

What is brimofinet 5 mg/1.5 mg eye drop used for?

Brimofinet 5 mg/1.5 mg Eye Drop is a combination of Timolol (a beta-blocker) and Brimonidine (an alpha-2 agonist) used to lower intraocular pressure in patients with open-angle glaucoma or ocular hypertension. It works by reducing the production of aqueous humor and increasing its outflow, thereby protecting the optic nerve from damage.

  • Generic Name: Timolol + Brimonidine
  • Manufacturer: Calix Health Care
  • Form: Allopathy
  • Pregnancy Category: C
  • Prescription Required: Yes
๐Ÿ’ก Did You Know? Over 80% of the antiretroviral drugs used globally to combat AIDS are supplied by Indian pharmaceutical companies.

๐Ÿ’Š brimofinet 5 mg/1.5 mg eye drop Uses & Benefits

Reduction of intraocular pressure in open-angle glaucoma or ocular hypertension

Off-label uses: None commonly reported

๐Ÿ“‹ Drug Information

Generic Name(s)Timolol + Brimonidine
Brand NameAbpress Eye Drop
ManufacturerCalix Health Care
Packaging / FormVaries by brand (Allopathy)
Therapeutic ClassOPHTHAL
Action ClassBeta-blocker + Alpha-2 adrenergic agonist
Route of AdministrationOphthalmic (topical)
StorageStore at 15-30ยฐC, protect from light, keep tightly closed
Shelf LifeAs per manufacturer

๐Ÿ”ฌ Pharmacology (PK/PD)

Pharmacokinetics

AbsorptionSystemic absorption occurs through the nasolacrimal duct and conjunctiva
DistributionDistributes to various tissues including the eye
Protein BindingTimolol: ~60%; Brimonidine: ~29%
MetabolismTimolol: Hepatic (CYP2D6); Brimonidine: Hepatic (aldehyde oxidase)
Half-LifeTimolol: 4-6 hours; Brimonidine: 2-3 hours
ExcretionTimolol: Renal (20% unchanged); Brimonidine: Renal (70-80% unchanged)
BioavailabilityLow systemic bioavailability due to extensive first-pass metabolism
Onset of ActionTimolol: 30 minutes; Brimonidine: 1-2 hours
Peak Plasma TimeTimolol: 1-2 hours; Brimonidine: 1-4 hours
Duration of ActionTimolol: 12-24 hours; Brimonidine: 8-12 hours

How It Works

Timolol reduces aqueous humor production by blocking beta-adrenergic receptors; Brimonidine reduces aqueous humor production and increases uveoscleral outflow by stimulating alpha-2 adrenergic receptors

Mechanism Steps

1Timolol blocks beta-1 and beta-2 adrenergic receptors in the ciliary body, reducing aqueous humor production
2Brimonidine selectively stimulates alpha-2 adrenergic receptors, decreasing aqueous humor production and increasing uveoscleral outflow
3Combined effect results in significant reduction of intraocular pressure

๐Ÿ’ก How to Take brimofinet 5 mg/1.5 mg eye drop

Follow your doctor's prescription exactly.

Dosage Timeline

๐ŸŒ… Morning โœ… โ˜€๏ธ Afternoon โŒ ๐ŸŒ† Evening โœ… ๐ŸŒ™ Night โŒ

โš ๏ธ Side Effects of brimofinet 5 mg/1.5 mg eye drop

โœ… Common Side Effects

  • Ocular burning/stinging
  • Blurred vision
  • Dry eye
  • Eye redness
  • Headache
  • Drowsiness

๐Ÿšจ Serious Side Effects

  • Bradycardia
  • Heart block
  • Bronchospasm
  • Hypotension
  • Syncope
  • Allergic reaction

โš ๏ธ Rare Side Effects

  • Depression
  • Insomnia
  • Corneal edema
  • Uveitis

Consult your doctor if you experience any unusual symptoms.

๐Ÿ”ฌ Drug Interactions

โš ๏ธ DrugSeverityEffect
Beta-blockers (oral) Moderate Additive systemic beta-blockade
MAO inhibitors Major Hypertensive crisis
Digoxin Moderate Bradycardia

๐Ÿšจ Major Interactions

  • Beta-blockers (systemic)
  • Calcium channel blockers
  • Digoxin
  • Clonidine
  • MAO inhibitors

โšก Moderate Interactions

  • Antihypertensives
  • Antidiabetic agents
  • Tricyclic antidepressants

โ„น๏ธ Minor Interactions

  • Corticosteroids
  • NSAIDs

๐Ÿฝ๏ธ Food Interactions

No significant food interactions

๐Ÿท Alcohol Interaction

May enhance hypotensive effect

๐Ÿ›ก๏ธ Safety & Warnings

Liver
Low
Kidney
Low
Heart
Moderate
Pregnancy
Category C

๐Ÿšซ Contraindications

Bronchial asthma, COPD, sinus bradycardia, second/third-degree AV block, cardiogenic shock, hypersensitivity to components

๐Ÿ“Š Monitoring Parameters

Intraocular pressure, heart rate, blood pressure, signs of ocular irritation

๐Ÿคฑ Lactation Safety

Not recommended; may be excreted in breast milk

๐Ÿ’Š Overdose Management

Supportive care; monitor heart rate and blood pressure; symptomatic treatment

โฐ Missed Dose

Apply as soon as remembered; if near next dose, skip missed dose

๐Ÿ‘จโ€โš•๏ธ Reviewed by Expert

SaathiMed Expert Panel

MD, PhD - Pharmacology

Last reviewed on: Aug 23, 2026

๐Ÿ”— View Profile

โญ User Reviews

Certified Buyer Jul 10, 2026

Good quality medicine. Satisfied with the outcome.

Happy Patient Jul 10, 2026

Good quality medicine. Satisfied with the outcome.

Trusted Reviewer Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

Happy Patient Jul 10, 2026

Found this to be a helpful product. Good results.

Certified Buyer Jul 10, 2026

This medicine was effective for me. I followed the doctor's advice.

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