Calcirol 100

Calcium (100mg) + Vitamin D3 (200IU)
Price: ₹70 - ₹110 for strip of 15 tablets
Mfr: Cadila Pharmaceuticals Ltd. | Form: Sugar-free Chewable Tablet

📋 Clinical Overview

A fixed-dose combination supplement containing elemental calcium (as calcium carbonate) and cholecalciferol (Vitamin D3). It is primarily used for the prevention and treatment of calcium and vitamin D deficiencies. Calcium is essential for bone mineralization, muscle contraction, nerve transmission, and blood coagulation. Vitamin D3 enhances intestinal absorption of calcium and phosphate, regulates bone remodeling, and supports immune function. This low-dose combination is often used for maintenance therapy or in populations with mild deficiency.

💊 Dosage & Administration

Adult: One tablet/capsule once or twice daily, as directed by physician. Typically 1-2 tablets daily. Should be taken with meals for better absorption of calcium carbonate.

Note: Take orally with or immediately after a meal to enhance calcium absorption and reduce gastric upset. Swallow whole with a full glass of water. Do not take within 2 hours of other medications (e.g., tetracyclines, bisphosphonates, levothyroxine) to avoid binding interactions. Can be taken in the morning or evening.

⚠️ Contraindications

  • Hypercalcemia (elevated serum calcium)
  • Hypervitaminosis D
  • Severe renal impairment (e.g., on dialysis) without specialist supervision
  • Known hypersensitivity to any component

🔬 Mechanism of Action

The combination works synergistically. Calcium provides the essential cation for physiological processes. Vitamin D3 (after activation to calcitriol) acts as a hormone that binds to the Vitamin D Receptor (VDR) in the intestines, bones, and kidneys. This complex regulates gene expression, increasing the synthesis of calcium-binding proteins (e.g., calbindin) in enterocytes, enhancing active transcellular calcium absorption. It also promotes renal reabsorption of calcium and phosphate and, in conjunction with PTH, stimulates bone resorption to mobilize calcium when needed.

🤕 Side Effects

  • Constipation
  • Abdominal discomfort, bloating, gas
  • Nausea

🤰 Special Populations

Pregnancy: Category A (Indian/old FDA) / Category C (US FDA for high doses). This dose is generally considered safe. Calcium and Vitamin D requirements increase during pregnancy. Use under medical supervision. Essential for fetal skeletal development.

Driving: No effect on driving ability.

🔄 Drug Interactions

Thiazide Diuretics (e.g., Hydrochlorothiazide)Reduce renal calcium excretion, increasing risk of hypercalcemia.Major
Oral Bisphosphonates (e.g., Alendronate)Calcium supplements interfere with absorption. Administer at least 2 hours apart.Moderate
LevothyroxineCalcium carbonate can decrease levothyroxine absorption. Administer 4-6 hours apart.Moderate
Oral Tetracycline/Quinolone AntibioticsCalcium binds to these drugs, reducing their absorption and efficacy.Moderate
Corticosteroids (e.g., Prednisolone)Reduce calcium absorption and increase excretion, potentially reducing efficacy.Moderate
OrlistatMay reduce absorption of fat-soluble Vitamin D3.Moderate
Cardiac Glycosides (Digoxin)Hypercalcemia potentiates digoxin toxicity, risk of arrhythmias.Major
Phenytoin, Phenobarbital, CarbamazepineInduce hepatic CYP450 enzymes, increasing metabolism of vitamin D3 to inactive metabolites, reducing efficacy.Moderate

🔁 Alternatives to Calcirol 100

Same composition (Calcium (100mg) + Vitamin D3 (200IU)), different brands:

Shelcal 100 Calcium Sandoz 100 mg + Vitamin D3 Calboral-D 100 Macalvit Plus Ostocalcium D3